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产品名称: AT1R antagonist 1;化合物 AT1R antagonist 1AT1R antagonist 1
产品简介:at1r antagonist 1 (compound 10) serves as a potent, selective ligand for at1r with considerable affinity, demonstrated by a k i value of 8.5 nm [1]...产品型号:T72606 原产地:中国大陆价格: ¥0.0
产品名称: GCGR antagonist 2;化合物 GCGR antagonist 2GCGR antagonist 2
产品简介:gcgr antagonist 2, a furan-2-carbohydrazide, serves as an orally active antagonist of the glucagon receptor. it exhibits affinity for the human glucagon recepto..产品型号:T72621 原产地:中国大陆价格: ¥0.0
产品名称: LTB4 antagonist 1;化合物 LTB4 antagonist 1LTB4 antagonist 1
产品简介:ltb4 antagonist 1, a carboxamide-acid derivative, potently inhibits leukotriene b4 (ltb4) activity with an ic50 value of 288 nm and exhibits notable anti-inflam..产品型号:T72625 原产地:中国大陆价格: ¥0.0
产品名称: A2AR-antagonist-1;化合物 A2AR-antagonist-1A2AR-antagonist-1
产品简介:a2ar-antagonist-1 (compound 38), an orally active adenosine a2a receptor antagonist with an ic50 value of 29 nm, demonstrates anti-tumor properties and stabilit..产品型号:T72626 原产地:中国大陆价格: ¥0.0
产品名称: CU-CPT-8m;化合物CU-CPT-8mTLR8-specific antagonist;TLR8-specific antagonist
产品简介:cu-cpt-8m (tlr8-specific antagonist) is an toll-like receptor 8 (tlr8) antagonist (ic50 : 67 nm)..产品型号:T7347 原产地:中国大陆价格: ¥0.0
产品名称: EP2 receptor antagonist-2;EP2受体拮抗剂2EP2 receptor antagonist-2
产品简介:ep2 receptor antagonist-2 (cid891729) is a compound that not only serves as an antagonist to the ep2 receptor, blocking its activation by pge2, but also reduces..产品型号:T67946 原产地:中国大陆价格: ¥0.0
产品名称: Y2-Antagonist-2;化合物 Y2-Antagonist-2Y2-Antagonist-2
产品简介:y2-antagonist-2 is a novel, selective, soluble non-?peptidic npy y2 receptor antagonist with enhanced cns exposure...产品型号:T71091 原产地:中国大陆价格: ¥0.0
产品名称: P2X7 receptor antagonist-3;化合物 P2X7 receptor antagonist-3P2X7 receptor antagonist-3
产品简介:p2x7 receptor antagonist-3 is a powerful inhibitor of the p2x7 receptor, exhibiting ic50 values of 4.2 nm in humans and 6.8 nm in rats, indicating its high pote..产品型号:T72198 原产地:中国大陆价格: ¥0.0
产品名称: NK1 receptor antagonist 2;化合物 NK1 receptor antagonist 2NK1 receptor antagonist 2
产品简介:nk1 receptor antagonist 2, a compound targeting the nk1 receptor, holds potential for tinnitus and hearing loss research...产品型号:T72224 原产地:中国大陆价格: ¥0.0
产品名称: Sortilin antagonist 1;化合物 Sortilin antagonist 1Sortilin antagonist 1
产品简介:sortilin antagonist 1, a potent sortilin antagonist, exhibits an inhibition constant (ic50) of 20 nm against neurotensin (nts) binding to sortilin. neurotensin ..产品型号:T72410 原产地:中国大陆价格: ¥0.0
产品名称: ADRA1D receptor antagonist 1 free base;化合物 ADRA1D receptor antagonist 1 free baseADRA1D receptor ant
产品简介:adra1d receptor antagonist 1 (free base) antagonist ( k i =1.6 nm). adra1d receptor antagonist 1 (free base) dose-dependently inhibits bladder contraction with..产品型号:T72091 原产地:中国大陆价格: ¥0.0
产品名称: NOD1/2 antagonist-1;化合物 NOD1/2 antagonist-1NOD1/2 antagonist-1
产品简介:nod1/2 antagonist-1 is a potent dual inhibitor of nucleotide-binding oligomerization domain-like receptors 1 and 2 (nod1/2), displaying inhibitory concentration..产品型号:T72473 原产地:中国大陆价格: ¥0.0
产品名称: CU-CPT9b;化合物CU-CPT9bCU-CPT-9b|||TLR8-specific antagonist 1;CU-CPT-9b|||TLR8-specific antagonist 1
产品简介:cu-cpt9b (tlr8-specific antagonist 1) is an antagonist of toll-like receptor 8 (tlr8; kd = 21 nm). it inhibits activation of nf- b induced by the tlr8 agonist r..产品型号:T7302 原产地:中国大陆价格: ¥0.0
产品名称: AZD-4818;化合物AZD-4818CCR1 antagonist;CCR1 antagonist
产品简介:azd-4818 (ccr1 antagonist) is a chemokine ccr1 antagonist for the treatment of chronic obstructive pulmonary disease...产品型号:T30258 原产地:中国大陆价格: ¥0.0
产品名称: Hedgehog Antagonist VIII;Hedgehog Antagonist VIIIHedgehog Antagonist VIII
产品简介:hedgehog (hh) proteins, important regulators of development, bind the cell-surface protein patched, allowing activation of smoothened. in vertebrates, this ulti..产品型号:T35537 原产地:中国大陆价格: ¥0.0
产品名称: Glucagon Receptor Antagonist Inactive Control;Glucagon Receptor Antagonist Inactive ControlGlucagon
产品简介:glucagon receptor antagonist inactive control is a glucagon receptor antagonist that can be used in related research in the field of life sciences. its product ..产品型号:T36580 原产地:中国大陆价格: ¥0.0
产品名称: CDK9 Antagonist-1;CDK9 Antagonist-1CDK9 Antagonist-1;CDK9 Antagonist-1
产品简介:cdk9 antagonist-1 (compounds 11c) is a potent and selective cdk9 degrader based on protac, with an ic50 of 17 μm in mcf-7 cell lines. natural product wogonin bi..产品型号:T36744 原产地:中国大陆价格: ¥0.0
产品名称: A2A receptor antagonist 1;化合物A2A receptor antagonist 1CPI-444 analog|||A2A receptor antagonist 1;CPI
产品简介:a2a receptor antagonist 1 (cpi-444 analog) is an antagonist of both adenosine a2a receptor and a1 receptor with kis of 4 and 264 nm, respectively...产品型号:T37792 原产地:中国大陆价格: ¥0.0
产品名称: A2B receptor antagonist 2;化合物A2B receptor antagonist 2A2B receptor antagonist 2;A2B receptor antagon
产品简介:a2b receptor antagonist 2 is an antagonist of adenosine receptor a2b (ki = 2.30 μm for ra1, 6.8 μm for ra2a, 3.44 μm for ha2b)...产品型号:T37793 原产地:中国大陆价格: ¥0.0
产品名称: mGluR2 antagonist 1;mGluR2 antagonist 1mGluR2 antagonist 1
产品简介:mglur2 antagonist 1 is a potent and selective class of negative allosteric modulator targeting the metabotropic glutamate receptor 2 (mglur2) with high oral bio..产品型号:T38910 原产地:中国大陆价格: ¥0.0