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Rauwolscine hydrochloride;萝芙素盐酸盐Corynanthidine hydrochloride|||α-Yohimbine hydrochloride|||Isoyohimb
 
 
  • 产品名称:Rauwolscine hydrochloride;萝芙素盐酸盐Corynanthidine hydrochloride|||α-Yohimbine hydrochloride|||Isoyohimb
  • 产品型号:T4429
  • 产品产地:中国大陆
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  • 简介内容:Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes both α1- and α2-adrenergic receptors [1]. Rauwolscine hydrochloride also acts as a receptor antagonist at the serotonin 5-HT2B receptor (Ki: nM) and as a weak partial agonist at 5-HT1A (IC50: μM) [3]. The α2-adrenergic receptor has diverse physiological functions and anta
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