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产品名称: BRAF V600E/CRAF-IN-1;化合物 BRAF V600E/CRAF-IN-1BRAF V600E/CRAF-IN-1
产品简介:braf v600e/craf-in-1 is a potent inhibitor of brafv600e/craf. braf v600e/craf-in-1 acts in the g0/g1 phase of hct-116 colon cancer cells to arrest the cell cycl..产品型号:T63448 原产地:中国大陆价格: ¥0.0
产品名称: HIV-1 protease-IN-1;化合物 HIV-1 protease-IN-1HIV-1 protease-IN-1
产品简介:hiv-1 protease-in-1 is a potent inhibitor of hiv-1 protease (ic50: 90 pm). hiv-1 protease-in-1 has antiviral activity against b-hiv (ec50: 89 nm): hiv-1 proteas..产品型号:T63453 原产地:中国大陆价格: ¥0.0
产品名称: P-gp/BCRP-IN-1;化合物 P-gp/BCRP-IN-1P-gp/BCRP-IN-1
产品简介:p-gp/bcrp-in-1 (compound 19) is a relatively safe, orally active, and efficient inhibitor of the efflux transporters p-gp and bcrp. by inhibiting their efflux f..产品型号:T63267 原产地:中国大陆价格: ¥0.0
产品名称: HPK1-IN-29;化合物 HPK1-IN-29HPK1-IN-29
产品简介:hpk1-in-29 is a potent inhibitor of hpk1, in which hematopoietic progenitor kinase 1 (hpk1) is a negative regulator of the activation response of dendritic cell..产品型号:T63270 原产地:中国大陆价格: ¥0.0
产品名称: HPK1-IN-3;化合物 HPK1-IN-3HPK1-IN-3
产品简介:hpk1-in-3 is a selective, potent, atp-competitive inhibitor of hematopoietic progenitor cell kinase 1 (hpk1; map4k1) (ic50: 0.25 nm). hpk1-in-3 has il-2 cellula..产品型号:T63287 原产地:中国大陆价格: ¥0.0
产品名称: SCP1-IN-2;化合物 SCP1-IN-2SCP1-IN-2
产品简介:scp1-in-2 is a potent, selective, and metric inhibitor of scp1. scp1-in-2 is able to induce rest degradation and inhibit its transcriptional activity. high leve..产品型号:T63288 原产地:中国大陆价格: ¥0.0
产品名称: 3-Aminobenzamide;化合物INO10013-AB|||INO1001|||INO-1001|||3-ABA|||PARP-IN-1|||INO 1001;3-AB|||INO1001||
产品简介:3-aminobenzamide (parp-in-1) is an effective inhibitor of parp (ic50<50 nm in cho cells) and a mediator of oxidant-induced myocyte dysfunction during reperfusio..产品型号:T6329 原产地:中国大陆价格: ¥0.0
产品名称: (R,1R)-Tenofovir amibufenamide;(R,1R)-艾米替诺福韦(R,1R)-HS-10234;(R,1R)-HS-10234
产品简介:(r,1r)-tenofovir amibufenamide ((r,1r)-hs-10234) can be used as a tenofovir prodrug, which can be taken orally and has antiviral activity. tynofovir is a nucleo..产品型号:T63290 原产地:中国大陆价格: ¥0.0
产品名称: MALT1-IN-6;化合物 MALT1-IN-6MALT1-IN-6
产品简介:malt1-in-6 is a malt1 protease inhibitor (ki: 9 nm) that exhibits anticancer activity...产品型号:T63372 原产地:中国大陆价格: ¥0.0
产品名称: S100A2-p53-IN-1;化合物 S100A2-p53-IN-1S100A2-p53-IN-1
产品简介:s100a2-p53-in-1 (compound 51), an inhibitor of s100a2-p53 interactions, targets s100a2, a ca 2+ binding protein involved in cell signaling and commonly upregula..产品型号:T63373 原产地:中国大陆价格: ¥0.0
