联系我们
产品目录
产品展示/Products
产品名称: SP-13786;化合物SP-13786UAMC-1110;UAMC-1110|||(S)-N-[2-(2-氰基-4,4-二氟-1-吡咯烷基)-2-氧代乙基]喹啉-4-甲酰胺
产品简介:sp-13786 (uamc-1110) is an inhibitor of fibroblast activation protein (fap) (ic50 : 3.2 nm); also inhibits prolyl oligopeptidase (prep) ( ic50 : 1.8 μm)...产品型号:T7890 原产地:中国大陆价格: ¥0.0
产品名称: AD4;化合物 AD4AD4
产品简介:ad4, an artemisinin derivative functioning as a proteolytic targeting chimera (protac) for pclaf, effectively degrades pclaf in rs4;11 cells with an ic50 of 0.6..产品型号:T78805 原产地:中国大陆价格: ¥0.0
产品名称: NDNA4;化合物 NDNA4NDNA4
产品简介:ndna4 (compound 17) is a selective hsp90α inhibitor (ic50: 0.34 μm), characterized by its permanent charge and low membrane permeability. it exhibits minimal cy..产品型号:T78808 原产地:中国大陆价格: ¥0.0
产品名称: Anti-osteoporosis agent-4;化合物 Anti-osteoporosis agent-4Anti-osteoporosis agent-4
产品简介:anti-osteoporosis agent-4 (compound 11h) suppresses the differentiation of primary osteoclasts and attenuates rankl-induced osteoclastogenesis. it effectively i..产品型号:T78816 原产地:中国大陆价格: ¥0.0
产品名称: D4R agonist-1;D4R激动剂1D4R agonist-1
产品简介:d4r agonist-1 is a selective and potent d4r partial agonist (ki:2.2 nm).d4r agonist-1 can be used to study neurological diseases...产品型号:T78825 原产地:中国大陆价格: ¥0.0
产品名称: CYP51/PD-L1-IN-4;化合物 CYP51/PD-L1-IN-4CYP51/PD-L1-IN-4
产品简介:cyp51/pd-l1-in-4 (compound 14a-2) is a potent dual-target inhibitor of cyp51/pd-l1, displaying ic50 values of 0.17 and 0.021 μm, respectively. this compound dem..产品型号:T78902 原产地:中国大陆价格: ¥0.0
产品名称: IRAK4-IN-24;化合物 IRAK4-IN-24IRAK4-IN-24
产品简介:irak4-in-24 (compound 16), a potent irak4 inhibitor, exhibits high clearance (cl) and low oral bioavailability. it is utilized in research pertaining to inflamm..产品型号:T78744 原产地:中国大陆价格: ¥0.0
产品名称: DiPT-4;化合物 DiPT-4DiPT-4
产品简介:dipt-4, a dual top1/parp1 inhibitor, effectively induces dna double-strand breaks (dsbs), cell cycle arrest, and apoptosis in cancer cells, with potential to ci..产品型号:T78747 原产地:中国大陆价格: ¥0.0
产品名称: Aurora Kinases-IN-4;化合物 Aurora Kinases-IN-4Aurora Kinases-IN-4
产品简介:aurora kinases-in-4 (compound 11c) is a covalent, atp-competitive inhibitor of aurora kinase a with an ic50 value of 1.7 nm. it demonstrates cell proliferation ..产品型号:T78753 原产地:中国大陆价格: ¥0.0
产品名称: VEGFR2-IN-4;化合物 VEGFR2-IN-4VEGFR2-IN-4
产品简介:vegfr2-in-4 (compound 25) is a potent, selective inhibitor of the vegfr2 kinase, exhibiting a gi50 of 0.7 nm and demonstrating anti-angiogenic effects. it is ut..产品型号:T78759 原产地:中国大陆价格: ¥0.0
产品名称: MMP13-IN-4;化合物 MMP13-IN-4MMP13-IN-4
产品简介:mmp13-in-4 (compound 13) is a potent, selective mmp-13 inhibitor with an ic50 of 14.6 μm, implicated in the pathology of osteoarthritis (oa) [1]...产品型号:T78774 原产地:中国大陆价格: ¥0.0
产品名称: Multi-kinase-IN-4;化合物 Multi-kinase-IN-4Multi-kinase-IN-4
产品简介:multi-kinase-in-4 (compound 5d) is a multi-targeted kinase inhibitor active against vegfr2, egfr, her2, and cdk2, with respective ic50 values of 0.33, 0.22, 0.1..产品型号:T78792 原产地:中国大陆价格: ¥0.0
产品名称: IOX4;化合物IOX4IOX4
产品简介:iox4 is a potent phd2 inhibitor (ic50 = 1.6 nm)..产品型号:T7880 原产地:中国大陆价格: ¥0.0
产品名称: p38 Kinase inhibitor 4;化合物 p38 Kinase inhibitor 4p38 Kinase inhibitor 4
产品简介:compound 135, also known as p38 kinase inhibitor 4, is a potent inhibitor of p38 [1]...产品型号:T79028 原产地:中国大陆价格: ¥0.0
产品名称: Tazarotenic acid;化合物AGN-190299AGN-190299;6-[2-(3,4-二氢-4,4-二甲基-2H-1-苯并噻喃-6-基)乙炔基]-3-吡啶甲酸|||AGN-190299
产品简介:tazarotenic acid (agn-190299) is a retinoid prodrug which is converted to its active form..产品型号:T7894 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD3/BRD4-L degrader-2;化合物 PROTAC BRD3/BRD4-L degrader-2PROTAC BRD3/BRD4-L degrader-2
产品简介:protac brd3/brd4-l degrader-2, a protac molecule, selectively degrades cellular brd3 and brd4-l with k i values of 16.91 and 2.8 nm, respectively, and exhibits ..产品型号:T78956 原产地:中国大陆价格: ¥0.0
产品名称: FABP4-IN-2;化合物 FABP4-IN-2FABP4-IN-2
产品简介:fabp4-in-2 (compd 10g), a selective and orally active fabp4 inhibitor, exhibits k i values of 0.51 μm for fabp4 and 33.01 μm for fabp3, demonstrating its specif..产品型号:T78960 原产地:中国大陆价格: ¥0.0
产品名称: BRD4 Inhibitor-28;化合物 BRD4 Inhibitor-28BRD4 Inhibitor-28
产品简介:brd4 inhibitor-28 (compound 18), an orally active molecule, selectively inhibits the bromodomains of brd4 (brd4-bd1 and brd4-bd2) with ic50 values of 15 and 55 ..产品型号:T78851 原产地:中国大陆价格: ¥0.0
产品名称: AMPA receptor modulator-4;化合物 AMPA receptor modulator-4AMPA receptor modulator-4
产品简介:ampa receptor modulator-4, a 3,4-dihydro-2h-1,2,4-benzothiadiazine 1,1-dioxide (btd), serves as an orally active positive allosteric modulator of the ampa recep..产品型号:T78971 原产地:中国大陆价格: ¥0.0
产品名称: IRAK4-IN-28;化合物 IRAK4-IN-28IRAK4-IN-28
产品简介:irak4-in-28 (compound 42), an orally-active irak4 inhibitor (ic50=8.9 nm), exhibits strong binding affinity with a kd of 0.58 nm for the target enzyme. it is ut..产品型号:T79337 原产地:中国大陆价格: ¥0.0