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产品名称: 5-HT6/5-HT2A receptor ligand-2;化合物 5-HT6/5-HT2A receptor ligand-25-HT6/5-HT2A receptor ligand-2
产品简介:compound 42, a 5-ht6/5-ht2a receptor ligand-2, serves as a dual antagonist for the 5-ht6 and 5-ht2a receptors with ki values of 25 nm and 32 nm, respectively. t..产品型号:T61220 原产地:中国大陆价格: ¥0.0
产品名称: VEGFR-2/DHFR-IN-2;化合物 VEGFR-2/DHFR-IN-2VEGFR-2/DHFR-IN-2
产品简介:vegfr-2/dhfr-in-2 (compound 5b) is a dual inhibitor targeting vegfr-2 and dhfr, with respective ic50 values of 0.623 μm and 9.085 μm. it demonstrates potent cyt..产品型号:T61229 原产地:中国大陆价格: ¥0.0
产品名称: CXCR2 antagonist 5;化合物 CXCR2 antagonist 5CXCR2 antagonist 5
产品简介:cxcr2 antagonist 5 (compound 25) is a potent cxcr2 antagonist. cxcr2 antagonist 5 shows potent cxcr2 binding affinity ( ic 50 =0.013 μm) and calcium mobilizatio..产品型号:T61235 原产地:中国大陆价格: ¥0.0
产品名称: CXCR2 antagonist 7;化合物 CXCR2 antagonist 7CXCR2 antagonist 7
产品简介:cxcr2 antagonist 7 (compound 19) is a potent cxcr2 antagonist. cxcr2 antagonist 7 shows potent cxcr2 binding affinity ( ic 50 =0.044 μm) and calcium mobilizatio..产品型号:T61236 原产地:中国大陆价格: ¥0.0
产品名称: NAT2-IN-1;化合物 NAT2-IN-1NAT2-IN-1
产品简介:nat2-in-1 (apa) is a selective inhibitor of the drug metabolism enzyme n-acetyltransferase 2 (nat2), capable of targeting and eliminating cells with slow nat2 a..产品型号:T61238 原产地:中国大陆价格: ¥0.0
产品名称: MAT2A-IN-5;化合物 MAT2A-IN-5MAT2A-IN-5
产品简介:mat2a-in-5, a potent inhibitor of mat2a, effectively targets the abnormally elevated expression of mat2a found in various tumor types such as gastric, colon, li..产品型号:T61243 原产地:中国大陆价格: ¥0.0
产品名称: AhR agonist 2;化合物 AhR agonist 2AhR agonist 2
产品简介:ahr agonist 2 (compound 12a) is a highly potent agonist of the aryl hydrocarbon receptor (ahr), exhibiting an ec50 value of 0.03 nm. this compound rapidly induc..产品型号:T61244 原产地:中国大陆价格: ¥0.0
产品名称: α-Glucosidase-IN-2;化合物 α-Glucosidase-IN-2α-Glucosidase-IN-2
产品简介:α-glucosidase-in-2 (compound 5d) is a potent inhibitor of α-glucosidase, exhibiting an inhibitory concentration (ic50) of 9.48 μm, and functions as an antidiabe..产品型号:T61249 原产地:中国大陆价格: ¥0.0
产品名称: COX-2/5-LOX-IN-3;化合物 COX-2/5-LOX-IN-3COX-2/5-LOX-IN-3
产品简介:cox-2/5-lox-in-3 (compound 5b) is a powerful and dual inhibitor of cox-2 and 5-lox, with ic50 values of 45.73 μm, 5.45 μm, and 4.33 μm for cox-1, cox-2, and 5-l..产品型号:T61352 原产地:中国大陆价格: ¥0.0
产品名称: PqsR-IN-2;化合物 PqsR-IN-2PqsR-IN-2
产品简介:pqsr-in-2 (compound 19) is a highly potent inhibitor of pqsr, the transcriptional regulator responsible for quorum sensing in pseudomonas aeruginosa. it effecti..产品型号:T61353 原产地:中国大陆价格: ¥0.0
