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产品名称: Dopamine D3 receptor antagonist-1;化合物 Dopamine D3 receptor antagonist-1Dopamine D3 receptor antagoni
产品简介:dopamine d3 receptor antagonist-1 is a dopamine d3 receptor selective or multi-targeting ligand with a ki value of 1.58 nm that has demonstrated therapeutic pot..产品型号:T64024 原产地:中国大陆价格: ¥0.0
产品名称: CYP3A4-IN-3;化合物 CYP3A4-IN-3CYP3A4-IN-3
产品简介:cyp3a4-in-3 is a specific, highly affinity cytochrome p450 3a4 (cyp3a4) (cytochrome p450 3a4 (cyp3a4)) inhibitor (ic50: 0.075 μm). cyp3a4-in-3 is an analogue of..产品型号:T64032 原产地:中国大陆价格: ¥0.0
产品名称: CYP3A4-IN-2;化合物 CYP3A4-IN-2CYP3A4-IN-2
产品简介:cyp3a4-in-2 is a specific inhibitor of cytochrome p450 3a4 (cyp3a4) (ic50: 0.055 μm). cyp3a4-in-2 is a ritonavir analogue with a more hydrophobic r2 side group ..产品型号:T64037 原产地:中国大陆价格: ¥0.0
产品名称: Galectin-3-IN-2;化合物 Galectin-3-IN-2Galectin-3-IN-2
产品简介:galectin-3-in-2 is a potent inhibitor of polyvalent galactose lectin-3, with an ic50 value of 8.3 μm for gal-3. galectin-3 is involved in many metabolic process..产品型号:T64040 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/mTOR Inhibitor-7;化合物 PI3K/mTOR Inhibitor-7PI3K/mTOR Inhibitor-7
产品简介:pi3k/mtor inhibitor-7 is a potent dual pi3k/mtor inhibitor. pi3k/mtor inhibitor-7 is 4.7-fold more potent than gedatolisib, with ic50 values of 1.4 μm and 0.3 μ..产品型号:T64041 原产地:中国大陆价格: ¥0.0
产品名称: EZH2-IN-13;EZH2抑制剂3EZH2-IN-13
产品简介:ezh2-in-13 is a potent ezh2 inhibitor with potential anticancer activity.ezh2-in-13 may be used to study diseases associated with ezh2 activity...产品型号:T64043 原产地:中国大陆价格: ¥0.0
产品名称: Mps1-IN-3 hydrochloride;化合物 Mps1-IN-3 hydrochlorideMps1-IN-3 hydrochloride
产品简介:mps1-in-3 hydrochloride is a potent and selective inhibitor of mps1 (ic50: 50 nm). mps1-in-3 hydrochloride exhibits inhibitory effects on the proliferation of g..产品型号:T64061 原产地:中国大陆价格: ¥0.0
产品名称: CSF1R-IN-3;化合物CSF1R-IN-3CSF1R-IN-3
产品简介:csf1r-in-3 is an orally effective csf-1r inhibitor with an ic50 value of 2.1 nm. csf1r-in-3 has anti-proliferative activity against colorectal cancer cells. csf..产品型号:T64066 原产地:中国大陆价格: ¥0.0
产品名称: KIF18A-IN-3;化合物 KIF18A-IN-3KIF18A-IN-3
产品简介:kif18a-in-3 is a potent inhibitor of kif18a with an ic50 value of 61 nm. kif18a-in-3 significantly causes mitotic arrest and increases the number of mitotic cel..产品型号:T64068 原产地:中国大陆价格: ¥0.0
产品名称: β-Lapachone;化合物Beta-LapachoneBeta-Lapachone|||NSC-26326|||SL-11001|||ARQ-501;3,4-二氢-2,2-二甲基-2H-萘并[1,
产品简介:β-lapachone (arq-501) is a specific dna topoisomerase i inhibitor, and no inhibitory activities against dna topoisomerase ii or ligase...产品型号:T6407 原产地:中国大陆价格: ¥0.0
