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产品名称: URAT1 inhibitor 4;化合物 URAT1 inhibitor 4URAT1 inhibitor 4
产品简介:urat1 inhibitor 4, derived from lesinurad, is a potent, orally active inhibitor of urat1 with an ic50 value of 7.56 μm, demonstrating greater in vivo urate-lowe..产品型号:T72632 原产地:中国大陆价格: ¥0.0
产品名称: β-catenin-IN-4;化合物 β-catenin-IN-4β-catenin-IN-4
产品简介:β-catenin-in-4 is a β-catenin inhibitor characterized by a k_i value of 0.64 μm. this compound effectively lowers the protein expression levels of cyclin d1 and..产品型号:T72829 原产地:中国大陆价格: ¥0.0
产品名称: SHP2/CDK4-IN-1;化合物 SHP2/CDK4-IN-1SHP2/CDK4-IN-1
产品简介:shp2/cdk4-in-1 (compound 10) is a dual inhibitor targeting shp2 and cdk4, exhibiting oral activity and high potency with ic50 values of 4.3 nm for shp2 and 18.2..产品型号:T72836 原产地:中国大陆价格: ¥0.0
产品名称: Tankyrase-IN-4;化合物 Tankyrase-IN-4Tankyrase-IN-4
产品简介:tankyrase-in-4 is a potent inhibitor of tankyrase 1 (tnks1), exhibiting an ic50 of 0.8 nm, and is utilized in cancer research...产品型号:T72847 原产地:中国大陆价格: ¥0.0
产品名称: BRD4 Inhibitor-26;化合物 BRD4 Inhibitor-26BRD4 Inhibitor-26
产品简介:brd4 inhibitor-26, a bromodomain protein 4 (brd4) inhibitor/nitric oxide-donator, exhibits inhibitory activity against brd4 (bd1) and brd4 (bd2) with ic50 value..产品型号:T72636 原产地:中国大陆价格: ¥0.0
产品名称: (3S,4S)-A2-32-01;化合物 (3S,4S)-A2-32-01(3S,4S)-A2-32-01
产品简介:(3s,4s)-a2-32-01, a less active (s,s)-enantiomer of a2-32-01. a2-32-01 is a potent caseinolytic protein proteases (clpp) inhibitor [1] ...产品型号:T72657 原产地:中国大陆价格: ¥0.0
产品名称: NMDAR/TRPM4-IN-2;化合物NMDAR/TRPM4-IN-2NMDAR/TRPM4-IN-2
产品简介:nmdar/trpm4-in-2 is a potent interfacial inhibitor of nmdar/trpm4 interaction.nmdar/trpm4-in-2 protects against mcao-induced brain damage and nmda-induced retin..产品型号:T72662 原产地:中国大陆价格: ¥0.0
产品名称: P-gp inhibitor 4;化合物 P-gp inhibitor 4P-gp inhibitor 4
产品简介:p-gp inhibitor 4 is a selective p-glycoprotein modulator with an ec 50 of 94 nm. p-gp inhibitor 4 increases drug transport across gastro-intestinal barrier and..产品型号:T72678 原产地:中国大陆价格: ¥0.0
产品名称: GLS1 Inhibitor-4;化合物 GLS1 Inhibitor-4GLS1 Inhibitor-4
产品简介:gls1 inhibitor-4 (compound 41e) is a powerful gls1 inhibitor, demonstrating an ic50 of 11.86 nm. it exhibits antiproliferative effects, substantial metabolic st..产品型号:T72679 原产地:中国大陆价格: ¥0.0
产品名称: RSV604;化合物RSV604(S)-1-(2-Fluorophenyl)-3-(2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)u
产品简介:rsv604 ((s)-1-(2-fluorophenyl)-3-(2-oxo-5-phenyl-2,3-dihydro-1h-benzo[e][1,4]diazepin-3-yl)urea) is an inhibitor of respiratory syncytial virus (rsv) that binds..产品型号:T7353 原产地:中国大陆价格: ¥0.0
