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产品名称: hCYP3A4-IN-1;化合物 hCYP3A4-IN-1hCYP3A4-IN-1
产品简介:hcyp3a4-in-1 (compound c6) is a potent, orally active inhibitor of hcyp3a4, exhibiting ic50 values of 43.93 nm in human liver microsomes (hlms) and 153.00 nm in..产品型号:T79343 原产地:中国大陆价格: ¥0.0
产品名称: 2-Aminothiazol-4-acetic acid;2-氨基-4-噻唑乙酸2-Aminothiazol-4-acetic acid
产品简介:2-aminothiazol-4-acetic acid acts by inhibiting the activity of certain enzymes and proteins related to inflammation, tumor growth and oxidative stress, and has..产品型号:T7935 原产地:中国大陆价格: ¥0.0
产品名称: PRMT4-IN-3;化合物 PRMT4-IN-3PRMT4-IN-3
产品简介:prmt4-in-3 (compound 56) serves as a potent class i protein arginine methyltransferase (prmt) inhibitor, specifically targeting prmt4 with an ic50 value of 37 n..产品型号:T79355 原产地:中国大陆价格: ¥0.0
产品名称: hCA/VEGFR-2-IN-4;化合物 hCA/VEGFR-2-IN-4hCA/VEGFR-2-IN-4
产品简介:hca/vegfr-2-in-4 (compound 15b), an indolinylbenzenesulfonamide, serves as a potential dual inhibitor targeting cancer-related human carbonic anhydrases hca ix/..产品型号:T79591 原产地:中国大陆价格: ¥0.0
产品名称: COX-1/2-IN-4;化合物 COX-1/2-IN-4COX-1/2-IN-4
产品简介:cox-1/2-in-4 (compound 2b) is a dual cox-1 and cox-2 inhibitor with respective ic50 values of 0.239 μm for cox-1 and 0.191 μm for cox-2. additionally, it demons..产品型号:T79592 原产地:中国大陆价格: ¥0.0
产品名称: NSD2-IN-4;化合物 NSD2-IN-4NSD2-IN-4
产品简介:nsd2-in-4 is a potent, selective inhibitor of the nsd2-set domain, showing promise for the treatment of diseases related to nsd2 [1]...产品型号:T79617 原产地:中国大陆价格: ¥0.0
产品名称: M3/PDE4 modulator-1;化合物 M3/PDE4 modulator-1M3/PDE4 modulator-1
产品简介:m3/pde4 modulator-1 (compound 10f) serves as a bifunctional entity functioning both as an m3 machr antagonist and a pde4 inhibitor. when administered intravenou..产品型号:T79618 原产地:中国大陆价格: ¥0.0
产品名称: Mtb-IN-4;化合物 Mtb-IN-4Mtb-IN-4
产品简介:mtb-in-4 (compound 17h) is a non-toxic isoxazole that exhibits anti-mycobacterium tuberculosis (mtb) activity, with an ic50 value of 0.70 μm. it impedes mtb res..产品型号:T79559 原产地:中国大陆价格: ¥0.0
产品名称: 22-(4′-py)-JA;化合物 22-(4′-py)-JA22-(4′-Pyridinecarbonyl) jorunnamycin A;22-(4′-Pyridinecarbonyl) joru
产品简介:22-(4′-py)-ja, a semisynthetic derivative of junamycin a isolated from the thai blue sponge (xestospongia sp.), exhibits antimetastatic properties by inhibiting..产品型号:T79560 原产地:中国大陆价格: ¥0.0
产品名称: Sirt1/2-IN-4;化合物 Sirt1/2-IN-4Sirt1/2-IN-4
产品简介:sirt1/2-in-4 (compound ps3) is a potent triple inhibitor of sirt1, sirt2, and sirt3, exhibiting ic50 values of 1.2 μm (sirt1), 1.9 μm (sirt2), and 18.6 μm (sirt..产品型号:T79565 原产地:中国大陆价格: ¥0.0
