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产品名称: BRD4-BD1-IN-1;化合物 BRD4-BD1-IN-1BRD4-BD1-IN-1
产品简介:brd4-bd1-in-1 (compound 9a) is a brd4-bd1 inhibitor(ic50= 38.20 μm)...产品型号:T62030 原产地:中国大陆价格: ¥0.0
产品名称: Dyrk1A/B-IN-1;化合物 Dyrk1A/B-IN-1Dyrk1A/B-IN-1
产品简介:dyrk1a/b-in-1 (compound 3n) is a potent, selective and cell-permeable inhibitor of dyrk1a and dyrk1b. dyrk1a/b-in-1 inhibits dyrk1a and dyrk1b with kis of 67.8 ..产品型号:T62043 原产地:中国大陆价格: ¥0.0
产品名称: pan-HER-IN-1;化合物 pan-HER-IN-1pan-HER-IN-1
产品简介:pan-her-in-1 (compound c5) is an irreversible, orally active pan- her inhibitor. pan-her-in-1 exhibits ic 50s of 0.38, 1.6, 2.2 and 3.5 nm for egfr, her4, egfr ..产品型号:T62047 原产地:中国大陆价格: ¥0.0
产品名称: Topo I-IN-1;化合物 Topo I-IN-1Topo I-IN-1
产品简介:topo i-in-1 (compound 14d) is a potent topo i inhibitor. topo i-in-1 exhibits antitumor activity and dna intercalative capability. topo i-in-1 can induce cell a..产品型号:T62048 原产地:中国大陆价格: ¥0.0
产品名称: NVS-BET-1;化合物 NVS-BET-1NVS-BET-1
产品简介:nvs-bet-1 is a bet bromodomain inhibitor. nvs-bet-1 can regulate keratinocyte plasticity...产品型号:T62055 原产地:中国大陆价格: ¥0.0
产品名称: TLR9-IN-1;化合物 TLR9-IN-1TLR9-IN-1
产品简介:tlr9-in-1 is a selective and potent tlr9 inhibitor that acts on human tlr9 (ic50: 7 nm). tlr9-in-1 can be used in the study of adverse immune response-related d..产品型号:T62254 原产地:中国大陆价格: ¥0.0
产品名称: GPR84 antagonist 1;化合物 GPR84 antagonist 1GPR84 antagonist 1
产品简介:gpr84 antagonist 1 is a highly selective, high-affinity competitive antagonist of human gpr84...产品型号:T62261 原产地:中国大陆价格: ¥0.0
产品名称: PPARα agonist 1;化合物 PPARα agonist 1PPARα agonist 1
产品简介:pparα agonist 1 is a complete and potent pparα agonist...产品型号:T62266 原产地:中国大陆价格: ¥0.0
产品名称: μ opioid receptor agonist 1;化合物 μ opioid receptor agonist 1μ opioid receptor agonist 1
产品简介:μ opioid receptor agonist 1 (compound h-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an mor receptor agonist that can b..产品型号:T62268 原产地:中国大陆价格: ¥0.0
产品名称: PARP-1-IN-2;化合物PARP-1-IN-2PARP-1-IN-2
产品简介:parp-1-in-2 is a potent parp1 inhibitor that crosses the blood-brain barrier (ic50: 149 nm).parp-1-in-2 showed significant antiproliferative activity against th..产品型号:T62281 原产地:中国大陆价格: ¥0.0
产品名称: JAK1-IN-9;化合物 JAK1-IN-9JAK1-IN-9
产品简介:jak1-in-9 (compound 23a) is a potent, selective inhibitor of jak1, demonstrating an ic50 of 72 nm. it exhibits over 12-fold selectivity against other jak family..产品型号:T62155 原产地:中国大陆价格: ¥0.0
产品名称: HIV-1 integrase inhibitor 9;化合物 HIV-1 integrase inhibitor 9HIV-1 integrase inhibitor 9
产品简介:hiv-1 integrase inhibitor 9 (compound 8a) is a potent inhibitor of hiv-1 rnase h (ic50: 12.3 μm) and has antiviral effects...产品型号:T62156 原产地:中国大陆价格: ¥0.0
产品名称: Bim-IN-1;化合物 Bim-IN-1Bim-IN-1
产品简介:bim-in-1 is a potent inhibitor of bim expression with low toxicity, bim-in-1 reduces bim expression levels with little inhibition of protein kinase a...产品型号:T62157 原产地:中国大陆价格: ¥0.0
产品名称: ALPK1-IN-2;化合物 ALPK1-IN-2ALPK1-IN-2
产品简介:alpk1-in-2 is a potent inhibitor of alpk1 (α-kinase 1) (ic50: 95 nm). alpk1-in-2 inhibits nf-κb (ic50: 1.31 μm)...产品型号:T62162 原产地:中国大陆价格: ¥0.0
产品名称: TNK2-IN-1;化合物 TNK2-IN-1TNK2-IN-1
产品简介:tnk2-in-1 is a tnk2 inhibitor (ic50: 224 nm) that can be used in cancer research...产品型号:T62164 原产地:中国大陆价格: ¥0.0
产品名称: HDAC8/BRPF1-IN-1;化合物 HDAC8/BRPF1-IN-1HDAC8/BRPF1-IN-1
产品简介:hdac8/brpf1-in-1 (compound 23a) is a dual hdac8 and brpf1 inhibitor that acts on human hdac8 (ic50: 443 nm) and human brpf1 (kd: 67 nm). hdac8/brpf1-in-1 has lo..产品型号:T62171 原产地:中国大陆价格: ¥0.0
产品名称: Dual AChE-MAO B-IN-1;化合物 Dual AChE-MAO B-IN-1Dual AChE-MAO B-IN-1
产品简介:dual ache-mao b-in-1 (compound 15) is a safe, metabolically stable neuroprotective agent.dual ache-mao b-in-1 is a potent, orally active cns-permeable inhibitor..产品型号:T62172 原产地:中国大陆价格: ¥0.0
产品名称: GPR41 agonist-1;化合物 GPR41 agonist-1GPR41 agonist-1
产品简介:gpr41 agonist-1 (compound 9) is a potent agonist of gpr41 and can be used in studies of insulin-related diseases...产品型号:T62173 原产地:中国大陆价格: ¥0.0
产品名称: Protein deglycase DJ-1 against-1;化合物 Protein deglycase DJ-1 against-1Protein deglycase DJ-1 against-
产品简介:protein deglycase dj-1 against-1 is a dj-1-binding compound that crosses the blood-brain barrier and targets dj1 in a dependent manner. protein deglycase dj-1 a..产品型号:T62174 原产地:中国大陆价格: ¥0.0
产品名称: POLA1 inhibitor 1;化合物 POLA1 inhibitor 1POLA1 inhibitor 1
产品简介:pola1 inhibitor 1 (compound 12) is an orally active inhibitor of pola1. pola1 inhibitor 1 exhibits antitumour effects on several tumour tissue types and adarote..产品型号:T62176 原产地:中国大陆价格: ¥0.0