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产品名称: Sigma-1 receptor antagonist 4;化合物 Sigma-1 receptor antagonist 4Sigma-1 receptor antagonist 4
产品简介:sigma-1 receptor antagonist 4 (compound 32) is a potent σ1r antagonist that significantly enhances morphine´s analgesic effects and reverses morphine-indu..产品型号:T74813 原产地:中国大陆价格: ¥0.0
产品名称: PKM2/PDK1-IN-1;化合物 PKM2/PDK1-IN-1PKM2/PDK1-IN-1
产品简介:pkm2/pdk1-in-1, a shikonin thioether derivative, serves as a dual inhibitor for pkm2/pdk1. this compound effectively inhibits the proliferation and induces apop..产品型号:T74814 原产地:中国大陆价格: ¥0.0
产品名称: Complement C1s-IN-1;化合物 Complement C1s-IN-1Complement C1s-IN-1
产品简介:complement c1s-in-1 is a potent and selective c1s inhibitor that is orally active and capable of crossing the blood-brain barrier, demonstrating an ic50 value o..产品型号:T74816 原产地:中国大陆价格: ¥0.0
产品名称: IL-1β-IN-1;化合物 IL-1β-IN-1IL-1β-IN-1
产品简介:il-1β-in-1, a cannabidiol derivative, acts as a potent inhibitor of il-1β, exhibiting significant anti-inflammatory and pain relief properties [1]...产品型号:T74819 原产地:中国大陆价格: ¥0.0
产品名称: S1R agonist 1;化合物 S1R agonist 1S1R agonist 1
产品简介:compound 6b, also known as s1r agonist 1, is a selective agonist for s1r with dissociation constants (ki) of 0.93 nm for s1r and 72 nm for s2r. this compound de..产品型号:T74822 原产地:中国大陆价格: ¥0.0
产品名称: TGR5 agonist 1;化合物 TGR5 agonist 1TGR5 agonist 1
产品简介:compound 18 (tgr5 agonist 1) is a potent agonist of tgr5, exhibiting an ec50 value of 0.31 ?m [1]...产品型号:T74824 原产地:中国大陆价格: ¥0.0
产品名称: AcrB-IN-1;化合物 AcrB-IN-1AcrB-IN-1
产品简介:acrb-in-1 (compound h6) is a highly effective inhibitor of acrb, utilized for the reversal of bacterial multidrug resistance [1]...产品型号:T74826 原产地:中国大陆价格: ¥0.0
产品名称: PDK-IN-1;化合物 PDK-IN-1PDK-IN-1
产品简介:pdk-in-1 (compound 7o), a pyruvate dehydrogenase kinase (pdk) inhibitor, exhibits ic50 values of 0.03 and 0.1 μm against pdk1 and hsp90, respectively. this comp..产品型号:T74830 原产地:中国大陆价格: ¥0.0
产品名称: MTHFD2-IN-1;化合物 MTHFD2-IN-1MTHFD2-IN-1
产品简介:mthfd2-in-1 (compound 12) is a potent inhibitor of methylenetetrahydrofolate dehydrogenase (mthfd2) [1]...产品型号:T74834 原产地:中国大陆价格: ¥0.0
产品名称: ITK degrader 1;化合物 ITK degrader 1ITK degrader 1
产品简介:itk degrader 1, a highly selective interleukin-2-inducible t-cell kinase (itk; dc50=3.6 nm in vivo in mice) degrader, induces rapid and prolonged degradation of..产品型号:T74843 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC pan-IAP degrader-1;化合物 PROTAC pan-IAP degrader-1PROTAC pan-IAP degrader-1
产品简介:protac pan-iap degrader-1 (compound 9) is a pan- iap degrader protac . protac pan-iap degrader-1 degrades xiap , ciap1 and ciap2 with dc 50 s of 0.7, 2.4, and 6..产品型号:T74847 原产地:中国大陆价格: ¥0.0
产品名称: GluN2B-NMDAR antagonist-1;化合物 GluN2B-NMDAR antagonist-1GluN2B-NMDAR antagonist-1
产品简介:glun2b-nmdar antagonist-1, an orally active compound, functions as a glun2b-nmdar antagonist with neuroprotective properties. it is applicable in the research o..产品型号:T74854 原产地:中国大陆价格: ¥0.0
产品名称: LSD1-IN-25;化合物 LSD1-IN-25LSD1-IN-25
产品简介:lsd1-in-25 (compound 9j) is a potent, selective, and orally active inhibitor of lsd1, exhibiting an ic50 of 46 nm (ki = 30.3 nm) and capable of inducing apoptos..产品型号:T74855 原产地:中国大陆价格: ¥0.0
产品名称: LSD1-IN-26;化合物 LSD1-IN-26LSD1-IN-26
产品简介:lsd1-in-26 (compound 12u), a potent lsd1 inhibitor, exhibits an ic50 of 25.3 nm. it also demonstrates inhibition of mao-a (ic50 = 1234.57 nm) and mao-b (ic50 = ..产品型号:T74858 原产地:中国大陆价格: ¥0.0
产品名称: SLC7A11-IN-1;化合物 SLC7A11-IN-1SLC7A11-IN-1
产品简介:slc7a11-in-1 is a potent inhibitor of the solute carrier family 7 member 11 (slc7a11, xct), exhibiting antiproliferative, anti-tumor activities, and the ability..产品型号:T74859 原产地:中国大陆价格: ¥0.0
产品名称: 1,5-Dihexadecyl N-(3-carboxy-1-oxopropyl)-L-glutamate;化合物 1,5-Dihexadecyl N-(3-carboxy-1-oxopropyl)-
产品简介:1,5-dihexadecyl n-(3-carboxy-1-oxopropyl)-l-glutamate, a lipid, plays a crucial role in the synthesis of phospholipid vesicles and enhances the encapsulation ef..产品型号:T74875 原产地:中国大陆价格: ¥0.0
产品名称: Enzyme-IN-1;化合物 Enzyme-IN-1Enzyme-IN-1
产品简介:enzyme-in-1 (compound 1), a peptide-based inhibitor of n-terminal nucleophile (ntn) hydrolases, specifically targets and inhibits the chymotrypsin-like activity..产品型号:T74878 原产地:中国大陆价格: ¥0.0
产品名称: RNA splicing modulator 1;化合物 RNA splicing modulator 1RNA splicing modulator 1
产品简介:rna splicing modulator 1 (compound 233) is a modulator of rna splicing, exhibiting an ac50 value of less than 100 nm [1]...产品型号:T74884 原产地:中国大陆价格: ¥0.0
产品名称: MART-1 (26-35) (human);化合物MART-1 (26-35) humanMART-1 (26-35) human;MART-1 (26-35) human
产品简介:mart-1 (26-35) (human) (mart-1 (26-35) human) is a peptide fragment of mart-1 protein...产品型号:T7489 原产地:中国大陆价格: ¥0.0
产品名称: SIRT1/2/3-IN-1;化合物 SIRT1/2/3-IN-1SIRT1/2/3-IN-1
产品简介:sirt1/2/3-in-1 (compound 10) is a potent, selective, and cell-permeable inhibitor targeting sirt1, sirt2, and sirt3, demonstrating inhibitory concentrations (ic..产品型号:T74894 原产地:中国大陆价格: ¥0.0