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产品名称: Spermine Prodrug-1;化合物 Spermine Prodrug-1Spermine Prodrug-1
产品简介:spermine prodrug-1 is a redox-sensitive spermine prodrug. spermine prodrug-1 inhibits wild-type (cms-24949) and spermine synthase gene (sms) mutant (cms-26559, ..产品型号:T64076 原产地:中国大陆价格: ¥0.0
产品名称: Mutant p53 modulator-1;化合物 Mutant p53 modulator-1Mutant p53 modulator-1
产品简介:mutant p53 modulator-1 is a mutant p53 modulator. mutant p53 modulator-1 is able to hinder the progression of cancers containing p53 mutations...产品型号:T64079 原产地:中国大陆价格: ¥0.0
产品名称: PD-1/PD-L1-IN-20;化合物 PD-1/PD-L1-IN-20PD-1/PD-L1-IN-20
产品简介:pd-1/pd-l1-in-20 is a small molecule inhibitor of pd-1/pd-l1 protein-protein interaction. pd-1/pd-l1-in-20 blocks the pd-1/pd-l1 interaction (ic50: 5.29 nm). pd..产品型号:T64086 原产地:中国大陆价格: ¥0.0
产品名称: BRD4 D1-IN-1;化合物 BRD4 D1-IN-1BRD4 D1-IN-1
产品简介:brd4 d1-in-1 is a selective inhibitor of brd4 d1 with an ic50 <0.092 μm. brd4 d1-in-1 has an affinity of 18 nm and over 500-fold selectivity for brd4 d1 and brd..产品型号:T64089 原产地:中国大陆价格: ¥0.0
产品名称: ALK kinase inhibitor-1;化合物SAR348830SAR348830;SAR348830
产品简介:sar348830 is an alk inhibitor, targeting anaplastic lymphoma kinase...产品型号:T6409 原产地:中国大陆价格: ¥0.0
产品名称: JAK2/FLT3-IN-1 TFA;化合物 JAK2/FLT3-IN-1 TFAJAK2/FLT3-IN-1 TFA
产品简介:jak2/flt3-in-1 (tfa) is an orally active dual inhibitor of jak2/flt3 that exhibits anticancer effects, acting on jak2 (ic50: 0.7 nm), flt3 (ic50: 4 nm), jak1 (i..产品型号:T64104 原产地:中国大陆价格: ¥0.0
产品名称: FGFR3-IN-1;化合物 FGFR3-IN-1FGFR3-IN-1
产品简介:fgfr3-in-1 (compound 1) is a fibroblast growth factor receptor (fgfr) inhibitor that inhibits fgfr1 (ic50: 40 nm), fgfr2 (ic50: 5.1 nm) and fgfr3 (ic50: 12 nm)...产品型号:T64107 原产地:中国大陆价格: ¥0.0
产品名称: AChE/GSK-3β-IN-1;化合物 AChE/GSK-3β-IN-1AChE/GSK-3β-IN-1
产品简介:ache/gsk-3β-in-1 is a potent dual ache/gsk-3β inhibitor that crosses the blood-brain barrier and acts on hache (ic50: 1.2 nm), hbche (ic50: 149.8 nm) and hgsk-3..产品型号:T64143 原产地:中国大陆价格: ¥0.0
产品名称: FXR antagonist 1;化合物 FXR antagonist 1FXR antagonist 1
产品简介:fxr antagonist 1 is a selective, orally active intestinal fxr antagonist with an ic50 value of 2.1 μm. fxr antagonist 1 antagonises intestinal fxr and selective..产品型号:T64144 原产地:中国大陆价格: ¥0.0
产品名称: RORγt/DHODH-IN-1;化合物 RORγt/DHODH-IN-1RORγt/DHODH-IN-1
产品简介:rorγt/dhodh-in-1 (compound (r)-14d) is a potent, orally active dual inhibitor of rorγt (ic50: 0.083 μm) and dhodh (ic50: 0.172 μm), which exhibits significant i..产品型号:T64145 原产地:中国大陆价格: ¥0.0
