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产品名称: Opiranserin hydrochlorideVVZ 149,analgesic,postoperative,VVZ-149,5-hydroxytryptamine Receptor,5-HT R
产品简介:opiranserin (vvz-149) hydrochloride is a dual antagonist of glycine transporter type 2 (glyt2) and serotonin receptor 2a (5ht2a), with ic50s of 0.86 and 1.3 μm,..产品型号:T9833 原产地:中国大陆价格: ¥0.0
产品名称: Netupitantorally,Neurokinin Receptor,Tachykinin receptor,Netupitant,Inhibitor,substance P,NK recepto
产品简介:netupitant is a specific neurokinin 1 (nk1) receptor antagonist (ki: 0.95 nm)...产品型号:T6905 原产地:中国大陆价格: ¥0.0
产品名称: MCC950 sodiumCP 456773,MCC-950 sodium,MCC-950,inhibit,Inhibitor,CP456773,NOD-like Receptor (NLR),CRI
产品简介:mcc950 sodium salt (ic50 of 7.5 um in bmdms) is an effective, selective nlrp3 inhibitor...产品型号:T6887 原产地:中国大陆价格: ¥0.0
产品名称: FGFR4-IN-1Fibroblast growth factor receptor,FGFR-4-IN-1,FGFR,inhibit,FGFR4IN1,Inhibitor,FGFR4 IN 1
产品简介:fgfr4-in-1 is a potent fgfr4 inhibitor (ic50: 0.7 nm)...产品型号:TQ0256 原产地:中国大陆价格: ¥0.0
产品名称: INCB3344CC chemokine receptor,INCB3344,CCR,Inhibitor,inhibit,INCB-3344,INCB 3344
产品简介:incb3344 is an effective, specific and orally bioavailable ccr2 antagonist with ic50 values of 9.5 nm (mccr2) and 5.1 nm (hccr2) in binding antagonism and 7.8 n..产品型号:TQ0103 原产地:中国大陆价格: ¥0.0
产品名称: Lerisetron5-HT Receptor,Serotonin Receptor,Serotonin,Lerisetron,Bradycardia,Inhibitor,5-hydroxytrypt
产品简介:lerisetron is an antagonist of serotonin type 3 (5-ht3) receptor, with antiemetic activity...产品型号:T8441 原产地:中国大陆价格: ¥0.0
产品名称: AMG 517AMG 517,Inhibitor,inhibit,Transient receptor potential channels,TRP Channel
产品简介:amg 517 is an effective and specific trpv1 antagonist, antagonizes proton (ic50: 0.76 nm), capsaicin (ic50: 0.62 nm), and heat activation (ic50: 1.3 nm) of trpv..产品型号:T6379 原产地:中国大陆价格: ¥0.0
产品名称: Cariprazine hydrochlorideDopamine Receptor,Cariprazine,5-hydroxytryptamine Receptor,RGH188,Inhibitor
产品简介:cariprazine hcl is an antipsychotic drug, is a d3 and d2 receptor partial agonist((ki of 0.085 nm and 0.49 nm, respectively)..产品型号:T8382 原产地:中国大陆价格: ¥0.0
产品名称: σ1 Receptor antagonist-1anti-nociceptive,Sigma Receptor,cycle,σ1 Receptor antagonist1,σ1 Receptor an
产品简介:σ1 receptor antagonist-1 is a selective sigma 1 receptor antagonist...产品型号:T9244 原产地:中国大陆价格: ¥0.0
产品名称: ZuranoloneInhibitor,inhibit,γ-Aminobutyric acid Receptor,Gamma-aminobutyric acid Receptor,GABA Recep
产品简介:zuranolone is an agonist of gabaa receptor...产品型号:T7794 原产地:中国大陆价格: ¥0.0
产品名称: Mepenzolate BromideHCAR2,PUMA-G,inhibit,Muscarinic acetylcholine receptor,Inhibitor,hM3R,gastrointes
产品简介:mepenzolate bromide is a muscarinic antagonist used to treat gastrointestinal conditions...产品型号:T0794 原产地:中国大陆价格: ¥0.0
产品名称: FluocinonideFluocinonide,Glucocorticoid Receptor,inhibit,Inhibitor
产品简介:fluocinonide (vanos) is an effective glucocorticoid steroid, utilized in the treatment as the skin disorders anti-inflammatory agent...产品型号:T6502 原产地:中国大陆价格: ¥0.0
产品名称: HypaconitineInhibitor,TNFR,TNF Receptor,inhibit,Tumor Necrosis Factor Receptor,Hypaconitine
产品简介:hypaconitine, an active and highly toxic constituent derived from aconitum species, has anti-inflammatory activity, is widely used to treat rheumatism...产品型号:T6S0630 原产地:中国大陆价格: ¥0.0
产品名称: Guanabenz AcetateAdrenergic Receptor,Guanabenz Acetate,Wy 8678,Guanabenz,Beta Receptor,Wy8678,BR 750
产品简介:guanabenz acetate is a specific agonist of adrenergic receptor. the pec50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor is 8...产品型号:T6522 原产地:中国大陆价格: ¥0.0
产品名称: Melanotan IInhibitor,MC1R,Melanocortin Receptor,skin cancers,α-MSH,melanotropic peptide,Melanotan,Me
产品简介:melanotan-i has the amino acid sequence of ser-tyr-ser-nle-glu-his-d-phe-arg-trp-gly-lys-pro-val and a molecular weight of 1647.4 dalton...产品型号:TP1097 原产地:中国大陆价格: ¥0.0
产品名称: AzaperoneR1929,R 1929,inhibit,Inhibitor,Dopamine Receptor,Azaperone
产品简介:azaperone is a pyridinylpiperazine and butyrophenone neuroleptic drug with sedative and antiemetic effects, which is used mainly as a tranquilizer in veterinary..产品型号:T6398 原产地:中国大陆价格: ¥0.0
产品名称: GSK805GSK 805,immunity,RAR-related orphan receptor,Inhibitor,GSK805,inhibit,ROR,oral,CNS penetrant,G
产品简介:gsk805 is a potent, orally bioavailable retinoid-related orphan receptor gamma t (rorγt) inverse agonist that interacts with the receptor´s putative ligan..产品型号:T7388 原产地:中国大陆价格: ¥0.0
产品名称: AnamorelinONO 7643,GHSR,RC1291,ONO7643,Growth hormone secretagogue receptor,Inhibitor,RC 1291,inhibi
产品简介:anamorelin is a novel ghrelin receptor agonist (ec50: 0.74 nm in the flipr assay)...产品型号:T10319 原产地:中国大陆价格: ¥0.0
产品名称: VelsecoratAZD 7594,Inhibitor,AZD-7594,Velsecorat,Glucocorticoid Receptor,AZ-13189620,AZ 13189620,inh
产品简介:azd7594 is an effective and selective nonsteroidal glucocorticoid receptor modulator (ic50: 0.9 nm)...产品型号:TQ0225 原产地:中国大陆价格: ¥0.0
产品名称: GeraniinGeraniin,Tumor Necrosis Factor Receptor,inhibit,TNF Receptor,Inhibitor,TNFR
产品简介:1. geraniin has a protective effect against ovx-induced rat osteoporosis. 2. geraniin has cytotoxic activity towards cancer cells in vitro and in vivo. 3. geran..产品型号:T6S2099 原产地:中国大陆价格: ¥0.0