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产品名称: NMDAinhibit,iGluR,Inhibitor,NMDA,Ionotropic glutamate receptors,Endogenous Metabolite
产品简介:n-methyl-d-aspartic acid is an amino acid that, as the d-isomer, is the defining agonist for the nmda receptor subtype of glutamate receptors...产品型号:T6608 原产地:中国大陆价格: ¥0.0
产品名称: OSBPL7-IN-1OSBPL7,orally active,ABCA1,OSBPL7 IN 1,Inhibitor,OSBPL-7-IN-1,OSBPL7IN1,inhibit
产品简介:osbpl7-in-1 is an orally active inhibitor of oxysterol binding protein like 7 (osbpl7). osbpl7-in-1 promotes an increase of abca1 at the plasma membrane without..产品型号:T9565 原产地:中国大陆价格: ¥0.0
产品名称: YO-01027二苯并氮卓;DBZ;gamma-Secretase Inhibitor XX;Dibenzazepine
产品简介:yo-01027 is a potent γ-secretase inhibitor...产品型号:T6135 原产地:中国大陆价格: ¥0.0
产品名称: TCS 359FLT3 Inhibitor
产品简介:tcs 359 is a potent flt3 inhibitor with ic50 of 42 nm...产品型号:T6138 原产地:中国大陆价格: ¥0.0
产品名称: IMD-0354IMD 0354;IKK2 Inhibitor V
产品简介:imd-0354 is an ikkβ inhibitor and inhibits iκbα phosphorylation in nf-κb pathway...产品型号:T6141 原产地:中国大陆价格: ¥0.0
产品名称: ZM39923 hydrochlorideZM 39923 HCl;JAK3 Inhibitor IV
产品简介:zm 39923 hcl is an jak1/3 inhibitor with pic50 of 4.4/7.1, almost no activity to jak2 and modestly potent to egfr; also found to be sensitive to transglutaminas..产品型号:T6145 原产地:中国大陆价格: ¥0.0
产品名称: IKK 16IKK Inhibitor VII;IKK16;IKK-16
产品简介:ikk-16 (ikk inhibitor vii) is a selective iκb kinase (ikk) inhibitor for ikk-2, ikk complex and ikk-1 with ic50 of 40 nm, 70 nm and 200 nm, respectively...产品型号:T6176 原产地:中国大陆价格: ¥0.0
产品名称: RepSoxALK5 Inhibitor II;SJN 2511;E-616452
产品简介:repsox is a potent and selective of the tgfβr-1/alk5 inhibitor...产品型号:T6337 原产地:中国大陆价格: ¥0.0
产品名称: NSC 23766 trihydrochlorideNSC 23766;Rac1 Inhibitor
产品简介:nsc 23766 is an inhibitor of rac gtpase targeting rac activation by gefs (ic50: ~50 μm); no inhibitory for the closely related targets, rhoa or cdc42...产品型号:T6342 原产地:中国大陆价格: ¥0.0
产品名称: 4μ8CIRE1 Inhibitor III
产品简介:4μ8c(ic50=76 nm) is an effective and specific ire1 rnase inhibitor...产品型号:T6363 原产地:中国大陆价格: ¥0.0
产品名称: A 922500(1R,2R)-2-[[4-[[(苯基氨基)羰基]氨基][1,1-联苯]-4-基]甲酰基]环戊烷羧酸;DGAT-1 Inhibitor 4a;A922500
产品简介:a922500 is an inhibitor for human and mouse dgat-1 with ic50 of 7 nm and 24 nm, respectively, good selectivity over related acyltransferases, herg, and a panel ..产品型号:T6365 原产地:中国大陆价格: ¥0.0
产品名称: H-89 dihydrochlorideH 89 2HCl;5-Isoquinolinesulfonamide;Protein kinase inhibitor H-89 dihydrochlorid
产品简介:h 89 is a potent inhibitor of protein kinase a (pka; ic50: 0.14 μm, ki: 48 nm)...产品型号:T6250 原产地:中国大陆价格: ¥0.0
产品名称: TDZD-8TDZD8;GSK-3β Inhibitor I;TDZD 8;NP 01139
产品简介:tdzd-8 is an inhibitor of gsk-3β, with an ic50 of 2 μm; minimal inhibitory effect observed on cdk1, casein kinase ii, pka and pkc...产品型号:T6187 原产地:中国大陆价格: ¥0.0
产品名称: StatticSTAT3 Inhibitor V
产品简介:stattic is a small molecule inhibitor of stat3. it selectively inhibits stat3 activation, dimerization, and nuclear translocation (ic50: 5.1 μm)...产品型号:T6308 原产地:中国大陆价格: ¥0.0
产品名称: BMS-345541BMS345541;IKK Inhibitor III;BMS 345541;BMS-345541 free base
产品简介:bms-345541 is a highly selective inhibitor of the catalytic subunits of ikk-2 and ikk-1 with ic50 of 0.3 μm and 4 μm, respectively...产品型号:T6326 原产地:中国大陆价格: ¥0.0
产品名称: MM-102MM102;MM 102;HMTase Inhibitor IX
产品简介:mm-102 is a high-affinity peptidomimetic mll1 inhibitor with ic50 of 0.4 μm...产品型号:T6333 原产地:中国大陆价格: ¥0.0
产品名称: Tie2 kinase inhibitor 1Tie2 kinase inhibitor
产品简介:tie2 kinase inhibitor, an optimized compound of sb-203580, is selective to tie2 with ic50 of 0.25 μm, which is 200-fold more effective than p38...产品型号:T6335 原产地:中国大陆价格: ¥0.0
产品名称: PaltusotinePaltusotine,Somatostatin Receptor,CRN-00808,CRN 00808,Inhibitor,IGF-1,orally,CRN00808,SST
产品简介:paltusotine is a nonpeptide, small molecule somatostatin type 2 (sst2) receptor agonist with high oral bioavailability. paltusotine maintains gh and igf-1 level..产品型号:T9692 原产地:中国大陆价格: ¥0.0
产品名称: Creatine-d3 hydrateEndogenous Metabolite,inhibit,Inhibitor,Creatine d3 hydrate,Creatine-d-3 hydrate,
产品简介:creatine d3 hydrate is a deuterium labeled creatine hydrate. under physiological and in pathological conditions, creatine hydrate is pivotal in energy metabolis..产品型号:T9087 原产地:中国大陆价格: ¥0.0
产品名称: XL177AMCF7,XL177A,Deubiquitinase,inhibit,Inhibitor,cancer,XL-177A,DUBs,p53,USP7
产品简介:xl177a is a selective irreversible usp7 inhibitor(ic50 : 0.34 nm). xl177a elicits cancer cell killing through a p53-dependent mechanism...产品型号:T9122 原产地:中国大陆价格: ¥0.0