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产品名称: ET receptor antagonist 2;化合物 ET receptor antagonist 2ET receptor antagonist 2
产品简介:et receptor antagonist 2 (compound 16j) is an orally active et receptor antagonist with an ic50 of 0.22 nm, suitable for pulmonary arterial hypertension (pah) r..产品型号:T79574 原产地:中国大陆价格: ¥0.0
产品名称: CB2 PET Radioligand 1;化合物 CB2 PET Radioligand 1CB2 PET Radioligand 1
产品简介:cb2 pet radioligand 1 (compound [18f]9) is a positron emission tomography (pet) radioligand with high affinity for the human cannabinoid receptor 2 (hcb2, ki=7...产品型号:T79577 原产地:中国大陆价格: ¥0.0
产品名称: ddUTP;化合物 ddUTP2′,3′-Dideoxyuridine-5′-triphosphate;2′,3′-Dideoxyuridine-5′-triphosphate
产品简介:ddutp (2′,3′-dideoxyuridine-5′-triphosphate) serves as a selective inhibitor of hiv and amv reverse transcriptases with ki values of 0.05 ?m for hiv and 1 ?m fo..产品型号:T79579 原产地:中国大陆价格: ¥0.0
产品名称: JAK2-IN-9;化合物 JAK2-IN-9JAK2-IN-9
产品简介:compound a8, known as jak2-in-9, is a selective jak2 inhibitor with an ic50 of 5 nm. it effectively inhibits the phosphorylation of jak2, stat3, and stat5, poss..产品型号:T79581 原产地:中国大陆价格: ¥0.0
产品名称: Benzopinacole;1,1,2,2-四苯基-1,2-乙二醇Benzopinacole
产品简介:benzopinacole is an anti-amoeba drug that can be used as an intermediate to synthesize a variety of compounds...产品型号:T7936 原产地:中国大陆价格: ¥0.0
产品名称: COX-2/15-LOX-IN-2;化合物 COX-2/15-LOX-IN-2COX-2/15-LOX-IN-2
产品简介:cox-2/15-lox-in-2 is a potent inhibitor of both cox-2 and 15-lox, demonstrating ic50 values of 0.065 μm for cox-2 and 1.86 μm for 15-lox. additionally, it exhib..产品型号:T79360 原产地:中国大陆价格: ¥0.0
产品名称: COX-2/15-LOX-IN-3;化合物 COX-2/15-LOX-IN-3COX-2/15-LOX-IN-3
产品简介:cox-2/15-lox-in-3 (compound 5k) serves as a dual inhibitor for cox-2 and 15-lox, demonstrating inhibitory concentrations (ic50) of 0.075 μm and 1.97 μm, respect..产品型号:T79361 原产地:中国大陆价格: ¥0.0
产品名称: COX-2/15-LOX-IN-4;化合物 COX-2/15-LOX-IN-4COX-2/15-LOX-IN-4
产品简介:cox-2/15-lox-in-4 (compound 5i) is a dual inhibitor with ic50 values of 0.075 μm for cox-2 and 1.97 μm for 15-lox. it inhibits lps-induced production of pro-inf..产品型号:T79362 原产地:中国大陆价格: ¥0.0
产品名称: TIM-3-IN-2;TIM-3 抑制剂2TIM-3-IN-2
产品简介:tim-3-in-2 is a tim3 inhibitor that inhibits the binding of tim-3 to ptdser, ceacam1, and gal-9 and inhibits the action of tim-3.tim-3-in-2 is able to reverse t..产品型号:T79365 原产地:中国大陆价格: ¥0.0
产品名称: SP-2-225;化合物 SP-2-225SP-2-225
产品简介:sp-2-225, a selective inhibitor of hdac6, augments the production of cancer-associated antigens and enhances macrophage antigen cross-presentation to t cells, d..产品型号:T79366 原产地:中国大陆价格: ¥0.0
产品名称: A3AR agonist 2;化合物 A3AR agonist 2A3AR agonist 2
产品简介:compound 19, a selective a3 adenosine receptor (a3ar) agonist (k i : 22.1 nm), effectively stimulates β-arrestin2 recruitment with an ec 50 value of 4.36 nm. th..产品型号:T79373 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2 3CLpro-IN-19;化合物 SARS-CoV-2 3CLpro-IN-19SARS-CoV-2 3CLpro-IN-19
产品简介:sars-cov-2 3clpro-in-19 (compound c5a), a non-covalent, non-peptide inhibitor of the sars-cov-2 3clpro enzyme, exhibits potent in vitro activity with an ic50 of..产品型号:T79376 原产地:中国大陆价格: ¥0.0
产品名称: Galectin-3/galectin-8-IN-2;化合物 Galectin-3/galectin-8-IN-2Galectin-3/galectin-8-IN-2
产品简介:galectin-3/galectin-8-in-2 (compound 57) is a dual inhibitor targeting the c-terminal domains of galectin-3 and galectin-8, exhibiting dissociation constants (k..产品型号:T79381 原产地:中国大陆价格: ¥0.0
产品名称: LTB4-IN-2;化合物 LTB4-IN-2LTB4-IN-2
产品简介:ltb4-in-2 (compound 6x) is a selective inhibitor of leukotriene b4 (ltb4), acting by specifically targeting the 5-lipoxygenase-activating protein (flap) with an..产品型号:T79389 原产地:中国大陆价格: ¥0.0
产品名称: Fingolimod;芬戈莫德FTY-720A|||FTY-720;2-氨基-2-[2-(4-辛基苯基)乙基]-1,3-丙二醇|||FTY-720A|||FTY-720|||芬戈莫德
产品简介:fingolimod (fty-720a) is an antagonist of sphingosine 1-phosphate (s1p) (ic50 of 0.033 nm in k562 and nk cells)...产品型号:T7939 原产地:中国大陆价格: ¥0.0
产品名称: ABCG2-IN-1;化合物 ABCG2-IN-1ABCG2-IN-1
产品简介:abcg2-in-1 (compound k2), an analog of ko143, constitutes an orally active inhibitor targeting abcg2 with an inhibitory concentration (ic50) of 0.13 μm. demonst..产品型号:T79513 原产地:中国大陆价格: ¥0.0
产品名称: ABCG2-IN-2;化合物 ABCG2-IN-2ABCG2-IN-2
产品简介:abcg2-in-2 is a potent inhibitor of abcg2, exhibiting favorable oral pharmacokinetic profiles in mice, and is applicable for investigating tumor multidrug resis..产品型号:T79514 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2 Mpro-IN-10;化合物 SARS-CoV-2 Mpro-IN-10SARS-CoV-2 Mpro-IN-10
产品简介:sars-cov-2 mpro-in-10 (27h) is a potent inhibitor of the mpro enzyme, exhibiting ic50 and ec50 values of 10.9 nm and 43.6 nm, respectively. it is utilized in re..产品型号:T79515 原产地:中国大陆价格: ¥0.0
产品名称: ROS inducer 2;化合物 ROS inducer 2ROS inducer 2
产品简介:compound i16 (ros inducer 2) is a potent inducer of reactive oxygen species (ros) with an effective concentration (ec 50) of 3.43 μg/ml demonstrated in vitro. i..产品型号:T79517 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2 nsp14-IN-4;化合物 SARS-CoV-2 nsp14-IN-4SARS-CoV-2 nsp14-IN-4
产品简介:sars-cov-2 nsp14-in-4 (compound 12q), a non-cytotoxic and cell-permeable inhibitor of sars-cov-2 nsp14 methyltransferase (ic50 = 19 nm), is employed in covid-19..产品型号:T79526 原产地:中国大陆价格: ¥0.0