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产品名称: Dorsomorphin dihydrochloride6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶;Dorsomorphin (Compound C) 2
产品简介:dorsomorphin is a potent, selective and atp-competitive ampk inhibitor (ki: 109 nm) and does not exhibit significant activity on structurally related kinases...产品型号:T6146 原产地:中国大陆价格: ¥0.0
产品名称: Ruxolitinib (S enantiomer)S-Ruxolitinib;INCB018424;INCB18424;Ruxolitinib S enantiomer;环丙基[4-[3-(1H-咪
产品简介:ruxolitinib s enantiomer is the s-enantiomer of ruxolitinib. ruxolitinib is the first potent, selective jak1/2 inhibitor...产品型号:T6156 原产地:中国大陆价格: ¥0.0
产品名称: BI 25364-[[(7R)-8-环戊基-7-乙基-5,6,7,8-四氢-5-甲基-6-氧代-2-喋啶基]氨基]-3-甲氧基-N-(1-甲基-4-哌啶基)苯甲酰胺
产品简介:bi2536 is an effective plk1 inhibitor (ic50: 0.83 nm). it has 4- and 11-fold greater selectivity than plk2 and plk3...产品型号:T6173 原产地:中国大陆价格: ¥0.0
产品名称: Domatinostat4SC-202;4SC-202 (free base);4SC 202;4SC202
产品简介:4sc-202 is a selective class i hdac inhibitor with ic50 of 1.20 μm, 1.12 μm, and 0.57 μm for hdac1, hdac2, and hdac3, respectively. also displays inhibitory act..产品型号:T6362 原产地:中国大陆价格: ¥0.0
产品名称: 4μ8CIRE1 Inhibitor III
产品简介:4μ8c(ic50=76 nm) is an effective and specific ire1 rnase inhibitor...产品型号:T6363 原产地:中国大陆价格: ¥0.0
产品名称: A 922500(1R,2R)-2-[[4-[[(苯基氨基)羰基]氨基][1,1-联苯]-4-基]甲酰基]环戊烷羧酸;DGAT-1 Inhibitor 4a;A922500
产品简介:a922500 is an inhibitor for human and mouse dgat-1 with ic50 of 7 nm and 24 nm, respectively, good selectivity over related acyltransferases, herg, and a panel ..产品型号:T6365 原产地:中国大陆价格: ¥0.0
产品名称: A-9664922-[2-氟-4-[(2S)-2-吡咯烷基]苯基]-1H-苯并咪唑-7-甲酰胺;A966492;A 966492
产品简介:a-96649 is a new-type and effective inhibitor. the ki of a-966492 for parp1 and parp2 is 1 nm and 1.5 nm, respectively...产品型号:T6366 原产地:中国大陆价格: ¥0.0
产品名称: Iniparib3-硝基-4-碘苯甲酰胺;BSI-201;IND-71677;NSC-746045
产品简介:iniparib (bsi-201) , a parp1 inhibitor, exhibits potency in triple-negative breast y (tnbc)...产品型号:T6224 原产地:中国大陆价格: ¥0.0
产品名称: Fosbretabulin DisodiumCA 4DP;Combretastatin A4 disodium phosphate;CA 4P;Fosbretabulin (Combretastati
产品简介:fosbretabulin (combretastatin a4 phosphate (ca4p)) disodium, a water-soluble prodrug of combretastatin a4 (ca4), is a microtubule-targeting agent that binds β-t..产品型号:T6272 原产地:中国大陆价格: ¥0.0
产品名称: Vadimezan伐地美生;ASA-404;NSC 640488;5,6-Dimethylxanthenone-4-acetic Acid;DMXAA
产品简介:vadimezan is a fused tricyclic analogue of flavone acetic acid with potential antineoplastic activity. vadimezan induces the cytokines tumor necrosis alpha (tnf..产品型号:T6273 原产地:中国大陆价格: ¥0.0