产品名称: Ralfinamide(S)-2-[[4-[(2-氟苄基)氧基]苄基]氨基]丙酰胺(S)-2-[[4-[(2-氟苄基)氧基]苄基]氨基]丙酰胺|||Priralfinamide|||FCE-26742
产品简介:ralfinamide (priralfinamide) is an orally available na-channel blocker for the treatment of neuropathic pain and other pain conditions...产品型号:T7349 原产地:中国大陆价格: ¥0.0
产品名称: NP118809;化合物NP11880939-1B4;39-1B4|||1-【4-(二苯甲基)-1-哌嗪基】-3,3-二苯基-1-丙酮
产品简介:np118809 (39-1b4) is a potent n-type calcium channel blocker(ic50 : 0.11 μm)...产品型号:T7334 原产地:中国大陆价格: ¥0.0
产品名称: Nelotanserin;化合物NelotanserinAPD125;1-[3-(4-溴-1-甲基-1H-吡唑-5-基)-4-甲氧基苯基]-3-(2,4-二氟苯基)脲|||APD125
产品简介:nelotanserin (apd125) is a potent 5-ht2a inverse agonist(ic50 : 1.7 nm), a moderately potent 5-ht2c partial inverse agonist t(ic50 :79 nm )and a weak 5-ht2b inv..产品型号:T7350 原产地:中国大陆价格: ¥0.0
产品名称: Pridopidine;4-[3-(甲磺酰基)苯基]-1-丙基哌啶ACR16|||ASP2314|||FR310826;ACR16|||ASP2314|||FR310826|||4-[3-(甲磺酰基)
产品简介:pridopidine (fr310826), a dopamine (da) stabilizer, acts as a low affinity dopamine d2 receptor (d2r) antagonist, improves motor performance and shows neuroprot..产品型号:T7352 原产地:中国大陆价格: ¥0.0
产品名称: ICA-121431;化合物ICA-1214312,2-Diphenyl-N-[4-(thiazol-2-ylsulfamoyl;2,2-Diphenyl-N-[4-(thiazol-2-ylsulf
产品简介:ica-121431 (2,2-diphenyl-n-[4-(thiazol-2-ylsulfamoyl) is a nanomolar potent small molecule nav1.7 channel inhibitor with ic50 of 19 nm for rat nav1.7, with litt..产品型号:T7336 原产地:中国大陆价格: ¥0.0
产品名称: CK2-IN-4;CK2抑制剂4CK2-IN-4
产品简介:ck2-in-4 is a protein kinase (ck2) inhibitor with an ic50 value of 8.6 ?m. ck2-in-4 has potential anticancer ah and anti-inflammatory activity for the study of ..产品型号:T73375 原产地:中国大陆价格: ¥0.0
产品名称: CPT-Se4;化合物 CPT-Se4CPT-Se4
产品简介:cpt-se4, a seleno-derivative of camptothecin (cpt), exhibits enhanced efficacy in cancer cell eradication and tumor suppression. it reduces the gsh/gssg balance..产品型号:T73422 原产地:中国大陆价格: ¥0.0
产品名称: 7-Hydroxy-4H-chromen-4-one;7-羟基色原酮7-hydroxy-4-benzopyrone|||7-Hydroxy-4-chromone|||7-Hydroxychromone
产品简介:7-hydroxy-4h-chromen-4-one (7-hydroxy-4-benzopyrone) is a src kinase inhibitor (ic50 of <300 μm)...产品型号:T7345 原产地:中国大陆价格: ¥0.0
产品名称: iBRD4-BD1;化合物 iBRD4-BD1iBRD4-BD1
产品简介:ibrd4-bd1 is a selective inhibitor of the brd4 bromodomain, exhibiting inhibition activity with an ic50 value of 12 nm. it is utilized in the research of inflam..产品型号:T73296 原产地:中国大陆价格: ¥0.0
产品名称: Nucleozin化合物Nucleozin[4-(2-氯-4-硝基苯基)-1-哌嗪基](5-甲基-3-苯基-4-异噁唑基)-甲酮
产品简介:nucleozin targets influenza a nucleoprotein (np), a multifunctional, rna-binding protein necessary for virus replication...产品型号:T7330 原产地:中国大陆价格: ¥0.0