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Zeteletinib hemiadipateZeteletinib hemiadipateBOS-172738 hemiadipate|||DS-5010hemiadipate|||Zeteleti
 
 
  • 产品名称:Zeteletinib hemiadipateZeteletinib hemiadipateBOS-172738 hemiadipate|||DS-5010hemiadipate|||Zeteleti
  • 产品型号:T39927
  • 产品产地:中国大陆
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  • 简介内容:Zeteletinib hemiadipate (BOS-172738; DS-5010) is an orally active compound that functions as a selective inhibitor of RET kinase. It exhibits nanomolar potency against RET and a 300-fold selectivity towards VEGFR2. Notably, Zeteletinib hemiadipate demonstrates exceptional effectiveness against various forms of RET, including the wild type, RET V804M/L gatekeeper mutants, and the oncogenic RET mutation M918T. Additionally, Zeteletinib hemiadipate exerts potent antitumor effects.
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Zeteletinib hemiadipateZeteletinib hemiadipateBOS-172738 hemiadipate|||DS-5010hemiadipate|||Zeteleti

Product Introduction
Bioactivity


名称: Zeteletinib hemiadipateZeteletinib hemiadipate

描述: Zeteletinib hemiadipate。

关键字: BOS-172738 hemiadipate |DS-5010hemiadipate |Zeteletinib hemiadipate |


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原创作者:上海陶术生物科技有限公司

标签:Zeteletinib   hemiadipate   

Zeteletinib hemiadipateZeteletinib hemiadipateBOS-172738 hemiadipate|||DS-5010hemiadipate|||Zeteleti产品询价/message

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