产品名称: ERK1/2 inhibitor 6;化合物 ERK1/2 inhibitor 6ERK1/2 inhibitor 6
产品简介:erk1/2 inhibitor 6 is a potent inhibitor of erk1/2. erk1/2 inhibitor 6 has shown potential for the study or prevention of cancer, inflammation or other prolifer..产品型号:T64147 原产地:中国大陆价格: ¥0.0
产品名称: Glyoxalase I inhibitor 1;化合物 Glyoxalase I inhibitor 1Glyoxalase I inhibitor 1
产品简介:glyoxalase i inhibitor 1 is a potent inhibitor of glyoxalase i (glo1) (ic50: 26 nm)...产品型号:T64153 原产地:中国大陆价格: ¥0.0
产品名称: CYP51/HDAC-IN-1;化合物 CYP51/HDAC-IN-1CYP51/HDAC-IN-1
产品简介:cyp51/hdac-in-1 is an orally active, potent, dual cyp51/hdac inhibitor that inhibits important virulence factors and down-regulates the expression of associated..产品型号:T64154 原产地:中国大陆价格: ¥0.0
产品名称: AChE/BChE-IN-1;化合物 AChE/BChE-IN-1AChE/BChE-IN-1
产品简介:ache/bche-in-1 is a potent dual inhibitor of acetylcholinesterase and butyrylcholinesterase with blood-brain barrier permeability, exhibiting an ic50 value of 1..产品型号:T64156 原产地:中国大陆价格: ¥0.0
产品名称: XIAP degrader-1;化合物 XIAP degrader-1XIAP degrader-1
产品简介:xiap degrader-1 is a small primary amine molecule that promotes the degradation of x-linked apoptosis inhibitory protein (xiap)...产品型号:T64161 原产地:中国大陆价格: ¥0.0
产品名称: BML-190;吲哚美辛吗啉代酰胺Indomethacin morpholinylamide|||IMMA|||BML 190;2-[1-(4-氯苯甲酰基)-5-甲氧基-2-甲基-1H-吲哚-3-基]
产品简介:bml-190 (indomethacin morpholinylamide) is a specific cb2 receptor inverse agonist (ki: 435 nm), with 50-fold selectivity over cb1 receptor...产品型号:T6417 原产地:中国大陆价格: ¥0.0
产品名称: GLS1 Inhibitor-3;化合物 GLS1 Inhibitor-3GLS1 Inhibitor-3
产品简介:gls1 inhibitor-3 (compound c147) is a potent inhibitor of gls1 (ic50: 27.98 nm) and exhibits anti-proliferative effects...产品型号:T64211 原产地:中国大陆价格: ¥0.0
产品名称: Keap1-Nrf2-IN-1 TFA;化合物 Keap1-Nrf2-IN-1 TFAKeap1-Nrf2-IN-1 TFA
产品简介:keap1-nrf2-in-1 tfa (compound35) is a keap1-nrf2 protein-protein interaction inhibitor (ic50: 43 nm) that activates nrf2-regulated cytoprotective responses. kea..产品型号:T64218 原产地:中国大陆价格: ¥0.0
产品名称: JAK2 JH2 binder-1;化合物 JAK2 JH2 binder-1JAK2 JH2 binder-1
产品简介:jak2 jh2 binder-1 is a potent and selective jak2 jh2 binder (ki: 37.1 nm). jak2 jh2 binder-1 has the potential to be used in the study of various myeloprolifera..产品型号:T64227 原产地:中国大陆价格: ¥0.0
产品名称: ALDH1A1-IN-3;化合物 ALDH1A1-IN-3ALDH1A1-IN-3
产品简介:aldh1a1-in-3 is a good and selective inhibitor of aldehyde dehydrogenase 1a1 (aldh1a1) (ic50: μm).aldh1a1-in-3 is effective in improving glucose consumption in ..产品型号:T64228 原产地:中国大陆价格: ¥0.0