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产品目录

产品展示/Products

  • 1-(2-Pyridyl)piperazine1-(2-Pyridyl)piperazine,NSC13778,

    产品名称: 1-(2-Pyridyl)piperazine1-(2-Pyridyl)piperazine,NSC13778,

    产品简介:1-(2-pyridyl)piperazine is a selective α2-adrenoceptor antagonists. 1-(2-pyridyl)piperazine shows sympatholytic activity. 1-(2-pyridyl)piperazine is also a meta..

    产品型号:T5105 原产地:美洲价格: ¥0.0

  • BTSA1BTSA1

    产品名称: BTSA1BTSA1

    产品简介:btsa1 is a bax activator that binds with high affinity and specificity to the n-terminal activation site and induces conformational changes to bax leading to ba..

    产品型号:T5104 原产地:美洲价格: ¥0.0

  • NMDAR antagonist 1NMDAR antagonist 1

    产品名称: NMDAR antagonist 1NMDAR antagonist 1

    产品简介:na..

    产品型号:T5522 原产地:美洲价格: ¥0.0

  • BivalirudinBivalirudin,Hirulog-1,BG-8967

    产品名称: BivalirudinBivalirudin,Hirulog-1,BG-8967

    产品简介:bivalirudin is a reversible inhibitor of α- and ζ-thrombin (kis = 2.56 and 1.84 nm, respectively), enzymes that exhibit high fibrinogen-clotting activities...

    产品型号:T5519 原产地:美洲价格: ¥0.0

  • diABZI STING agonist-1 trihydrochloridediABZI STING agonist-1 trihydrochloride

    产品名称: diABZI STING agonist-1 trihydrochloridediABZI STING agonist-1 trihydrochloride

    产品简介:diabzi sting agonist-1 (trihydrochloride) is stimulator of interferon genes (sting) receptor agonist...

    产品型号:T5516 原产地:美洲价格: ¥0.0

  • OSU-T315 (1,5-regioisomer)OSU-T315 (1,5-regioisomer),ILK-IN-2,

    产品名称: OSU-T315 (1,5-regioisomer)OSU-T315 (1,5-regioisomer),ILK-IN-2,

    产品简介:osu-t315 (1,5-regioisomer) is a ilk inhibitor...

    产品型号:T5485 原产地:美洲价格: ¥0.0

  • TRi-1TRi-1

    产品名称: TRi-1TRi-1

    产品简介:tri-1 is irreversible inhibitor of cytosolic thioredoxin reductase 1 (txnrd1), with an ic50 of 12 nm. tri-1 has little mitochondrial toxicity for anticancer the..

    产品型号:T5481 原产地:美洲价格: ¥0.0

  • mAChr-in-1mAChr-in-1

    产品名称: mAChr-in-1mAChr-in-1

    产品简介:machr-in-1 is muscarinic cholinergic receptor(machr) antagonist (ic50=17 nm)...

    产品型号:T5476 原产地:美洲价格: ¥0.0

  • GSK1940029GSK1940029,SCD inhibitor 1,

    产品名称: GSK1940029GSK1940029,SCD inhibitor 1,

    产品简介:gsk1940029 is a stearoyl-coa desaturase (scd) inhibitor...

    产品型号:T5427 原产地:美洲价格: ¥0.0

  • DDR1-IN-2DDR1-IN-2,DDR1 inhibitor 7rh,

    产品名称: DDR1-IN-2DDR1-IN-2,DDR1 inhibitor 7rh,

    产品简介:ddr1-in-2 (ddr1 inhibitor 7rh) is a potent, selective, atp-competitive discoidin domain receptor 1 (ddr1) inhibitor (ic50: 6.8 nm in cell-free kinase assays)...

    产品型号:T5402 原产地:美洲价格: ¥0.0

  • GSK2983559GSK2983559,RIPK2 inhibitor 1,RIPK2-IN-1

    产品名称: GSK2983559GSK2983559,RIPK2 inhibitor 1,RIPK2-IN-1

    产品简介:gsk 2983559 (rip2 kinase inhibitor 1) is a potent, selective receptor-interacting protein-2 (rip2) kinase inhibitor...

    产品型号:T5401 原产地:美洲价格: ¥0.0

  • CK1-IN-1CK1-IN-1,PUN51207,

    产品名称: CK1-IN-1CK1-IN-1,PUN51207,

    产品简介:ck1-in-1, compound 1c reported in patent wo2015119579a1, is a casein kinase 1 (ck1) inhibitor. it has ic50s of 15 nm, 16 nm, 73 nm for ck1δ, and ck1ε, p38σ mapk..

    产品型号:T5393 原产地:美洲价格: ¥0.0

  • ERK5-IN-1ERK5-IN-1

    产品名称: ERK5-IN-1ERK5-IN-1

    产品简介:erk5-in-1 is a potent erk5 inhibitor (ic50: 87 nm). it also inhibits lrrk2[g2019s] (ic50: 26 nm)...

    产品型号:T5184 原产地:美洲价格: ¥0.0

  • AUT1AUT1

    产品名称: AUT1AUT1

    产品简介:aut1 (aut-1) is a novel specific modulator of kv3 channels (ec50: 4.7 and 4.9 um for kv3.1b and kv3.2a)...

    产品型号:T5183 原产地:美洲价格: ¥0.0

  • SGC-GAK-1SGC-GAK-1

    产品名称: SGC-GAK-1SGC-GAK-1

    产品简介:sgc-gak-1 is a selective cyclin g-associated kinase (gak) inhibitor (ki: 3.1 nm)...

    产品型号:T5169 原产地:美洲价格: ¥0.0

  • K-Ras-IN-1K-Ras-IN-1,K-Ras-IN-1,

    产品名称: K-Ras-IN-1K-Ras-IN-1,K-Ras-IN-1,

    产品简介:k-ras-in-1 is a k-ras inhibitor...

    产品型号:T5469 原产地:美洲价格: ¥0.0

  • Tyrosine kinase-IN-1Tyrosine kinase-IN-1

    产品名称: Tyrosine kinase-IN-1Tyrosine kinase-IN-1

    产品简介:tyrosine kinase-in-1 is a multi-targeted tyrosine kinase inhibitor(kdr, flt-1, fgfr1 and pdgfrα with ic50s of 4nm, 20nm, 4nm, 2 nm ,respectively)..

    产品型号:T5466 原产地:美洲价格: ¥0.0

  • Ehp-inhibitor-1Ehp-inhibitor-1

    产品名称: Ehp-inhibitor-1Ehp-inhibitor-1

    产品简介:ehp-inhibitor-1 is an eph family tyrosine kinase inhibitor targeting eph receptors...

    产品型号:T5451 原产地:美洲价格: ¥0.0

  • JQ-1 carboxylic acidJQ-1 carboxylic acid

    产品名称: JQ-1 carboxylic acidJQ-1 carboxylic acid

    产品简介:jq-1 carboxylic acid is a cell-permeable brd4 inhibitor with ic50s of 77 nm for brd4(1) and 33 nm for brd4(2)..

    产品型号:T5443 原产地:美洲价格: ¥0.0

  • MZ1MZ1,MZ 1,

    产品名称: MZ1MZ1,MZ 1,

    产品简介:mz 1 is a brd4 protein degrader based on protac technology...

    产品型号:T5436 原产地:美洲价格: ¥0.0

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