产品名称: Pan-Trk-IN-3;化合物 Pan-Trk-IN-3Pan-Trk-IN-3
产品简介:pan-trk-in-3 is a potent, broad-spectrum inhibitor of trk and its drug-resistant mutants, acting on trka (ic50: 2 nm), trkb (ic50: 3 nm), trkc (ic50: 2 nm), trk..产品型号:T64070 原产地:中国大陆价格: ¥0.0
产品名称: JAK2/FLT3-IN-1 TFA;化合物 JAK2/FLT3-IN-1 TFAJAK2/FLT3-IN-1 TFA
产品简介:jak2/flt3-in-1 (tfa) is an orally active dual inhibitor of jak2/flt3 that exhibits anticancer effects, acting on jak2 (ic50: 0.7 nm), flt3 (ic50: 4 nm), jak1 (i..产品型号:T64104 原产地:中国大陆价格: ¥0.0
产品名称: FGFR3-IN-1;化合物 FGFR3-IN-1FGFR3-IN-1
产品简介:fgfr3-in-1 (compound 1) is a fibroblast growth factor receptor (fgfr) inhibitor that inhibits fgfr1 (ic50: 40 nm), fgfr2 (ic50: 5.1 nm) and fgfr3 (ic50: 12 nm)...产品型号:T64107 原产地:中国大陆价格: ¥0.0
产品名称: AChE/GSK-3β-IN-1;化合物 AChE/GSK-3β-IN-1AChE/GSK-3β-IN-1
产品简介:ache/gsk-3β-in-1 is a potent dual ache/gsk-3β inhibitor that crosses the blood-brain barrier and acts on hache (ic50: 1.2 nm), hbche (ic50: 149.8 nm) and hgsk-3..产品型号:T64143 原产地:中国大陆价格: ¥0.0
产品名称: RORγt/DHODH-IN-3;化合物 RORγt/DHODH-IN-3RORγt/DHODH-IN-3
产品简介:rorγt/dhodh-in-3 (compound (s)-14d) is a potent, orally active dual inhibitor of rorγt (ic50: 0.098 μm) and dhodh (ic50: 0.432 μm).rorγt/dhodh-in-1 has signific..产品型号:T64146 原产地:中国大陆价格: ¥0.0
产品名称: MraY-IN-3;化合物 MraY-IN-3MraY-IN-3
产品简介:mray-in-3 (12a) is a potent inhibitor of the bacterial translocase mray (ic50: 140 μm). 46 μg/ml)...产品型号:T64160 原产地:中国大陆价格: ¥0.0
产品名称: BML-190;吲哚美辛吗啉代酰胺Indomethacin morpholinylamide|||IMMA|||BML 190;2-[1-(4-氯苯甲酰基)-5-甲氧基-2-甲基-1H-吲哚-3-基]
产品简介:bml-190 (indomethacin morpholinylamide) is a specific cb2 receptor inverse agonist (ki: 435 nm), with 50-fold selectivity over cb1 receptor...产品型号:T6417 原产地:中国大陆价格: ¥0.0
产品名称: GLS1 Inhibitor-3;化合物 GLS1 Inhibitor-3GLS1 Inhibitor-3
产品简介:gls1 inhibitor-3 (compound c147) is a potent inhibitor of gls1 (ic50: 27.98 nm) and exhibits anti-proliferative effects...产品型号:T64211 原产地:中国大陆价格: ¥0.0
产品名称: Cap-dependent endonuclease-IN-3;化合物 Cap-dependent endonuclease-IN-3Cap-dependent endonuclease-IN-3
产品简介:cap-dependent endonuclease-in-3 is a potent inhibitor of cap-dependent nucleic acid endonucleases (cen). cap-dependent endonuclease-in-3 has shown potential for..产品型号:T64213 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/mTOR Inhibitor-6;化合物 PI3K/mTOR Inhibitor-6PI3K/mTOR Inhibitor-6
产品简介:pi3k/mtor inhibitor-6 (compound 19c) is a potent dual pi3k/mtor inhibitor that is more stable than gedatolisib in artificial gastric fluid. 10 μm of pi3k/mtor i..产品型号:T64219 原产地:中国大陆价格: ¥0.0