简介内容:Dynole 2 24 is an indole-based dynamin GTPase inhibitor ( IC 50 = μM for dynamin I). Dynole 2 24 is nontoxic and shows increased potency against dynamin I and II in vitro and in cells (IC (CME) = μM). Dynole 2 24 also shows selectivity for dynamin I. Dynole 2 24 is active in-cell inhibitor of clathrin-mediated endocytosis [1]. CME: Clathrin mediated endocytosis