产品名称: CXCR2 antagonist 3;化合物 CXCR2 antagonist 3CXCR2 antagonist 3
产品简介:cxcr2 antagonist 3 (compound 11h) is a highly effective antagonist of cxc chemokine receptor 2 (cxcr2). it displays potent activity in inhibiting neutrophil inf..产品型号:T61356 原产地:中国大陆价格: ¥0.0
产品名称: CXCR2 antagonist 6;化合物 CXCR2 antagonist 6CXCR2 antagonist 6
产品简介:cxcr2 antagonist 6 (compound 35c) is a potent cxcr2 antagonist. cxcr2 antagonist 6 shows potent cxcr2 binding affinity ( ic 50 =0.044 μm) and calcium mobilizati..产品型号:T61359 原产地:中国大陆价格: ¥0.0
产品名称: HIF-2α-IN-6;化合物 HIF-2α-IN-6HIF-2α-IN-6
产品简介:hif-2α-in-6 (117) is a hif-2α inhibitor [1]...产品型号:T61367 原产地:中国大陆价格: ¥0.0
产品名称: p53 Activator 2;化合物 p53 Activator 2p53 Activator 2
产品简介:p53 activator 2 (compound 10ah) intercalates into dna, causing significant dna double-strand breaks and upregulates the expression of p53, p-p53, cdk4, and p21,..产品型号:T61369 原产地:中国大陆价格: ¥0.0
产品名称: 5-HT7 agonist 2;化合物 5-HT7 agonist 25-HT7 agonist 2
产品简介:5-ht7 agonist 2 is a highly potent 5-ht7 receptor agonist, exhibiting an ic50 value of 28.7 nm. this compound holds promise for studying and understanding vario..产品型号:T61375 原产地:中国大陆价格: ¥0.0
产品名称: CXCR4 modulator-2;化合物 CXCR4 modulator-2CXCR4 modulator-2
产品简介:cxcr4 modulator-2 (compound z7r) is a potent modulator of cxcr4 (ic50: 1.25 nm). cxcr4 modulator-2 exhibits good stability in mouse serum (t1/2= 77.1 min) and h..产品型号:T62352 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2 nsp13-IN-3;化合物 SARS-CoV-2 nsp13-IN-3SARS-CoV-2 nsp13-IN-3
产品简介:sars-cov-2 nsp13-in-3 (compound c3) is a small molecule inhibitor of sars-cov-2 non-structural protein 13 (nsp13) that acts on nsp13 ssdna+atpase (ic50: 32 μm)...产品型号:T62375 原产地:中国大陆价格: ¥0.0
产品名称: (1R,2R)-ML-SI3;化合物 (1R,2R)-ML-SI3(1R,2R)-ML-SI3
产品简介:(1r,2r)-ml-si3 is a potent inhibitor of trpml1 (ic50: 1.6 μm) and trpml2 (ic50: 2.3 μm). (1r,2r)-ml-si3 is also a weak inhibitor of trpml3 with an ic50 value of..产品型号:T62378 原产地:中国大陆价格: ¥0.0
产品名称: Anti-MRSA agent 2;化合物 Anti-MRSA agent 2Anti-MRSA agent 2
产品简介:anti-mrsa agent 2 (compound 14) is a good inhibitor of methicillin-resistant staphylococcus aureus (mrsa) (mic: 0.098 μg/ml) with relatively low toxicity to nor..产品型号:T62383 原产地:中国大陆价格: ¥0.0
产品名称: α7 nAchR-JAK2-STAT3 agonist 1;化合物 α7 nAchR-JAK2-STAT3 agonist 1α7 nAchR-JAK2-STAT3 agonist 1
产品简介:α7 nachr-jak2-stat3 agonist 1 is a potent inhibitor of the α7 nachr-jak2-stat3 pathway that acts on nitric oxide (no) (ic50: 0.32 μm). α7 nachr-jak2-stat3 agoni..产品型号:T62317 原产地:中国大陆价格: ¥0.0