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产品名称: Tau-aggregation-IN-1;化合物 Tau-aggregation-IN-1Tau-aggregation-IN-1
产品简介:tau-aggregation-in-1 is a dopamine d2 and d3 receptor agonist and an inhibitor of tau441 protein aggregation (ic50: 21 μm)...产品型号:T63481 原产地:中国大陆价格: ¥0.0
产品名称: Snail/HDAC-IN-1;Snail/HDAC 抑制剂1Snail/HDAC-IN-1
产品简介:snail/hdac-in-1 is a snail/hdac inhibitor agent with antimicrobial and anticancer activity, reduces snail protein expression, induces apoptosis, and can be used..产品型号:T63260 原产地:中国大陆价格: ¥0.0
产品名称: HDAC1-IN-4;化合物 HDAC1-IN-4HDAC1-IN-4
产品简介:hdac1-in-4 is a potent inhibitor of plasmodium falciparum hdac1 (pfhdac1) with low cytotoxicity and antimalarial effects (ic50<5 nm)...产品型号:T63482 原产地:中国大陆价格: ¥0.0
产品名称: INSCoV-614(1B);化合物 INSCoV-614(1B)INSCoV-614(1B)
产品简介:inscov-614(1b) is a potent mpro(3clpro) inhibitor. proteases (plpro and 3clpro) are associated with viral transcription and replication. inscov-614(1b) has show..产品型号:T63483 原产地:中国大陆价格: ¥0.0
产品名称: CYP2C1/CYP2C19-IN-2;化合物 CYP2C1/CYP2C19-IN-2CYP2C1/CYP2C19-IN-2
产品简介:cyp2c1/cyp2c19-in-2 is a potent inhibitor of cyp2c9/cyp2c19 without liver toxicity or genotoxicity and can be used to study zika virus (zikv) infection...产品型号:T63495 原产地:中国大陆价格: ¥0.0
产品名称: PI3Kδ/γ-IN-1;化合物 PI3Kδ/γ-IN-1PI3Kδ/γ-IN-1
产品简介:pi3kδ/γ-in-1 is a selective and effective inhibitor of pi3kδ/γ that can be used in the treatment of hematologic malignancies...产品型号:T63497 原产地:中国大陆价格: ¥0.0
产品名称: HIV-1 inhibitor-28;化合物 HIV-1 inhibitor-28HIV-1 inhibitor-28
产品简介:hiv-1 inhibitor-28 is a potent and selective hiv-1 inhibitor with ec50=58 nm for wild-type hiv-1, ic50=3.37 μm for wild-type hiv-1 reverse transcription, and re..产品型号:T63499 原产地:中国大陆价格: ¥0.0
产品名称: Chroman 1 dihydrochloride;化合物 Chroman 1 dihydrochlorideChroman 1 dihydrochloride
产品简介:chroman 1 dihydrochloride is a selective and potent inhibitor of rock, acting more strongly on rock2 (ic50: 1 pm) than rock1 (ic50: 52 pm) and also inhibiting m..产品型号:T63506 原产地:中国大陆价格: ¥0.0
产品名称: Top/HDAC-IN-1;化合物 Top/HDAC-IN-1Top/HDAC-IN-1
产品简介:top/hdac-in-1 is a dual topoisomerase (top)/hdac inhibitor that acts on hdac1 (ic50: 18 nm), hdac2 (ic50: 230 nm), hdac3 (ic50: 790 nm), hdac6 (ic50: 87 nm) and..产品型号:T63509 原产地:中国大陆价格: ¥0.0
产品名称: IRE1α kinase-IN-4;化合物 IRE1α kinase-IN-4IRE1α kinase-IN-4
产品简介:ire1α kinase-in-4 (compound 6) is a potent inhibitor of ire1α, exhibiting a ki value of 140 nm. it acts as an atp-competitive ligand for ire1α [1]...产品型号:T63511 原产地:中国大陆价格: ¥0.0
