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产品名称: MALT1-IN-3;化合物 MALT1-IN-3MALT1-IN-3
产品简介:malt1-in-3 is a potent inhibitor of malt1 protease (ic50: 0.06 μm) with ic50 values of 0.14 and 0.13 μm for human il6 and il10, respectively, in oci-ly3 cells...产品型号:T63053 原产地:中国大陆价格: ¥0.0
产品名称: FLT3-IN-14;化合物 FLT3-IN-14FLT3-IN-14
产品简介:flt3-in-14 is a potent inhibitor of flt3, acting on flt3-wt (ic50: 5.6 nm) and flt3-itd (ic50: 1.4 nm). flt3-in-14 inhibits flt3 (y591) phosphorylation, arrests..产品型号:T63058 原产地:中国大陆价格: ¥0.0
产品名称: Dopamine D3 receptor antagonist-2;化合物 Dopamine D3 receptor antagonist-2Dopamine D3 receptor antagoni
产品简介:dopamine d3 receptor antagonist-2 is a dopamine d3 receptor selective (ki=2.16 nm) or multi-targeting dual ligand that shows potential effects in cns disorders...产品型号:T62946 原产地:中国大陆价格: ¥0.0
产品名称: PI3Kβ-IN-1;化合物 PI3Kβ-IN-1PI3Kβ-IN-1
产品简介:pi3kβ-in-1 is a selective, orally active pi3kβ inhibitor (ic50: 2 nm)...产品型号:T62948 原产地:中国大陆价格: ¥0.0
产品名称: (1R,3S)-THCCA-Asn;化合物 (1R,3S)-THCCA-Asn(1R,3S)-THCCA-Asn
产品简介:(1r,3s)-thcca-asn (4j) is a selective inhibitor of thrombin (ic50: 0.07-0.14 μm) with anti-thrombotic effects...产品型号:T62949 原产地:中国大陆价格: ¥0.0
产品名称: Axl-IN-3;化合物 Axl-IN-3Axl-IN-3
产品简介:axl-in-3 is a selective, potent and orally active inhibitor of axl kinase (ic50: 41.5 nm) and has a low inhibitory effect on other kinases...产品型号:T62962 原产地:中国大陆价格: ¥0.0
产品名称: HIV-IN-3;化合物 HIV-IN-3HIV-IN-3
产品简介:hiv-in-3 (compound 22a) is a potent inhibitor of hiv (ic50: 1.5 μm). hiv-in-3 has potential for the study of hiv-related diseases...产品型号:T62978 原产地:中国大陆价格: ¥0.0
产品名称: FLT3/CDK4-IN-1;化合物 FLT3/CDK4-IN-1FLT3/CDK4-IN-1
产品简介:flt3/cdk4-in-1 is a highly selective, potent, orally active dual inhibitor of flt3/cdk4, acting on flt3 (ic50: 7 nm) and cdk4 (ic50: 11 nm).flt3/cdk4-in-1 has g..产品型号:T63135 原产地:中国大陆价格: ¥0.0
产品名称: DX3-213B;化合物DX3-213BDX3-213B
产品简介:dx3-213b is a potent, orally active inhibitor of oxidative phosphorylation (oxphos) complex i with an ic50 of 3.6 nm. dx3-213b blocks atp production (ic50: 11 n..产品型号:T63136 原产地:中国大陆价格: ¥0.0
产品名称: LY-411575 (isomer 3);化合物 LY-411575 (isomer 3)LY-411575 (isomer 3)
产品简介:ly-411575 isomer 3 is an isomer of ly411575. ly411575 is a potent γ-secretase inhibitor...产品型号:T63150 原产地:中国大陆价格: ¥0.0
产品名称: MMP-9-IN-3;化合物 MMP-9-IN-3MMP-9-IN-3
产品简介:mmp-9-in-3 is an mmp-9 inhibitor (ic50: 5.56 nm) that forms hydrogen bonds with mmp-9. mmp-9-in-3 inhibits akt activity (ic50: 2.11 nm). mmp-9-in-3 is cytotoxic..产品型号:T63155 原产地:中国大陆价格: ¥0.0
