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产品名称: CDK1-IN-4;化合物 CDK1-IN-4CDK1-IN-4
产品简介:cdk1-in-4 (10d) is a selective cdk1 inhibitor that acts on cdk1 (ic50: 44.52 nm), cdk2 (ic50: 624.93 nm) and cdk5 (ic50: 135.22 nm). cdk1-in-4 affects the cell ..产品型号:T63080 原产地:中国大陆价格: ¥0.0
产品名称: SOS1-IN-4;化合物 SOS1-IN-4SOS1-IN-4
产品简介:sos1-in-4 is a potent inhibitor of sos1 (ic50: 56 nm) and can be used in the study of kras-c12c/sos1 interactions...产品型号:T63083 原产地:中国大陆价格: ¥0.0
产品名称: (R)-IL-17 modulator 4;化合物 (R)-IL-17 modulator 4(R)-IL-17 modulator 4
产品简介:(r)-il-17 modulator 4 is the r-configured form of il-17 modulator 4 and is a prodrug of il-17 modulator 1. il-il-17 modulator 1 is a potent, orally active il-17..产品型号:T63089 原产地:中国大陆价格: ¥0.0
产品名称: EP4 receptor antagonist 2;化合物 EP4 receptor antagonist 2EP4 receptor antagonist 2
产品简介:ep4 receptor antagonist 2 (compound 2-13) is a potent agonist of the ep4 receptor (ic50: 7.8 nm) and has antitumour effects...产品型号:T63100 原产地:中国大陆价格: ¥0.0
产品名称: Estrogen receptor antagonist 4;化合物 Estrogen receptor antagonist 4Estrogen receptor antagonist 4
产品简介:estrogen receptor antagonist 4 is a potent inhibitor of the estrogen receptor (er), crucial for regulating cell growth, differentiation, and apoptosis. this com..产品型号:T63106 原产地:中国大陆价格: ¥0.0
产品名称: IRAK4-IN-18;化合物 IRAK4-IN-18IRAK4-IN-18
产品简介:irak4-in-18 is a potent inhibitor of interleukin 1 receptor-associated kinase 4 (irak4) (ic50: 15 nm). irak4-in-18 inhibits lps-induced il23 production in thp a..产品型号:T62950 原产地:中国大陆价格: ¥0.0
产品名称: IQTub4P;化合物 IQTub4PIQTub4P
产品简介:iqtub4p is a potent inhibitor of microtubules. iqtub4p exhibits cytotoxicity in hela cells (ec50: 170 nm)...产品型号:T62966 原产地:中国大陆价格: ¥0.0
产品名称: PDE4-IN-6;化合物 PDE4-IN-6PDE4-IN-6
产品简介:pde4-in-6 is a safe, potent and moderately selective inhibitor of pde4, acting on pde4b (ic50: 0.125 μm) and pde4d (ic50: 0.43 μm). pde4-in-6 is able to down-re..产品型号:T62969 原产地:中国大陆价格: ¥0.0
产品名称: FLT3/CDK4-IN-1;化合物 FLT3/CDK4-IN-1FLT3/CDK4-IN-1
产品简介:flt3/cdk4-in-1 is a highly selective, potent, orally active dual inhibitor of flt3/cdk4, acting on flt3 (ic50: 7 nm) and cdk4 (ic50: 11 nm).flt3/cdk4-in-1 has g..产品型号:T63135 原产地:中国大陆价格: ¥0.0
产品名称: Glutaminase-IN-4;化合物 Glutaminase-IN-4Glutaminase-IN-4
产品简介:glutaminase-in-4 (compound 2a) is a glutaminase (gls) inhibitor (ic50: 2.3 μm)...产品型号:T63137 原产地:中国大陆价格: ¥0.0
产品名称: RORγt modulator 4;化合物 RORγt modulator 4RORγt modulator 4
产品简介:rorγt modulator 4 is a rorγt modulator that regulates il-17a production activity in cells derived from mouse spleen...产品型号:T63124 原产地:中国大陆价格: ¥0.0
产品名称: IRAK4-IN-12;化合物 IRAK4-IN-12IRAK4-IN-12
产品简介:irak4-in-12 (compound 37) is a potent inhibitor of irak4 (ic50: 0.015 μm) with cellular pirak4 potency (ic50: 0.5 μm)...产品型号:T62989 原产地:中国大陆价格: ¥0.0
产品名称: Butein;紫铆因2’,3,4,4’-tetrahydroxy Chalcone;2’,3,4,4’-tetrahydroxy Chalcone|||紫铆因
产品简介:butein (2’,3,4,4’-tetrahydroxy chalcone), a plant polyphenol, is isolated from rhus verniciflua. it can inhibit the activation of protein tyrosine kinase, nf-κb..产品型号:T6427 原产地:中国大陆价格: ¥0.0
产品名称: BRD4-BD1-IN-2;BRD4-BD1抑制剂2BRD4-BD1-IN-2
产品简介:brd4-bd1-in-2 is a selective and potent brd4-bd1 inhibitor with an ic50 value of 2.51 ?m, which is 20-fold greater than the inhibitory activity against brd4-bd2..产品型号:T64117 原产地:中国大陆价格: ¥0.0
产品名称: FGFR4-IN-6;化合物 FGFR4-IN-6FGFR4-IN-6
产品简介:fgfr4-in-6 is a covalent, reversible fgfr4 inhibitor (ic50: 5.4 nm) that exhibits good oral pharmacokinetic properties. in a xenograft mouse model of the hep3b2..产品型号:T64015 原产地:中国大陆价格: ¥0.0
产品名称: Glyoxalase I inhibitor 4;化合物 Glyoxalase I inhibitor 4Glyoxalase I inhibitor 4
产品简介:glyoxalase i inhibitor 4 is a potent inhibitor of glyoxalase i (glo1) (ki: 10 nm)...产品型号:T64023 原产地:中国大陆价格: ¥0.0
产品名称: CYP3A4-IN-3;化合物 CYP3A4-IN-3CYP3A4-IN-3
产品简介:cyp3a4-in-3 is a specific, highly affinity cytochrome p450 3a4 (cyp3a4) (cytochrome p450 3a4 (cyp3a4)) inhibitor (ic50: 0.075 μm). cyp3a4-in-3 is an analogue of..产品型号:T64032 原产地:中国大陆价格: ¥0.0
产品名称: CYP3A4-IN-2;化合物 CYP3A4-IN-2CYP3A4-IN-2
产品简介:cyp3a4-in-2 is a specific inhibitor of cytochrome p450 3a4 (cyp3a4) (ic50: 0.055 μm). cyp3a4-in-2 is a ritonavir analogue with a more hydrophobic r2 side group ..产品型号:T64037 原产地:中国大陆价格: ¥0.0
产品名称: Trypanothione synthetase-IN-4;化合物 Trypanothione synthetase-IN-4Trypanothione synthetase-IN-4
产品简介:trypanothione synthetase-in-4 is a l. infantumtrys inhibitor whose activity is dependent on the concentration of the polyamine substrate. trypanothione syntheta..产品型号:T64056 原产地:中国大陆价格: ¥0.0
产品名称: PLK1/BRD4-IN-1;化合物 PLK1/BRD4-IN-1PLK1/BRD4-IN-1
产品简介:plk1/brd4-in-1 (9b) is an orally active dual inhibitor of plk1 (ic50: 22 nm) and brd4 (ic50: 109 nm). it has been shown to have good anti-tumour effects in vivo..产品型号:T64058 原产地:中国大陆价格: ¥0.0