产品名称: PPARγ agonist 1;化合物 PPARγ agonist 1PPARγ agonist 1
产品简介:pparγ agonist 1 is a potent agonist of pparγ that efficiently activates hpparγ without causing full agonism, thereby avoiding adverse effects. pparγ agonist 1 h..产品型号:T63514 原产地:中国大陆价格: ¥0.0
产品名称: USP1-IN-2;USP1 抑制剂2USP1-IN-2
产品简介:usp1-in-2 is a potent usp1 inhibitor with potential anti-tumor activity for the study of cancer...产品型号:T63518 原产地:中国大陆价格: ¥0.0
产品名称: DCN1-UBC12-IN-1;化合物 DCN1-UBC12-IN-1DCN1-UBC12-IN-1
产品简介:dcn1-ubc12-in-1 is a potent and specific dcn1-ubc12 inhibitor with an ic50 value of 2.86 nm and anti-cardiac fibrogenic activity...产品型号:T63647 原产地:中国大陆价格: ¥0.0
产品名称: EGFR kinase inhibitor 1;化合物 EGFR kinase inhibitor 1EGFR kinase inhibitor 1
产品简介:egfr kinase inhibitor 1 is a potent inhibitor of egfr that acts on wt (ic50: 37 nm), l885r/t790m (ic50: 1.7 nm), and l858r/t790m/c797s (ic50>300 nm). egfr kinas..产品型号:T63648 原产地:中国大陆价格: ¥0.0
产品名称: A 922500;化合物A922500A922500|||DGAT-1 Inhibitor 4a;A922500|||(1R,2R)-2-[[4-[[(苯基氨基)羰基]氨基][1,1-联苯]-4-基]
产品简介:a 922500 (dgat-1 inhibitor 4a) is an inhibitor for human and mouse dgat-1 with ic50 of 7 nm and 24 nm, respectively, good selectivity over related acyltransfera..产品型号:T6365 原产地:中国大陆价格: ¥0.0
产品名称: IDO1/2-IN-1 hydrochloride;化合物 IDO1/2-IN-1 hydrochlorideIDO1/2-IN-1 hydrochloride
产品简介:ido1/2-in-1 hydrochloride is the first potent dual inhibitor of ido1 (ic50: 28 nm) and ido2 (ic50: 144 nm) that is orally active.ido1/2-in-1 hydrochloride exhib..产品型号:T63651 原产地:中国大陆价格: ¥0.0
产品名称: HPK1-IN-10;化合物 HPK1-IN-10HPK1-IN-10
产品简介:hpk1-in-10 is a potent inhibitor of hpk1, a serine/threonine protein kinase cloned from hematopoietic progenitor cells and a member of the map4k family of mamma..产品型号:T63659 原产地:中国大陆价格: ¥0.0
产品名称: A-966492化合物A9664922-[2-氟-4-[(2S)-2-吡咯烷基]苯基]-1H-苯并咪唑-7-甲酰胺
产品简介:a-96649 is a new-type and effective inhibitor. the ki of a-966492 for parp1 and parp2 is 1 nm and 1.5 nm, respectively...产品型号:T6366 原产地:中国大陆价格: ¥0.0
产品名称: EIF2α activator 1;化合物 EIF2α activator 1EIF2α activator 1
产品简介:eif2α activator 1 (compound 40) is a chemical compound that activates the phosphorylation of eukaryotic initiation factor 2 alpha (eif2α), enhancing the express..产品型号:T63665 原产地:中国大陆价格: ¥0.0
产品名称: HPK1-IN-9;化合物 HPK1-IN-9HPK1-IN-9
产品简介:hpk1-in-9 is a potent hpk1 inhibitor. hpk1 is a serine/threonine protein kinase cloned from hematopoietic progenitor cells and is a member of the map4k family o..产品型号:T63670 原产地:中国大陆价格: ¥0.0