产品名称: ON-01910N-[2-甲氧基-5-[[[2-(2,4,6-三甲氧基苯基)乙烯基]磺酰]甲基]苯基]甘氨酸钠盐
产品简介:on-01910 is a non-atp-competitive plk1 inhibitor(ic50 of 9 nm, in a cell-free assay). it shows 30-fold greater selectivity against plk2 and no activity to plk3...产品型号:T6070 原产地:中国大陆价格: ¥0.0
产品名称: PCI-34051N-羟基-1-(4-甲氧基苄基)-1H-吲哚-6-甲酰胺;PCI 34051;PCI34051
产品简介:pci-34051 is an effective and selective hdac8 inhibitor (ic50: 10 nm)...产品型号:T6325 原产地:中国大陆价格: ¥0.0
产品名称: Ethyl 2-amino-4-methyl-5-[(3-nitrophenyl)carbamoyl]thiophene-3-carboxylateHistone Methyltransferase,
产品简介:ethyl 2-amino-4-methyl-5-[(3-nitrophenyl)carbamoyl]thiophene-3-carboxylate is a selective inhibitor of histone methyltransferase setd7 (ic50 = 4.59 μm) with ant..产品型号:T60002 原产地:中国大陆价格: ¥0.0
产品名称: Methyl arachidateLTA4H,natural,Methyl arachidate,Aminopeptidase,inhibit,Inhibitor,compound,Methyl ei
产品简介:methyl icosanoate is an esterified form of arachidic acid..产品型号:T7958 原产地:中国大陆价格: ¥0.0
产品名称: tcY-NH2 TFA(327177-34-4 free base)tcY-NH-2 TFA(327177-34-4 free base),tcY NH2 TFA(327177 34 4 free b
产品简介:tcy-nh2 tfa is a selective par4 antagonist peptide. inhibits endostatin release and platelet aggregation induced by thrombin...产品型号:TP1925L 原产地:中国大陆价格: ¥0.0
产品名称: FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CARFMOCL1,2,3,4TETRAHYDRONORHARMAN3CAR,FMOC L 1,2,3,4 TETRAHYDR
产品简介:fmoc-l-1,2,3,4-tetrahydronorharman-3-car is a chemical compound...产品型号:T8673 原产地:中国大陆价格: ¥0.0
产品名称: d[Cha4]-AVP acetate(500170-27-4 free base)d[Cha4]AVP acetate(500170274 free base),d[Cha4] AVP acetat
产品简介:d[cha4]-avp acetate is a potent and selective human vasopressin v1b receptor agonist (ki values are 1.2, 151, 240 and 750 nm for v1b, v1a, oxytocin and v2 recep..产品型号:TP2082L 原产地:中国大陆价格: ¥0.0
产品名称: (E)-Flavokawain AFLAVOKAVAIN A(P);(E)-1-(2-羟基-4,6-二甲氧基苯基)-3-(4-甲氧基苯基)-2-丙烯-1-酮;卡瓦胡椒素A
产品简介:flavokavin a, a novel chalcone from kava extract, induces apoptosis in bladder cancer cells by involvement of bax protein-dependent and mitochondria-dependent a..产品型号:T5715 原产地:中国大陆价格: ¥0.0
产品名称: 4-Phenoxybenzylamine
产品简介:4-phenoxybenzylamine inhibits the function of the ns3 protein by stabilizing an inactive conformation with an ic50 of about 500 μm against hcv ns3/4a ...产品型号:T5938 原产地:中国大陆价格: ¥0.0
产品名称: KPT-65662-[[4-[[[4-(叔丁基)苯基]磺酰基]亚氨基]-1-氧代-1,4-二氢-2-萘基]硫基]乙酸
产品简介:kpt-6566 is a novel selective covalent pin1 inhibitor, kpt-6566 shows an ic50 of 640 nm and a ki of 625.2 nm for pin1 ppiase domain,and has anti-cancer activity..产品型号:T5994 原产地:中国大陆价格: ¥0.0