联系我们
产品目录
产品展示/Products
产品名称: PROTAC CDK12/13 Degrader-1;化合物 PROTAC CDK12/13 Degrader-1PROTAC CDK12/13 Degrader-1
产品简介:protac cdk12/13 degrader-1 (7f) is a potent and selective dual degrader of the cell cycle protein-dependent kinases cdk12 (dc50: 2.2 nm) and cdk13 (dc50: 2.1 nm..产品型号:T64284 原产地:中国大陆价格: ¥0.0
产品名称: Protease-Activated Receptor-1 antagonist 2;化合物 Protease-Activated Receptor-1 antagonist?2Protease-Ac
产品简介:protease-activated receptor-1 antagonist 2 is a selective, orally active protease-activated receptor-1 (par-1) antagonist (ic50: 7 nm). it has shown good pharma..产品型号:T64285 原产地:中国大陆价格: ¥0.0
产品名称: sEH inhibitor-1;化合物 sEH inhibitor-1sEH inhibitor-1
产品简介:seh inhibitor-1 (compound tcpu) is a potent, orally active inhibitor of soluble epoxide hydrolase (seh) with ic50 values of 0.4 and 5.3 nm for human and murine ..产品型号:T64291 原产地:中国大陆价格: ¥0.0
产品名称: HIV-1 protease-IN-5;化合物 HIV-1 protease-IN-5HIV-1 protease-IN-5
产品简介:hiv-1 protease-in-5 is an hiv-1 protease inhibitor (ic50: 1.64 nm). hiv-1 protease-in-5 exhibits significant effects on wild-type and drv-resistant hiv-1...产品型号:T64112 原产地:中国大陆价格: ¥0.0
产品名称: BRD4-BD1-IN-2;BRD4-BD1抑制剂2BRD4-BD1-IN-2
产品简介:brd4-bd1-in-2 is a selective and potent brd4-bd1 inhibitor with an ic50 value of 2.51 ?m, which is 20-fold greater than the inhibitory activity against brd4-bd2..产品型号:T64117 原产地:中国大陆价格: ¥0.0
产品名称: AT1R antagonist 2;化合物 AT1R antagonist 2AT1R antagonist 2
产品简介:at1r antagonist 2 is a potent at1r selective ligand with good at1r affinity (ki: 26 nm)...产品型号:T64122 原产地:中国大陆价格: ¥0.0
产品名称: HIV-1 inhibitor-17;化合物 HIV-1 inhibitor-17HIV-1 inhibitor-17
产品简介:hiv-1 inhibitor-18 is a potent inhibitor of the hiv-1 capsid and is able to act on the hiv-1 nl4-3 strain (ec50: 2.57 μm). hiv-1 inhibitor-18 exhibits some cyto..产品型号:T64131 原产地:中国大陆价格: ¥0.0
产品名称: Cap-dependent endonuclease-IN-16;化合物 Cap-dependent endonuclease-IN-16Cap-dependent endonuclease-IN-1
产品简介:cap-dependent endonuclease-in-16 is a pyridone polycyclic derivative and a potent inhibitor of cap-dependent nucleic acid endonucleases (cen). cap-dependent end..产品型号:T64138 原产地:中国大陆价格: ¥0.0
产品名称: Lipid-lowering agent-1;化合物 Lipid-lowering agent-1Lipid-lowering agent-1
产品简介:lipid-lowering agent-1 is a potent lipid-lowering agent that significantly inhibits the pharmacological effects of low-density lipoprotein cholesterol (ldlc) an..产品型号:T64006 原产地:中国大陆价格: ¥0.0
产品名称: GLP-1R agonist 10;化合物 GLP-1R agonist 10GLP-1R agonist 10
产品简介:glp-1r agonist 10 is a glp-1 agonist (ec50: 0.051 nm)...产品型号:T64007 原产地:中国大陆价格: ¥0.0
产品名称: HIV-1 inhibitor-23;化合物 HIV-1 inhibitor-23HIV-1 inhibitor-23
产品简介:hiv-1 inhibitor-23 is a highly potent inhibitor of hiv-1 non-nucleoside reverse transcriptase, acting on both wild-type hiv-1 (ec50: 24.9 nm) and mutant strain ..产品型号:T64009 原产地:中国大陆价格: ¥0.0
产品名称: Dopamine D3 receptor antagonist-1;化合物 Dopamine D3 receptor antagonist-1Dopamine D3 receptor antagoni
产品简介:dopamine d3 receptor antagonist-1 is a dopamine d3 receptor selective or multi-targeting ligand with a ki value of 1.58 nm that has demonstrated therapeutic pot..产品型号:T64024 原产地:中国大陆价格: ¥0.0
产品名称: ERα antagonist 1;化合物 ERα antagonist 1ERα antagonist 1
产品简介:erα antagonist 1 is a selective, potent, covalent estrogen receptor alpha (erα) antagonist that blocks the cell cycle of mcf-7 cells in g0/g1 phase and induces ..产品型号:T64026 原产地:中国大陆价格: ¥0.0
产品名称: 5-HT6R/MAO-B modulator 1;化合物 5-HT6R/MAO-B modulator 15-HT6R/MAO-B modulator 1
产品简介:5-ht6r/mao-b modulator 1 is an antagonist of 5-ht6r at gs signaling and an irreversible inhibitor of mao-b that exhibits glial protective activity. 5-ht6r/mao-b..产品型号:T64036 原产地:中国大陆价格: ¥0.0
产品名称: PLK1/BRD4-IN-1;化合物 PLK1/BRD4-IN-1PLK1/BRD4-IN-1
产品简介:plk1/brd4-in-1 (9b) is an orally active dual inhibitor of plk1 (ic50: 22 nm) and brd4 (ic50: 109 nm). it has been shown to have good anti-tumour effects in vivo..产品型号:T64058 原产地:中国大陆价格: ¥0.0
产品名称: Mps1-IN-3 hydrochloride;化合物 Mps1-IN-3 hydrochlorideMps1-IN-3 hydrochloride
产品简介:mps1-in-3 hydrochloride is a potent and selective inhibitor of mps1 (ic50: 50 nm). mps1-in-3 hydrochloride exhibits inhibitory effects on the proliferation of g..产品型号:T64061 原产地:中国大陆价格: ¥0.0
产品名称: RIPK1-IN-10;化合物 RIPK1-IN-10RIPK1-IN-10
产品简介:ripk1-in-10 is a potent inhibitor of ripk1...产品型号:T64064 原产地:中国大陆价格: ¥0.0
产品名称: CSF1R-IN-3;化合物CSF1R-IN-3CSF1R-IN-3
产品简介:csf1r-in-3 is an orally effective csf-1r inhibitor with an ic50 value of 2.1 nm. csf1r-in-3 has anti-proliferative activity against colorectal cancer cells. csf..产品型号:T64066 原产地:中国大陆价格: ¥0.0
产品名称: β-Lapachone;化合物Beta-LapachoneBeta-Lapachone|||NSC-26326|||SL-11001|||ARQ-501;3,4-二氢-2,2-二甲基-2H-萘并[1,
产品简介:β-lapachone (arq-501) is a specific dna topoisomerase i inhibitor, and no inhibitory activities against dna topoisomerase ii or ligase...产品型号:T6407 原产地:中国大陆价格: ¥0.0
产品名称: BACE1-IN-8;化合物 BACE1-IN-8BACE1-IN-8
产品简介:bace1-in-8 is a potent inhibitor of bace1 (β-site app lyase 1) (ic50: 3.9 μm)...产品型号:T64074 原产地:中国大陆价格: ¥0.0