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产品名称: Rotigaptide TFA(355151-12-1 free base)Rotigaptide TFA
产品简介:rotigaptide tfa is a novel and specific modulator of cx43 and is a potent aap. rotigaptide prevents the uncoupling of cx43-mediated gap junction communication a..产品型号:T16790L 原产地:中国大陆价格: ¥0.0
产品名称: Vatalanib free base
产品简介:vatalanib is a vegfr2/kdr inhibitor (ic50: 37 nm)...产品型号:T17219 原产地:中国大陆价格: ¥0.0
产品名称: WR-99210WR99210 hydrochloride(47326-86-3 free base);6,6-Dimethyl-1-[3-(2,4,5-trichlorophenoxy)propox
产品简介:wr-99210 is a potent inhibitor of plasmodium falciparum dihydrofolate reductase (pfdhfr), which is a major malarial drug target. it has subnanomolar potency for..产品型号:T17257L 原产地:中国大陆价格: ¥0.0
产品名称: SHU 9119 acetateSHU 9119 acetate (168482-23-3 free base)
产品简介:shu 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hmc3r, hmc4r) receptors and a partial hmc5r agonist. the ic50 values of human mc3r, m..产品型号:T16879L 原产地:中国大陆价格: ¥0.0
产品名称: CL2A-SN-38 DCA 1279680-68-0(free base)
产品简介:cl2a-sn-38 is a drug-linker conjugate composed of a potent a dna topoisomerase i inhibitor sn-38 and a linker cl2a to make antibody drug conjugate (adc).. cl2a-..产品型号:T17731L 原产地:中国大陆价格: ¥0.0
产品名称: Setmelanotide Acetate(920014-72-8 free base)BIM-22493 Acetate;RM-493 Acetate;IRC-022493 Acetate
产品简介:setmelanotide acetate is a selective agonist of melanocortin 4 receptor (mc4r)(human and rat mc4r with ec50s of 0.27 nm and 0.28 nm, respectively)...产品型号:T12882L 原产地:中国大陆价格: ¥0.0
产品名称: Shepherdin 79-87 acetateShepherdin 79-87 acetate (861224-28-4 free base)
产品简介:shepherdin 79-87 acetate is a peptidomimetic antagonist of the complex between hsp90 and survivin, another key regulator of tumor cell viability...产品型号:T12896L 原产地:中国大陆价格: ¥0.0
产品名称: Tat-NR2B9c acetateNA-1 acetate;Tat-NR2B9c acetate (500992-11-0 Free base)
产品简介:tat-nr2b9c acetate is a postsynaptic density-95 (psd-95) inhibitor, with ec50 values of 6.7 nm and 670 nm for psd-95d2 (psd-95 pdz domain 2) and psd-95d1, respe..产品型号:T13112L1 原产地:中国大陆价格: ¥0.0
产品名称: SN50 acetate (213546-53-3 free base)
产品简介:sn50 acetate is a cell permeable inhibitor of nf-κb translocation...产品型号:T12942L 原产地:中国大陆价格: ¥0.0
产品名称: TRPV4 agonist-1 free baseOUN67600
产品简介:trpv4 agonist-1 free base is an agonist of transient receptor potential vanilloid 4 (trpv4;ec50 of 60 nm, in the htrpv4 ca2+ assay)...产品型号:T13214L 原产地:中国大陆价格: ¥0.0
产品名称: WAY-213613 hydrochlorideWAY-213613 hydrochloride (868359-05-1 free base)
产品简介:way-213613 hydrochloride is a selective nonsubstrate reuptake glt-1/eaat2 inhibitor (ic50: 85 nm, eaat2). way-213613 hydrochloride displays 59- and 44-fold sele..产品型号:T13330 原产地:中国大陆价格: ¥0.0
产品名称: AZ7550 hydrochlorideAZ7550 hydrochloride (1421373-99-0 free base)
产品简介:az7550 hydrochloride, an active metabolite of azd9291, inhibits the activity of igf1r (ic50: 1.6 μm)...产品型号:T13564L 原产地:中国大陆价格: ¥0.0
产品名称: Motixafortide TFA(664334-36-5,Free)TF 14016 TFA;BKT140 TFA;T140 TFA;BL-8040 TFA
产品简介:motixafortide is an antagonist of cxcr4 with ic50 of ~1 nm. it induces the apoptosis of aml blasts by down-regulating erk, bcl-2, mcl-1 and cyclin-d1 via altere..产品型号:T14665L 原产地:中国大陆价格: ¥0.0
产品名称: Evatanepag2-[3-[N-(4-叔丁基苄基)-N-(吡啶-3-基磺酰基)氨基甲基]苯氧基]乙酸;CP-533536 free acid
产品简介:evatanepag is an ep2 receptor selective prostaglandin e2 (pge2) agonist that induces local bone formation with ec50 of 0.3 nm.cp-533536 demonstrated the ability..产品型号:T15259 原产地:中国大陆价格: ¥0.0
产品名称: AZD5582 acetate (1258392-53-8 free base)
产品简介:azd5582 acetate is an inhibitor of iaps, which binds to the bir3 domains ciap1, ciap2, and xiap with ic50s of 15, 21, and 15 nm, respectively. azd5582 induces a..产品型号:T14378L 原产地:中国大陆价格: ¥0.0
产品名称: Colistin sulfate (1066-17-7 free base)Colistin sulfate;Polymixin E Sulfate;Polymyxin E Sulfate;硫酸粘杆菌
产品简介:colistin is a cyclic polypeptide antibiotic from bacillus colistinus, composed of polymyxins e1 and e2...产品型号:T1245 原产地:中国大陆价格: ¥0.0
产品名称: PMX 205 acetate(514814-49-4 free base)
产品简介:pmx 205 acetate is an antagonist of complement c5a receptor (c5ar; cd88)...产品型号:T12506L1 原产地:中国大陆价格: ¥0.0
产品名称: CEP-28122 mesylate salt (1022958-60-6 free base)CEP-28122 mesylate salt
产品简介:cep-28122 mesylate salt is a highly selective orally active alk inhibitor (ic50: 1.9 nm in an enzyme-based trf assay)...产品型号:T10759 原产地:中国大陆价格: ¥0.0
产品名称: Ciraparantag acetateCiraparantag acetate(1438492-26-2 Free base)
产品简介:ciraparantag acetate, an anticoagulant reversal agent, is a small molecule specifically designed to bind noncovalently by charge-charge interaction to unfractio..产品型号:T10820L1 原产地:中国大陆价格: ¥0.0
产品名称: G3-C12 acetate(848301-94-0 free base)
产品简介:g3-c12 acetate shows anticancer activity.?is a galectin-3 binding peptide, with kd of 88 nm...产品型号:T11346L 原产地:中国大陆价格: ¥0.0