简介内容:B-Raf IN 7 (compound 6a) is a potent inhibitor of B-Raf with an IC 50 of nM. B-Raf IN 7 has antitumor activity against colon carcinoma cells(HCT-116), mammary gland cells(MCF-7), hepatocellular carcinoma cells(HEPG-2), human cervical carcinoma cells(Hela) and human prostate cancer cells(PC-3). The IC50 values are , , , and μM, respectively [1].