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产品名称: Calcium Channel antagonist 4;Calcium Channel拮抗剂4Calcium Channel antagonist 4
产品简介:calcium channel antagonist 4 is a voltage-gated calcium channel inhibitor (ic50 : 5-20 μm)...产品型号:T77711 原产地:中国大陆价格: ¥0.0
产品名称: Calcium Channel antagonist 3;Calcium Channe拮抗剂3Calcium Channel antagonist 3
产品简介:calcium channel antagonist 3 is a voltage-gated calcium channel inhibitor (ic50 : 5-20 μm)...产品型号:T77712 原产地:中国大陆价格: ¥0.0
产品名称: H4R antagonist 3;H4R拮抗剂3H4R antagonist 3
产品简介:h4r antagonist 3 is a novel histamine-4 receptor (h4r) antagonist with an ec50 <10 mm.h4r antagonist 3 has potential inflammatory activity for the study of auto..产品型号:T77715 原产地:中国大陆价格: ¥0.0
产品名称: D3R/MOR antagonist 1;化合物 D3R/MOR antagonist 1D3R/MOR antagonist 1
产品简介:compound 114 (d3r/mor antagonist 1) exhibits dual antagonistic activity at dopamine d3 receptors (d3r) and mu-opioid receptors (mor), with k i values of 46.5 nm..产品型号:T78778 原产地:中国大陆价格: ¥0.0
产品名称: D3R/MOR antagonist 2;化合物 D3R/MOR antagonist 2D3R/MOR antagonist 2
产品简介:compound 121, a d3r/mor antagonist with k i values of 361 nm and 85.2 nm for d3r and mor respectively, has the potential for analgesic effects through mor parti..产品型号:T78779 原产地:中国大陆价格: ¥0.0
产品名称: CaSR antagonist-1;化合物 CaSR antagonist-1CaSR antagonist-1
产品简介:casr antagonist-1 is a potent inhibitor of the calcium-sensing receptor (casr) with an inhibitory concentration (ic50) of 50 nm, suitable for the investigation ..产品型号:T79023 原产地:中国大陆价格: ¥0.0
产品名称: A1/A3 AR antagonist 3;化合物 A1/A3 AR antagonist 3A1/A3 AR antagonist 3
产品简介:a1/a3 ar antagonist 3 is a dual a1r/a3r antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful in th..产品型号:T79027 原产地:中国大陆价格: ¥0.0
产品名称: ET receptor antagonist 1;化合物 ET receptor antagonist 1ET receptor antagonist 1
产品简介:et receptor antagonist 1 (compound 16h), with an ic50 value of 0.18 nm, is an orally active agent that can be utilized for pulmonary arterial hypertension (pah)..产品型号:T79573 原产地:中国大陆价格: ¥0.0
产品名称: ET receptor antagonist 2;化合物 ET receptor antagonist 2ET receptor antagonist 2
产品简介:et receptor antagonist 2 (compound 16j) is an orally active et receptor antagonist with an ic50 of 0.22 nm, suitable for pulmonary arterial hypertension (pah) r..产品型号:T79574 原产地:中国大陆价格: ¥0.0
产品名称: ET receptor antagonist 3;化合物 ET receptor antagonist 3ET receptor antagonist 3
产品简介:"et receptor antagonist 3 (compound 17d) is an orally active et receptor antagonist with an ic50 of 0.26 nm, utilized for pulmonary arterial hypertension (pah) ..产品型号:T79575 原产地:中国大陆价格: ¥0.0
产品名称: NMDA receptor antagonist 7;化合物 NMDA receptor antagonist 7NMDA receptor antagonist 7
产品简介:compound (s)-10a, a glun2b subunit-selective nmda receptor antagonist, exhibits a k i of 93 nm and an ic 50 of 72 nm. it is potentially useful for research into..产品型号:T79374 原产地:中国大陆价格: ¥0.0
产品名称: NMDA receptor antagonist 8;化合物 NMDA receptor antagonist 8NMDA receptor antagonist 8
产品简介:compound (r)-10a, an nmda receptor antagonist, exhibits selectivity for the glun2b subunit, possessing a ki of 265 nm and an ic50 of 62 nm. this compound is uti..产品型号:T79375 原产地:中国大陆价格: ¥0.0
产品名称: BLT2 antagonist-1;化合物 BLT2 antagonist-1BLT2 antagonist-1
产品简介:blt2 antagonist-1 (compound 15b) is a selective inhibitor of the blt2 receptor, impeding the chemotaxis of cho-blt2 cells at an ic50 of 224 nm, while not affect..产品型号:T79418 原产地:中国大陆价格: ¥0.0
产品名称: RORγ antagonist 1;化合物 RORγ antagonist 1RORγ antagonist 1
产品简介:rorγ antagonist 1 (compound 22), a potent derivative of betulinic acid, acts as an antagonist to rorγ with a dissociation constant (k d) of 0.18 μm. it demonstr..产品型号:T79464 原产地:中国大陆价格: ¥0.0
产品名称: Mu opioid receptor antagonist 7;化合物 Mu opioid receptor antagonist 7Mu opioid receptor antagonist 7
产品简介:compound 24, also known as mu opioid receptor antagonist 7, is a potent, centrally-acting ?-opioid receptor (?or) antagonist with an inhibitory concentration (i..产品型号:T79431 原产地:中国大陆价格: ¥0.0
产品名称: P2X7 receptor antagonist-4;化合物 P2X7 receptor antagonist-4P2X7 receptor antagonist-4
产品简介:compound 14a (p2x7 receptor antagonist-4) is a p2x7r antagonist with ic50 values of 64.7 nm in humans and 10.1 nm in mice. it inhibits the activation of the nlr..产品型号:T81579 原产地:中国大陆价格: ¥0.0
产品名称: GPR34 receptor antagonist 3;化合物 GPR34 receptor antagonist 3GPR34 receptor antagonist 3
产品简介:compound 5e, a gpr34 receptor antagonist, exhibits selective inhibition of lysophosphatidylserine-induced erk1/2 phosphorylation in a dose-dependent manner, dem..产品型号:T82264 原产地:中国大陆价格: ¥0.0
产品名称: GABA receptor Antagonist 1;化合物 GABA receptor Antagonist 1GABA receptor Antagonist 1
产品简介:gaba receptor antagonist 1 (compound 7w) effectively inhibits the px rdl1 gabar at an ic50 of 7.08 nmol/l and demonstrates insecticidal efficacy against p. xylo..产品型号:T82357 原产地:中国大陆价格: ¥0.0
产品名称: Galectin-3 antagonist 2;化合物 Galectin-3 antagonist 2Galectin-3 antagonist 2
产品简介:galectin-3, a β-galactoside-specific carbohydrate recognition protein (lectin), facilitates the migration of b-cell precursor acute lymphoblastic leukemia (bcp-..产品型号:T74538 原产地:中国大陆价格: ¥0.0
产品名称: A2A/A3u00A0AR antagonist-1;化合物 A2A/A3u00A0AR antagonist-1A2A/A3u00A0AR antagonist-1
产品简介:compound 23, designated as a2a/a3 ar antagonist-1, is a dual fluorescent ligand targeting a2a and a3 adenosine receptors (ar), exhibiting dissociation constants..产品型号:T74606 原产地:中国大陆价格: ¥0.0