简介内容:E-4177 is an angiotensin type 1 receptor antagonist. In rat adrenal cortex and liver, E4177 competitively inhibited the specific binding of 125I-[Sar1,Ile8]Ang II, with IC50 being ( +/- ) x 10(-8) M for the adrenal cortex and ( +/- ) x 10(-7) M for the liver.