产品名称: S1PR1 agonist 1;化合物 S1PR1 agonist 1S1PR1 agonist 1
产品简介:s1pr1 agonist 1 is a potent agonist of s1pr1. s1pr1 agonist 1 has potential in autoimmune diseases...产品型号:T63378 原产地:中国大陆价格: ¥0.0
产品名称: DHFR-IN-1;化合物 DHFR-IN-1DHFR-IN-1
产品简介:dhfr-in-1 is a selective and potent inhibitor of dhfr (dihydrofolate reductase) (ic50: 40.71 nm). dhfr-in-1 exhibited some antifungal activity and good antibact..产品型号:T63379 原产地:中国大陆价格: ¥0.0
产品名称: Protease-Activated Receptor-1 antagonist 3;化合物 Protease-Activated Receptor-1 antagonist 3Protease-Ac
产品简介:protease-activated receptor-1 antagonist 3 is a potent antagonist (ic50: 7 nm) of protease-activated receptor 1protease-activated receptor-1. antagonist 3 exhib..产品型号:T63382 原产地:中国大陆价格: ¥0.0
产品名称: Pan-RAF kinase inhibitor 1;化合物 Pan-RAF kinase inhibitor 1Pan-RAF kinase inhibitor 1
产品简介:pan-raf kinase inhibitor 1 is a potent inhibitor of the pan-raf kinase pair that inhibits raf kinase and regulates mapk signaling, thereby affecting the prolife..产品型号:T63386 原产地:中国大陆价格: ¥0.0
产品名称: (S,S)-TAPI-1;化合物 (S,S)-TAPI-1(S,S)-TAPI-1
产品简介:(s,s)-tapi-1 is an isomer of tapi-1. among them, tapi-1 is a metalloproteinase (mmp) inhibitor and a tace (adam17) inhibitor that exhibits potent inhibition of ..产品型号:T63390 原产地:中国大陆价格: ¥0.0
产品名称: ACSS2-IN-1;化合物 ACSS2-IN-1ACSS2-IN-1
产品简介:acss2-in-1 is a potent inhibitor of acss2, capable of inhibiting acss2 activity with ic50 values ranging from 0.01 nm to <1 nm, and can be used in cancer resear..产品型号:T63397 原产地:中国大陆价格: ¥0.0
产品名称: COX-2/sEH-IN-1;化合物 COX-2/sEH-IN-1COX-2/sEH-IN-1
产品简介:cox-2/seh-in-1 is an orally active dual inhibitor of cox-2 (ic50: 1.24 μm) and seh (ic50: 0.40 μm), a soluble epoxide hydrolase. cox-2/seh-in-1 increases anti-i..产品型号:T63398 原产地:中国大陆价格: ¥0.0
产品名称: mTOR/HDAC-IN-1;化合物 mTOR/HDAC-IN-1mTOR/HDAC-IN-1
产品简介:mtor/hdac-in-1 (compound 50) is a dual inhibitor targeting both mtor and hdac with respective ic50 values of 0.49 nm and 0.91 nm. it holds potential as an anti-..产品型号:T63399 原产地:中国大陆价格: ¥0.0
产品名称: mTOR/HDAC-IN-1 HCl;mTOR/HDAC抑制剂1盐酸盐mTOR/HDAC-IN-1 HCl(2815286-02-1 Free base);mTOR/HDAC-IN-1 HCl(281
产品简介:mtor/hdac-in-1 hcl is a potent dual inhibitor of mtor and hdac with potential anti-inflammatory, anti-proliferative, autophagy and apoptosis-inducing effects fo..产品型号:T63399L 原产地:中国大陆价格: ¥0.0
产品名称: hA2A/hCA XII modulator 1;化合物 hA2A/hCA XII modulator 1hA2A/hCA XII modulator 1
产品简介:ha2a/hca xii modulator 1 is a potent antagonist of the ha2a adenosine receptor (ha2aar), a triazolopyrazine that acts on ha2aar (ki: 6.4 nm), ha1ar (ki: 4.819 μ..产品型号:T63400 原产地:中国大陆价格: ¥0.0