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产品名称: BGG463;化合物K 0859K 0859;K 0859
产品简介:bgg463 (k 0859) can inhibit c-abl-t334i, bcr-abl and bcr-abl-t315i variants with a 50% inhibitory concentration (ic50) of 0.25 μm, 0.09 μm and 0.590 μm, respect..产品型号:T4618 原产地:中国大陆价格: ¥0.0
产品名称: KN-92;化合物 T4530LK92|||KN-92 free base|||K 92;K92|||KN-92 free base|||K 92
产品简介:kn-92 is an inactive analog of the cam kinase ii inhibitor kn 93...产品型号:T4530L 原产地:中国大陆价格: ¥0.0
产品名称: Selective PI3Kδ Inhibitor 1;化合物Selective PI3Kδ Inhibitor 1Selective PI3Kδ Inhibitor 1
产品简介:selective pi3kδ inhibitor 1 is a pi3kδ inhibitor( ic50 = 0.9 nm)...产品型号:T5831 原产地:中国大陆价格: ¥0.0
产品名称: K783-0308;化合物 K783-0308K783-0308
产品简介:k783-0308 is a potent and selective mnk2 and flt3 dual inhibitor with ic 50 values of 406 and 680 nm, respectively. k783-0308 promotes the apoptosis and cell cy..产品型号:T61005 原产地:中国大陆价格: ¥0.0
产品名称: PI3Kα-IN-6;化合物 PI3Kα-IN-6PI3Kα-IN-6
产品简介:pi3kα-in-6 (compound 5b) is a pi3kα inhibitor that exhibits anticancer effects without toxicity to normal cells. pi3kα-in-6 increases ros production, decreases ..产品型号:T62073 原产地:中国大陆价格: ¥0.0
产品名称: COX-2/PI3K-IN-1;化合物 COX-2/PI3K-IN-1COX-2/PI3K-IN-1
产品简介:cox-2/pi3k-in-1 (compound 5d) is a potent inhibitor of pi3k (ic50: 1.14 nm). cox-2/pi3k-in-1 is a selective inhibitor of cox-2 (ki: 3.24 nm)...产品型号:T62103 原产地:中国大陆价格: ¥0.0
产品名称: PI3Kγ inhibitor 4;化合物 PI3Kγ inhibitor 4PI3Kγ inhibitor 4
产品简介:pi3kγ inhibitor 4 is a selective, potent, orally active pi3kγ inhibitor (ic50: 40 nm). pi3kγ inhibitor 4 is ~7-fold more selective for pi3kγ than the α subtype,..产品型号:T62165 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/HDAC-IN-2;化合物 PI3K/HDAC-IN-2PI3K/HDAC-IN-2
产品简介:pi3k/hdac-in-2 is a potent dual pi3k/hdac inhibitor, capable of acting on pi3kα (ic50: 226 nm), pi3kβ (ic50: 279 nm), pi3kγ (ic50: 467 nm), pi3kδ (ic50: 29 nm),..产品型号:T62912 原产地:中国大陆价格: ¥0.0
产品名称: PI3Kδ/γ-IN-3;化合物 PI3Kδ/γ-IN-3PI3Kδ/γ-IN-3
产品简介:pi3kδ/γ-in-3 (compound 58) is an orally active dual inhibitor of pi3kδ (ic50: 1 nm) and pi3kγ (ic50: 16 nm). pi3kδ/γ-in-3 can induce apoptosis of tumor cells, w..产品型号:T63078 原产地:中国大陆价格: ¥0.0
产品名称: PI3Kβ-IN-1;化合物 PI3Kβ-IN-1PI3Kβ-IN-1
产品简介:pi3kβ-in-1 is a selective, orally active pi3kβ inhibitor (ic50: 2 nm)...产品型号:T62948 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/AKT-IN-1;化合物 PI3K/AKT-IN-1PI3K/AKT-IN-1
产品简介:pi3k/akt-in-1 is a potent, dual pi3k/akt inhibitor that acts on pi3kγ (ic50: 6.99 μm), pi3kδ (ic50: 4.01 μm) and akt (ic50: 3.36 μm). pi3k/akt-in-1 induces casp..产品型号:T62997 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/mTOR Inhibitor-7;化合物 PI3K/mTOR Inhibitor-7PI3K/mTOR Inhibitor-7
产品简介:pi3k/mtor inhibitor-7 is a potent dual pi3k/mtor inhibitor. pi3k/mtor inhibitor-7 is 4.7-fold more potent than gedatolisib, with ic50 values of 1.4 μm and 0.3 μ..产品型号:T64041 原产地:中国大陆价格: ¥0.0
产品名称: Cathepsin K inhibitor 2;化合物 Cathepsin K inhibitor 2Cathepsin K inhibitor 2
产品简介:cathepsin k inhibitor 2 is a potent inhibitor of cathepsin k. cathepsin k (cat k) is a cysteine protease expressed under the control of the ctsk gene, which is ..产品型号:T64159 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/mTOR Inhibitor-6;化合物 PI3K/mTOR Inhibitor-6PI3K/mTOR Inhibitor-6
产品简介:pi3k/mtor inhibitor-6 (compound 19c) is a potent dual pi3k/mtor inhibitor that is more stable than gedatolisib in artificial gastric fluid. 10 μm of pi3k/mtor i..产品型号:T64219 原产地:中国大陆价格: ¥0.0
产品名称: all-trans-4-Oxoretinoic acid;4-KETO全反式维甲酸all-trans 4-Keto Retinoic Acid;4-KETO全反式维甲酸|||all-trans 4-K
产品简介:all-trans-4-oxoretinoic acid (all-trans 4-keto retinoic acid) is an active metabolite of vitamin a...产品型号:T7408 原产地:中国大陆价格: ¥0.0
产品名称: LL-K8-22;化合物 LL-K8-22LL-K8-22
产品简介:ll-k8-22 is a potent, selective, and durable dual degrader of cdk8-cyclin c, demonstrating dc50 values of 2.52 and 2.64 μm, respectively. this compound effectiv..产品型号:T74784 原产地:中国大陆价格: ¥0.0
产品名称: Ripasudil free base;化合物Ripasudil free baseK-115 (free base);K-115 (free base)
产品简介:ripasudil free base (k-115 (free base)) is a selective and potent rock inhibitor, is a novel and potent antiglaucoma agent...产品型号:T7492 原产地:中国大陆价格: ¥0.0
产品名称: M4K2234;化合物 M4K2234M4K2234
产品简介:m4k2234 (compound 26b), an alk2 inhibitor, demonstrates selective inhibition of alk2 and alk5 with ic50 values of 5 nm and 2144 nm, respectively. serving as a c..产品型号:T74660 原产地:中国大陆价格: ¥0.0
产品名称: cis-Vitamin K1;化合物 cis-Vitamin K1cis-Vitamin K1
产品简介:cis-vitamin k1 is an endogenous metabolite of vitamin k [1] ...产品型号:T75435 原产地:中国大陆价格: ¥0.0
产品名称: Guignardone K;化合物 Guignardone KGuignardone K
产品简介:guignardone k, a meroterpene compound extracted from solid cultures of the endophytic fungus guignardia sp., exhibits antifungal activity [1]...产品型号:T75480 原产地:中国大陆价格: ¥0.0