简介内容：CAY17c is an inhibitor of bromodomain-containing protein 4 (BRD4; IC50= μM), as well as class I histone deacetylases (HDACs; IC50s = , , , and μM for HDAC1, -2, -3, and -8, respectively) and class IIb HDACs (IC50s = and μM for HDAC6 and HDAC10, respectively).1It is selective for these enzymes over BRD2, -3, and -T (IC50s = >20 μM for all), as well as over HDAC4, -5, -7, -9, and -11 (IC50s = >10 μM for all). CAY17c inhibits the proliferation of HCT116, SW620,
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