产品名称: Calcitriol;骨化三醇Topitriol|||Rocaltrol|||Calcijex|||RO215535|||1,25-Dihydroxyvitamin D3;Topitriol|||Ro
产品简介:calcitriol (1,25-dihydroxyvitamin d3) is a metabolite of vitamin d and a vitamin d receptor (vdr) agonist (ic50=0.4 nm). calcitriol increases intestinal absorpt..产品型号:T6316 原产地:中国大陆价格: ¥0.0
产品名称: EGFR/HER2/CDK9-IN-3;化合物 EGFR/HER2/CDK9-IN-3EGFR/HER2/CDK9-IN-3
产品简介:egfr/her2/cdk9-in-3 (compound 10) is a potent inhibitor of egfr (ic50:191.08 nm), her2 (ic50:132.65 nm), and cdk9 (ic50:113.98 nm). egfr/her2/cdk9-in-3 showed s..产品型号:T63161 原产地:中国大陆价格: ¥0.0
产品名称: VEGFR-IN-3;化合物 VEGFR-IN-3VEGFR-IN-3
产品简介:vegfr-in-3 (compound 3f), a vegfr inhibitor, exhibits potent anticancer activity by inhibiting the growth of ovcar-4 and mda-mb-468 cancer cells with ic50 value..产品型号:T63112 原产地:中国大陆价格: ¥0.0
产品名称: PDGFRα/FLT3-ITD-IN-3;化合物 PDGFRα/FLT3-ITD-IN-3PDGFRα/FLT3-ITD-IN-3
产品简介:pdgfrα/flt3-itd-in-3 (compound 18d) is a potent inhibitor of pdgfrα (ic50: 0.153 μm), flt3 (ic50: 0.004 μm) and pdgfrα/flt3-itd-in-3 has the potential to be stu..产品型号:T63127 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/AKT-IN-1;化合物 PI3K/AKT-IN-1PI3K/AKT-IN-1
产品简介:pi3k/akt-in-1 is a potent, dual pi3k/akt inhibitor that acts on pi3kγ (ic50: 6.99 μm), pi3kδ (ic50: 4.01 μm) and akt (ic50: 3.36 μm). pi3k/akt-in-1 induces casp..产品型号:T62997 原产地:中国大陆价格: ¥0.0
产品名称: Butein;紫铆因2’,3,4,4’-tetrahydroxy Chalcone;2’,3,4,4’-tetrahydroxy Chalcone|||紫铆因
产品简介:butein (2’,3,4,4’-tetrahydroxy chalcone), a plant polyphenol, is isolated from rhus verniciflua. it can inhibit the activation of protein tyrosine kinase, nf-κb..产品型号:T6427 原产地:中国大陆价格: ¥0.0
产品名称: Calcifediol;25-羟基维生素 D3U 32070E|||25-hydroxy Vitamin D3|||RO 8-8892;25-羟基维生素 D3|||U 32070E|||25-hydr
产品简介:calcifediol (u 32070e)(ki of 3.9 μm), a major circulating metabolite of vitamin d3, works as a competitive inhibitor. it (ed50=2 nm)also inhibits pth secretion ..产品型号:T6430 原产地:中国大陆价格: ¥0.0
产品名称: DX3-235;化合物 DX3-235DX3-235
产品简介:dx3-235 is an inhibitor of oxidative phosphorylation (oxphos). in galactose-containing media, dx3-235 inhibits complex i function and atp production by nanomola..产品型号:T64108 原产地:中国大陆价格: ¥0.0
产品名称: AChE/BuChE-IN-3;化合物 AChE/BuChE-IN-3AChE/BuChE-IN-3
产品简介:ache/buche-in-3 is a potent inhibitor of ache (ic50: 0.65 μm) and buche (ic50: 5.77 μm) that crosses the blood-brain barrier and also exhibits an inhibitory eff..产品型号:T64137 原产地:中国大陆价格: ¥0.0