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产品名称: VA5 TG2 inhibitor;化合物 T29086VA5|||VA-5|||VA 5;VA5|||VA-5|||VA 5
产品简介:va5 is an transamidase inhibitor by direct binding at the transamidase site. va5 also inhibits gtp-binding activities. it interaction at the transamidase site l..产品型号:T29086 原产地:中国大陆价格: ¥0.0
产品名称: UK-122 TFA salt;化合物 T29051UK122|||uPA Inhibitor II|||UK122 TFA salt|||UK 122|||UK-122|||K122 triflor
产品简介:uk-122 is a potent and selective upa inhibitor (ki = 20 nm). the ic(50) of uk122 in a cell-free indirect upa assay is 0.2 micromol/l. uk122 showed little cytoto..产品型号:T29051 原产地:中国大陆价格: ¥0.0
产品名称: TrxR inhibitor D9;化合物 T29018D9|||TrxR inhibitor D-9|||D-9|||D9|||D9|||TrxR inhibitor D9|||TrxR-IN-D9
产品简介:trxr-in-d9 is a novel inhibitor of thioredoxin reductase (trxr)...产品型号:T29018 原产地:中国大陆价格: ¥0.0
产品名称: Prolyl Endopeptidase Inhibitor 1;化合物 T12546(Boc)-Prolyl-prolinal|||BPP|||Boc-Pro-prolinal;(Boc)-Prol
产品简介:prolyl endopeptidase inhibitor 1 is a potent inhibitor of prolyl endopeptidase (pep; pe)(ki : 15 nm) , has anti-amnesic effect...产品型号:T12546 原产地:中国大陆价格: ¥0.0
产品名称: Prolyl Hydroxylase inhibitor 1;化合物 T12547Prolyl Hydroxylase inhibitor 1
产品简介:prolyl hydroxylase inhibitor 1 is an orally active inhibitor of hypoxia inducible factor (hif)-prolyl hydroxylase (phd) (ic50 of 62.23 nm)...产品型号:T12547 原产地:中国大陆价格: ¥0.0
产品名称: Telomerase-IN-2;端粒酶抑制剂2Telomerase inhibitor 2;Telomerase inhibitor 2|||端粒酶抑制剂2
产品简介:telomerase-in-2 (telomerase inhibitor 2) shows potent inhibitory activity against telomerase by decreasing the expression of dyskerin (ic50: 0.89??m)...产品型号:T13115 原产地:中国大陆价格: ¥0.0
产品名称: β-Secretase Inhibitor IV;化合物 T13434β-Secretase Inhibitor IV
产品简介:β-secretase inhibitor iv is a potent, cell-active inhibitor of bace-1(ic50s of 15.6 and 16.3nm under bace-1 concentrations of 2 nm and 100 pm, respectively)...产品型号:T13434 原产地:中国大陆价格: ¥0.0
产品名称: URAT1 inhibitor 1;化合物 T13259URAT1 inhibitor 1
产品简介:urat1 inhibitor 1 (1g) is an inhibitor of uric acid transporter 1 (urat1) (ic50: 32 nm), has the potential to treat hyperuricemia associated with gout...产品型号:T13259 原产地:中国大陆价格: ¥0.0
产品名称: YAP/TAZ inhibitor-1;化合物 T13364YAP/TAZ inhibitor-1
产品简介:yap/taz inhibitor-1 is an inhibitor of yap/taz (ic50 of <0.100 μμ in firefly luciferase assay)...产品型号:T13364 原产地:中国大陆价格: ¥0.0
产品名称: WDR5-IN-4;化合物 T13342WIN site inhibitor 1;WIN site inhibitor 1
产品简介:win site inhibitor 1 is a win site of chromatin-associated wd repeat-containing protein 5 (wdr5) inhibitor (kd: 0.1 nm), with anti-cancer activity...产品型号:T13342 原产地:中国大陆价格: ¥0.0
