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产品名称: HIF-2α-IN-9;化合物 HIF-2α-IN-9HIF-2α-IN-9
产品简介:hif-2α-in-9 (compound 35r) serves as an hif-2α inhibitor, effectively suppressing vegf-a with an ic50 of 305 nm, and modulating growth-promoting genes within tu..产品型号:T78937 原产地:中国大陆价格: ¥0.0
产品名称: Tazarotenic acid;化合物AGN-190299AGN-190299;6-[2-(3,4-二氢-4,4-二甲基-2H-1-苯并噻喃-6-基)乙炔基]-3-吡啶甲酸|||AGN-190299
产品简介:tazarotenic acid (agn-190299) is a retinoid prodrug which is converted to its active form..产品型号:T7894 原产地:中国大陆价格: ¥0.0
产品名称: VDR agonist 2;化合物 VDR agonist 2VDR agonist 2
产品简介:vdr agonist 2 (compound 16i), a vitamin d receptor (vdr) agonist, effectively inhibits tgf-β1-induced hepatic stellate cell (hsc) activation, demonstrating nota..产品型号:T78944 原产地:中国大陆价格: ¥0.0
产品名称: MAT2A-IN-10;化合物 MAT2A-IN-10MAT2A-IN-10
产品简介:mat2a-in-10 (compound 28), an orally active inhibitor of mat2a, exhibits an ic50 of 26 nm and is utilized in cancer research [1]...产品型号:T78946 原产地:中国大陆价格: ¥0.0
产品名称: Analgesic agent-2;化合物 Analgesic agent-2Analgesic agent-2
产品简介:analgesic agent-2, a selective orally active inhibitor of the nav1.8 channel, demonstrates an ic50 of 50.18 nm in hek293 cells that stably express the human nav..产品型号:T78955 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD3/BRD4-L degrader-2;化合物 PROTAC BRD3/BRD4-L degrader-2PROTAC BRD3/BRD4-L degrader-2
产品简介:protac brd3/brd4-l degrader-2, a protac molecule, selectively degrades cellular brd3 and brd4-l with k i values of 16.91 and 2.8 nm, respectively, and exhibits ..产品型号:T78956 原产地:中国大陆价格: ¥0.0
产品名称: FABP4-IN-2;化合物 FABP4-IN-2FABP4-IN-2
产品简介:fabp4-in-2 (compd 10g), a selective and orally active fabp4 inhibitor, exhibits k i values of 0.51 μm for fabp4 and 33.01 μm for fabp3, demonstrating its specif..产品型号:T78960 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2-IN-38;化合物 SARS-CoV-2-IN-38SARS-CoV-2-IN-38
产品简介:sars-cov-2-in-38, also known as compound 24, is an inhibitor of sars-cov-2 that demonstrates favorable oral bioavailability in mice, with an absorption fraction..产品型号:T78961 原产地:中国大陆价格: ¥0.0
产品名称: Nrf2-IN-3;化合物 Nrf2-IN-3Nrf2-IN-3
产品简介:nrf2-in-3 (compound r16), a nrf2 inhibitor, binds to keap1 mutants (g333c mkeap1) thereby restoring the impaired keap1/nrf2 interactions. this restoration sensi..产品型号:T78841 原产地:中国大陆价格: ¥0.0
产品名称: MET/PDGFRA-IN-2;化合物 MET/PDGFRA-IN-2MET/PDGFRA-IN-2
产品简介:met/pdgfra-in-2 (compound 8h) serves as an inhibitor of met and pdgfra proteins, promoting apoptosis in cells and impeding the proliferation of met-positive cel..产品型号:T78844 原产地:中国大陆价格: ¥0.0
产品名称: FGFR1/VEGFR2-IN-1;化合物 FGFR1/VEGFR2-IN-1FGFR1/VEGFR2-IN-1
产品简介:fgfr1/vegfr2-in-1 (compound 2b) is an inhibitor of both fgfr1 and vegfr2, applicable in cancer research [1]...产品型号:T78845 原产地:中国大陆价格: ¥0.0
产品名称: EGFR/BRAFV600E-IN-2;化合物 EGFR/BRAFV600E-IN-2EGFR/BRAFV600E-IN-2
产品简介:e07 aptamer, targeting the human epidermal growth factor receptor (hegfr), competes with epidermal growth factor (egf) for binding to a unique epitope on egfr. ..产品型号:T78849 原产地:中国大陆价格: ¥0.0
产品名称: TWIK-1/TREK-1-IN-2;化合物 TWIK-1/TREK-1-IN-2TWIK-1/TREK-1-IN-2
产品简介:twik-1/trek-1-in-2 (compound 2g) serves as an inhibitor of both twik-1 and trek-1, targeting the trek-1 homodimer and twik-1/trek-1 heterodimer with ic50 values..产品型号:T78869 原产地:中国大陆价格: ¥0.0
产品名称: STAT3 degrader-2;化合物 STAT3 degrader-2STAT3 degrader-2
产品简介:stat3 degrader-2 is a protac-based compound that effectively reduces the total stat3 protein levels, and is utilized in the research of cancer and various disea..产品型号:T78983 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2-IN-54;化合物 SARS-CoV-2-IN-54SARS-CoV-2-IN-54
产品简介:sars-cov-2-in-54 (compound 2), a sars-cov-2 inhibitor, exhibits antiviral activity by impeding the virus in vero e6 cells with an inhibitory concentration (ic50..产品型号:T79328 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2-IN-56;化合物 SARS-CoV-2-IN-56SARS-CoV-2-IN-56
产品简介:sars-cov-2-in-56 (compound 63) is a sars-cov-2 inhibitor with antiviral activity, demonstrating inhibition of the virus in vero e6 cells with an ic50 of 0.7 μm ..产品型号:T79329 原产地:中国大陆价格: ¥0.0
产品名称: MAT2A-IN-11;化合物 MAT2A-IN-11MAT2A-IN-11
产品简介:mat2a allosteric inhibitor 1, also known as compound 5, is a selective inhibitor of methionine adenosyltransferase (mat) demonstrating potent activity with an i..产品型号:T79349 原产地:中国大陆价格: ¥0.0
产品名称: 2-Aminothiazol-4-acetic acid;2-氨基-4-噻唑乙酸2-Aminothiazol-4-acetic acid
产品简介:2-aminothiazol-4-acetic acid acts by inhibiting the activity of certain enzymes and proteins related to inflammation, tumor growth and oxidative stress, and has..产品型号:T7935 原产地:中国大陆价格: ¥0.0
产品名称: MAT2A-IN-12;化合物 MAT2A-IN-12MAT2A-IN-12
产品简介:mat2a allosteric inhibitor 2 is a potent, selective inhibitor exhibiting an ic50 of 5 nm and demonstrates nanomolar efficacy (ic50 = 5 μm) in proliferation assa..产品型号:T79350 原产地:中国大陆价格: ¥0.0
产品名称: RIPK2/3-IN-1;化合物 RIPK2/3-IN-1RIPK2/3-IN-1
产品简介:ripk2/3-in-1 is a potent inhibitor of both ripk2 and ripk3 kinases, exhibiting ic50 values of 3 nm for ripk2 and 117 nm for ripk3. additionally, in a 14-trilan-..产品型号:T79352 原产地:中国大陆价格: ¥0.0