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(±)-WIN 55,212 (mesylate);(±)-WIN 55,212 (mesylate)(±)-WIN 55,212 (mesylate)
 
 
  • 产品名称:(±)-WIN 55,212 (mesylate);(±)-WIN 55,212 (mesylate)(±)-WIN 55,212 (mesylate)
  • 产品型号:T38199
  • 产品产地:中国大陆
  • 采购热度:
  • 简介内容:(±)-WIN 55,212-2 is a potent aminoalkylindole cannabinoid (CB) receptor agonist with a Ki value of and nM for human recombinant central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, respectively. In contrast, the enantiomer (-)-WIN 55,212-3 acts a partial inverse agonist at CB1 (pIC50 = ) and as a competitive neutral antagonist of CB2, reversing the inverse agonism evoked by SR 144528 (pEC50 = ). (+)-WIN 55,212 (mesylate) is a mixture of the two enantiomers, (+)-WI
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(±)-WIN 55,212 (mesylate);(±)-WIN 55,212 (mesylate)(±)-WIN 55,212 (mesylate)

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名称: (±)-WIN 55,212 (mesylate);(±)-WIN 55,212 (mesylate)

描述: (±)-WIN 55,212 (mesylate)。

关键字: (±)-WIN 55,212 (mesylate) |


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原创作者:上海陶术生物科技有限公司

标签:(±)-WIN   55   212   (mesylate)   

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