产品名称: WIN site inhibitor 1 TFA (2407457-36-5 free base);化合物 T13342LWIN site inhibitor 1 TFA;WIN site inhib
产品简介:win site inhibitor 1 tfa is a win site of chromatin-associated wd repeat-containing protein 5 (wdr5) inhibitor (kd: 0.1 nm)...产品型号:T13342L 原产地:中国大陆价格: ¥0.0
产品名称: Ogerin;化合物OgerinG Protein-Coupled Receptor 68|||Inhibitor|||TGF-β|||inhibit|||Ogerin|||fibroblasts||
产品简介:ogerin is a selective gpr68 positive allosteric modulator (pec50: 6.83). ogerin blocks recall in fear conditioning in mice. ogerin displays inverse agonist and ..产品型号:T16378 原产地:中国大陆价格: ¥0.0
产品名称: NKY80化合物NKY80Adenylyl cyclase type V Inhibitor
产品简介:nky80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues. nky80 is a non-competitive inhibitor of adenylyl cyclase type v isoform (ic5..产品型号:T16333 原产地:中国大陆价格: ¥0.0
产品名称: Notch inhibitor 1;化合物 T16341Notch inhibitor 1
产品简介:notch inhibitor 1 is an effective notch inhibitor (ic50s: 7.8 and 8.5 nm for notch 1 and notch 3, respectively). notch inhibitor 1 is also used in the research ..产品型号:T16341 原产地:中国大陆价格: ¥0.0
产品名称: PIN1 inhibitor API-1;化合物PIN1 inhibitor API-1PIN1 inhibitor API-1
产品简介:pin1 inhibitor api-1 is a specific pin1 inhibitor (ic50: 72.3 nm). pin1 inhibitor api-1 retains the active conformation of pxpo5 and restores the ability of pxp..产品型号:T16538 原产地:中国大陆价格: ¥0.0
产品名称: BEBT-908;化合物BEBT-908PI3Kα inhibitor 1|||MDK9521;PI3Kα inhibitor 1|||MDK9521
产品简介:bebt-908 (pi3kα inhibitor 1) is a selective pi3kα inhibitor (ic50 <0.1 μm). bebt-908 also inhibits hdac (0.1 μm≤ic50≤1 μm)...产品型号:T16529 原产地:中国大陆价格: ¥0.0
产品名称: p32 Inhibitor M36化合物 T16423M36
产品简介:p32 inhibitor m36 is an inhibitor of p32 mitochondrial protein. it binds directly to p32 and inhibits the p32 association with lyp-1...产品型号:T16423 原产地:中国大陆价格: ¥0.0
产品名称: Cbz-NH-PEG3-CH2COOH;苯甲氧羰酰基二聚乙二醇羧乙基Inhibitor|||PROTAC Linkers|||inhibit|||CbzNHPEG3CH2COOH|||Cbz-NH-P
产品简介:cbz-nh-peg3-ch2cooh is a peg-based protac linker that can be used in protac synthesis...产品型号:T17722 原产地:中国大陆价格: ¥0.0
产品名称: OTSSP167;化合物OTSSP167MELK inhibitor|||OTS167;MELK inhibitor|||OTS167
产品简介:otssp167 (ots167) is an orally available inhibitor of maternal embryonic leucine zipper kinase (melk) with potential antineoplastic activity...产品型号:T1759 原产地:中国大陆价格: ¥0.0
产品名称: PEG3-O-CH2COOH;三聚乙二醇-乙酸PROTAC Linker 8|||PEG3OCH2COOH|||PEG-3-O-CH2COOH|||Inhibitor|||PROTAC Linker8
产品简介:peg3-o-ch2cooh (protac linker 8) (protac linker 8) is a peg-based protac linker. peg3-o-ch2cooh can be used in the synthesis of snipers...产品型号:T18629 原产地:中国大陆价格: ¥0.0