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产品名称: Vadimezan;伐地美生DMXAA|||5,6-Dimethylxanthenone-4-acetic Acid|||NSC 640488|||ASA-404;DMXAA|||伐地美生|||5,6
产品简介:vadimezan (dmxaa) is a vascular disrupting agent, a murine sting agonist, and an inducer of cytokines such as type i ifn. vadimezan has antitumor activity and i..产品型号:T6273 原产地:中国大陆价格: ¥0.0
产品名称: S1P1 agonist 5;化合物 S1P1 agonist 5S1P1 agonist 5
产品简介:s1p1 agonist 5 is a selective, orally active s1p1 agonist. s1p1 agonist 5 inhibits the drainage of lymphocytes from lymphoid tissue into peripheral blood. s1p1 ..产品型号:T62732 原产地:中国大陆价格: ¥0.0
产品名称: Mu opioid receptor antagonist 5;化合物 Mu opioid receptor antagonist 5Mu opioid receptor antagonist 5
产品简介:mu opioid receptor antagonist 5 (compound nap) is a selective mu opioid receptor (mor) antagonist that crosses the blood-brain barrier (ec50: 1.14 nm, ki: 0.37 ..产品型号:T62673 原产地:中国大陆价格: ¥0.0
产品名称: α5β1 integrin agonist-1;化合物 α5β1?integrin agonist-1α5β1 integrin agonist-1
产品简介:α5β1 integrin agonist-1 is an α5β1 integrin agonist that selectively delivers 5-fu to tumour cells and induces tumour cell death...产品型号:T63868 原产地:中国大陆价格: ¥0.0
产品名称: RAD51-IN-5;化合物 RAD51-IN-5RAD51-IN-5
产品简介:rad51-in-5 is a potent inhibitor of rad51. rad51-in-5 has shown potential for the study of mitochondrial deficiency disorders...产品型号:T63892 原产地:中国大陆价格: ¥0.0
产品名称: Benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)-;化合物
产品简介:benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αr)- is a dual pparα/γ agonist with ec50 of 0.358μm and 1.21μm. benz..产品型号:T63898 原产地:中国大陆价格: ¥0.0
产品名称: RECQL5-IN-1;化合物 RECQL5-IN-1RECQL5-IN-1
产品简介:recql5-in-1 is an orally active inhibitor of recql5 (targeting both enzymatic and non-enzymatic domains) and is a potent inhibitor of recql5 decapping activity ..产品型号:T63899 原产地:中国大陆价格: ¥0.0
产品名称: PDE5/HDAC-IN-1;化合物 PDE5/HDAC-IN-1PDE5/HDAC-IN-1
产品简介:pde5/hdac-in-1 is a potent inhibitor of phosphodiesterase 5 (pde5) and hdac, with ic50 values of 46.3 nm and 14.5 nm, respectively...产品型号:T63907 原产地:中国大陆价格: ¥0.0
产品名称: Cap-dependent endonuclease-IN-5;化合物 Cap-dependent endonuclease-IN-5Cap-dependent endonuclease-IN-5
产品简介:cap-dependent endonuclease-in-5 is a potent inhibitor of cap-dependent nucleic acid endonucleases (cen). cap-dependent endonuclease-in-5 has good influenza viru..产品型号:T63910 原产地:中国大陆价格: ¥0.0
产品名称: ERα degrader 5;化合物 ERα degrader 5ERα degrader 5
产品简介:erα degrader 5 is an orally active, selective estrogen receptor (er) reducer that acts on erα (ec50: 1.1 nm). erα degrader 5 shows anti-tumour effects in vivo...产品型号:T63922 原产地:中国大陆价格: ¥0.0
产品名称: ATR-IN-5;化合物 ATR-IN-5ATR-IN-5
产品简介:atr-in-5 is a potent inhibitor of atr, a member of the pikk family of proteins involved in genome stability and dna damage repair. atr is a member of the pikk f..产品型号:T63923 原产地:中国大陆价格: ¥0.0
产品名称: AS-604850化合物AS6048505-[(2,2-二氟-1,3-苯并二恶茂-5-基)亚甲基]噻唑烷-2,4-二酮
产品简介:as-604850 is a specific and atp-competitive pi3kγ inhibitor (ic50: 250 nm), 18-fold more selective for pi3kγ than pi3kα, and over 80-fold selectivity for pi3kγ ..产品型号:T6394 原产地:中国大陆价格: ¥0.0
产品名称: FTO-IN-5;化合物 FTO-IN-5FTO-IN-5
产品简介:fto-in-5 is a potent, selective inhibitor targeting the fat mass obesity-associated protein (fto)...产品型号:T63843 原产地:中国大陆价格: ¥0.0
产品名称: AGK2化合物AGK22-氰基-3-[5-(2,5-二氯苯基)-2-呋喃基]-N-5-喹啉基-2-丙烯酰胺
产品简介:agk2(ic50=3.5 μm) is an effective, and specific sirt2 inhibitor...产品型号:T6371 原产地:中国大陆价格: ¥0.0
产品名称: Sirt2-IN-5;化合物 Sirt2-IN-5Sirt2-IN-5
产品简介:sirt2-in-5 is a potent inhibitor of sirt2...产品型号:T63712 原产地:中国大陆价格: ¥0.0
产品名称: IRE1α kinase-IN-5;化合物 IRE1α kinase-IN-5IRE1α kinase-IN-5
产品简介:ire1α kinase-in-5 (compound 7) is a potent inhibitor of ire1α (ki: 98 nm) and is an atp-competitive ligand for ire1α...产品型号:T63734 原产地:中国大陆价格: ¥0.0
产品名称: WDR5-IN-5;化合物 WDR5-IN-5WDR5-IN-5
产品简介:wdr5-in-5 is a selective, orally active inhibitor targeting the wd repeat domain 5 (wdr5) win site.wdr5-in-5 exhibits high affinity for wdr5 (ki<0.02 nm).wdr5-i..产品型号:T63763 原产地:中国大陆价格: ¥0.0
产品名称: L5-DA;化合物 L5-DAL5-DA
产品简介:l5-da is a g-quadruplex (g4) ligand that selectively stabilizes g4s. l5-da exhibits significant cytotoxicity to hela cells with an ic50 value of 4.3 μm. l5-da s..产品型号:T63765 原产地:中国大陆价格: ¥0.0
产品名称: RET-IN-5;化合物 RET-IN-5RET-IN-5
产品简介:ret-in-5 is a potent inhibitor of ret (ic50: 4.57 nm)...产品型号:T63772 原产地:中国大陆价格: ¥0.0
产品名称: SOS1-IN-5;化合物 SOS1-IN-5SOS1-IN-5
产品简介:sos1-in-5 is a pyrimidine bicyclic derivative and a potent inhibitor of sos1. sos1-in-5 interferes with the ras-sos1 interaction, thereby blocking kras activati..产品型号:T63781 原产地:中国大陆价格: ¥0.0