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产品名称: EI1EI1,Ezh2 inhibitor,KB-145943
产品简介:ei1 is a potent and selective ezh2 inhibitor with ic50 of 15 nm and 13 nm for ezh2 (wt) and ezh2 (y641f), respectively...产品型号:T6484 原产地:美洲价格: ¥0.0
产品名称: CGP 57380CGP 57380,MNK1 Inhibitor,
产品简介:cgp 57380 is a potent mnk1 inhibitor with ic50 of 2.2 μm, exhibiting no inhibitory activity on p38, jnk1, erk1 and -2, pkc, or c-src-like kinases...产品型号:T6440 原产地:美洲价格: ¥0.0
产品名称: SU11274SU11274,PKI-SU11274,Met Kinase Inhibitor
产品简介:su11274(ic50=10 nm) is a specific met inhibitor. it shows no significant effects on pgdfrβ, egfr or tie2...产品型号:T6154 原产地:美洲价格: ¥0.0
产品名称: CX-6258 HClCX-6258 HCl,Pim-Kinase Inhibitor X,
产品简介:cx-6258 hcl is an effective, orally efficacious pim1/2/3 kinase inhibitor (ic50: 5/25/16 nm)...产品型号:T6148 原产地:美洲价格: ¥0.0
产品名称: ZM 39923 HClZM 39923 HCl,JAK3 Inhibitor IV,
产品简介:zm 39923 hcl is an jak1/3 inhibitor with pic50 of 4.4/7.1, almost no activity to jak2 and modestly potent to egfr; also found to be sensitive to transglutamina..产品型号:T6145 原产地:美洲价格: ¥0.0
产品名称: IMD 0354IMD 0354,IKK2 Inhibitor V,
产品简介:imd-0354 is an ikkβ inhibitor and inhibits iκbα phosphorylation in nf-κb pathway...产品型号:T6141 原产地:美洲价格: ¥0.0
产品名称: TCS 359TCS 359,FLT3 Inhibitor,
产品简介:tcs 359 is a potent flt3 inhibitor with ic50 of 42 nm...产品型号:T6138 原产地:美洲价格: ¥0.0
产品名称: Tie2 kinase inhibitorTie2 kinase inhibitor
产品简介:tie2 kinase inhibitor, an optimized compound of sb-203580, is selective to tie2 with ic50 of 0.25 μm, which is 200-fold more effective than p38...产品型号:T6335 原产地:美洲价格: ¥0.0
产品名称: StatticStattic,STAT3 Inhibitor V,
产品简介:stattic is a small molecule inhibitor of stat3. it selectively inhibits stat3 activation, dimerization, and nuclear translocation (ic50: 5.1 μm)...产品型号:T6308 原产地:美洲价格: ¥0.0
产品名称: Tuberculosis inhibitor 12;化合物 Tuberculosis inhibitor 12Tuberculosis inhibitor 12
产品简介:tuberculosis inhibitor 12, an oxadiazole derivative, effectively inhibits mycobacterium tuberculosis, demonstrating inhibition rates of 82% and 78% at a concent..产品型号:T80925 原产地:中国大陆价格: ¥0.0
产品名称: ALK inhibitor 2;化合物ALK inhibitor 2ALK inhibitor 2
产品简介:alk inhibitor 2 is a new-type and selective inhibitor for the alk kinase...产品型号:T3041 原产地:中国大陆价格: ¥0.0
产品名称: JAK2 Inhibitor V;化合物 JAK2 Inhibitor VJAK2 Inhibitor V Z3|||Z3;JAK2 Inhibitor V Z3|||Z3
产品简介:jak2 inhibitor v (jak2 inhibitor v z3) is a novel specific inhibitor of jak2, inhibiting jak2-v617f and jak2-wt autophosphorylation in a dose-dependent manner...产品型号:T3042 原产地:中国大陆价格: ¥0.0
产品名称: BMS-202;化合物PD1-PDL1 inhibitor 2PD1-PDL1 inhibitor 2|||PD-1/PD-L1 inhibitor 2;PD1-PDL1 inhibitor 2|||
产品简介:bms-202 (pd1-pdl1 inhibitor 2) is an inhibitor of the pd-1 (programmed death- 1) /pd-ll (programmed death-ligand 1) protein/protein interaction...产品型号:T3146 原产地:中国大陆价格: ¥0.0
产品名称: Wedelolactone;蟛蜞菊内酯IKK Inhibitor II;蟛蜞菊内酯|||IKK Inhibitor II
产品简介:wedelolactone (ikk inhibitor ii) inhibits nf-κb-mediated gene transcription in cells by blocking the phosphorylation and degradation of iκbα...产品型号:T3384 原产地:中国大陆价格: ¥0.0
产品名称: Miransertib;化合物MiransertibARQ-092|||AKT inhibitor 2;ARQ-092|||AKT inhibitor 2
产品简介:miransertib (arq-092) is an orally bioavailable, selective, and potent allosteric akt inhibitor...产品型号:T3467 原产地:中国大陆价格: ¥0.0
产品名称: JNJ-42153605化合物JNJ42153605Inhibitor|||Metabotropic glutamate receptors|||JNJ 42153605
产品简介:jnj-42153605 is a mglu2 receptor positive allosteric modulator (ec50: 17 nm)...产品型号:T3451 原产地:中国大陆价格: ¥0.0
产品名称: Ac-YVAD-CMK;化合物Ac-YVAD-CMKCaspase-1 Inhibitor II|||Ac-Tyr-Val-Ala-Asp-chloromethylketone|||Ac-Tyr-Va
产品简介:ac-yvad-cmk (ac-tyr-val-ala-asp-cmk) is a selective and irreversible inhibitor of caspase-1 and inhibits pyroptosis, il-1β and il-18. ac-yvad-cmk shows neuropro..产品型号:T36347 原产地:中国大陆价格: ¥0.0
产品名称: 15-LOX-1 inhibitor 19c(i472)15 LOX 1 inhibitor 1|||15LOX1 inhibitor 1
产品简介:9c(i472) is an inhibitor of 15-lipoxygenase-1 (15-lo-1; ic50 = 0.19 μm).1 it decreases lps- and ifn-γ-induced nf- b activity in raw-blue cells when used at con..产品型号:T36169 原产地:中国大陆价格: ¥0.0
产品名称: Btk inhibitor 1 hydrochloride;Btk inhibitor 1 hydrochlorideBtk inhibitor 1 hydrochloride
产品简介:btk inhibitor 1 hcl is a pyrazolo[3,4-d]pyrimidine derivative as a btk kinase inhibitor...产品型号:T36297 原产地:中国大陆价格: ¥0.0
产品名称: mTOR inhibitor-8;抑制剂8mTOR-IN-8;mTOR-IN-8
产品简介:mtor inhibitor-8 is a potent mtor inhibitor and autophagy inducer with antiviral and antitumor activity. mtor inhibitor-8 inhibits the growth of a549 cells, whi..产品型号:T36316 原产地:中国大陆价格: ¥0.0