产品名称: COX-2/15-LOX-IN-4;化合物 COX-2/15-LOX-IN-4COX-2/15-LOX-IN-4
产品简介:cox-2/15-lox-in-4 (compound 5i) is a dual inhibitor with ic50 values of 0.075 μm for cox-2 and 1.97 μm for 15-lox. it inhibits lps-induced production of pro-inf..产品型号:T79362 原产地:中国大陆价格: ¥0.0
产品名称: Antiangiogenic agent 4;化合物 Antiangiogenic agent 4Antiangiogenic agent 4
产品简介:compound 3b, an antiangiogenic agent, inhibits akt phosphorylation in both hff and huvec cells and is utilized in cancer research [1]...产品型号:T79364 原产地:中国大陆价格: ¥0.0
产品名称: LTB4-IN-2;化合物 LTB4-IN-2LTB4-IN-2
产品简介:ltb4-in-2 (compound 6x) is a selective inhibitor of leukotriene b4 (ltb4), acting by specifically targeting the 5-lipoxygenase-activating protein (flap) with an..产品型号:T79389 原产地:中国大陆价格: ¥0.0
产品名称: Fingolimod;芬戈莫德FTY-720A|||FTY-720;2-氨基-2-[2-(4-辛基苯基)乙基]-1,3-丙二醇|||FTY-720A|||FTY-720|||芬戈莫德
产品简介:fingolimod (fty-720a) is an antagonist of sphingosine 1-phosphate (s1p) (ic50 of 0.033 nm in k562 and nk cells)...产品型号:T7939 原产地:中国大陆价格: ¥0.0
产品名称: eIF4E-IN-5;化合物 eIF4E-IN-5eIF4E-IN-5
产品简介:eif4e-in-5 (compound 6n) is a cell-permeable eif4e inhibitor that binds to capped mrna, thereby inhibiting cap-dependent translation [1]...产品型号:T79525 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2 nsp14-IN-4;化合物 SARS-CoV-2 nsp14-IN-4SARS-CoV-2 nsp14-IN-4
产品简介:sars-cov-2 nsp14-in-4 (compound 12q), a non-cytotoxic and cell-permeable inhibitor of sars-cov-2 nsp14 methyltransferase (ic50 = 19 nm), is employed in covid-19..产品型号:T79526 原产地:中国大陆价格: ¥0.0
产品名称: PDE4-IN-13;化合物 PDE4-IN-13PDE4-IN-13
产品简介:pde4-in-13 is a phosphodiesterase 4 (pde4) inhibitor exhibiting anti-inflammatory and antioxidant activities, with an half maximal inhibitory concentration (ic5..产品型号:T79538 原产地:中国大陆价格: ¥0.0
产品名称: Neutrophil elastase inhibitor 4;化合物 Neutrophil elastase inhibitor 4Neutrophil elastase inhibitor 4
产品简介:neutrophil elastase inhibitor 4 (compound 4f) is a competitive inhibitor of human neutrophil elastase (hne) with ic50 of 42.30 nm and ki of 8.04 nm. it prompts ..产品型号:T79397 原产地:中国大陆价格: ¥0.0
产品名称: α-Amylase/α-Glucosidase-IN-4;化合物 α-Amylase/α-Glucosidase-IN-4α-Amylase/α-Glucosidase-IN-4
产品简介:α-amylase/α-glucosidase-in-4 (compound 5), a dual inhibitor targeting α-amylase (amylases) and α-glucosidase (glucosidase), exhibits potent inhibition with ic50..产品型号:T79402 原产地:中国大陆价格: ¥0.0
产品名称: IRAK4-IN-27;化合物 IRAK4-IN-27IRAK4-IN-27
产品简介:irak4-in-27 (compound 22) is a potent and selective irak4 inhibitor, demonstrating an ic50 of 8.7 nm. it effectively suppresses cell growth and induces apoptosi..产品型号:T79485 原产地:中国大陆价格: ¥0.0