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产品名称: CYP51/PD-L1-IN-3;化合物 CYP51/PD-L1-IN-3CYP51/PD-L1-IN-3
产品简介:cyp51/pd-l1-in-3 (compound l21), a quinazoline with antifungal properties, serves as a dual inhibitor targeting cyp51 (ic50: 0.205 μm) and pd-l1 (ic50: 0.039 μm..产品型号:T79740 原产地:中国大陆价格: ¥0.0
产品名称: CARM1 degrader-1;化合物 CARM1 degrader-1CARM1 degrader-1
产品简介:protac carm1 degrader-1 (compound 3b) serves as a highly potent degrader (dc50=8.1 nm) of the co-activator associated arginine methyltransferase (carm1). this c..产品型号:T79741 原产地:中国大陆价格: ¥0.0
产品名称: CARM1 degrader-2;化合物 CARM1 degrader-2CARM1 degrader-2
产品简介:protac carm1 degrader-2 (compound 3e), with a dc50 value of 8.8 nm, is a vhl- and proteasome-dependent degrader of co-activator associated argininemethyltransfe..产品型号:T79742 原产地:中国大陆价格: ¥0.0
产品名称: Caspase-3 activator 1;化合物 Caspase-3 activator 1Caspase-3 activator 1
产品简介:caspase-3 activator 1 (compound 4b), a ru(iii) metal complex, effectively inhibits gastric tumor growth and metastasis by mediating caspase-3 cleavage. this cle..产品型号:T79743 原产地:中国大陆价格: ¥0.0
产品名称: IDH2R140Q-IN-2;IDH2R140Q 抑制剂1IDH2R140Q-IN-2
产品简介:idh2r140q-in-2 is an orally active and potent idh2r140q inhibitor with an ic50 of 29 nm.idh2r140q-in-2 possesses potential antitumour activity, reducing d2hg pr..产品型号:T79745 原产地:中国大陆价格: ¥0.0
产品名称: Rhodamine B;罗丹明BRhodamineu00A0B|||Tetraethylrhodamine|||Brilliant Pink B|||Basic Violet 1|||Rhodamin
产品简介:rhodamine b (brilliant pink b) is used as a tracer dye in water to determine the rate and direction of flow and transport...产品型号:T7975 原产地:中国大陆价格: ¥0.0
产品名称: FIKK9.1-IN-1;化合物 FIKK9.1-IN-1FIKK9.1-IN-1
产品简介:fikk9.1-in-1 (compound 1), an antimalarial agent (ic50: 2.68 μg/ml), serves as a fikk9.1 inhibitor by interacting with the atp-binding residues within fikk9.1, ..产品型号:T79690 原产地:中国大陆价格: ¥0.0
产品名称: Casein kinase 1δ-IN-10;化合物 Casein kinase 1δ-IN-10Casein kinase 1δ-IN-10
产品简介:casein kinase 1δ-in-10 is an inhibitor of casein kinase 1δ (ck1δ)...产品型号:T79697 原产地:中国大陆价格: ¥0.0
产品名称: 8-Amino-1-Naphthalenesulfonic Acid;周位酸8-Amino-1-Naphthalenesulfonic Acid
产品简介:8-amino-1-naphthalenesulfonic acid is a naphthalene derivative used as a fluorescent dye and as a reagent in organic synthesis. it is a highly fluorescent compo..产品型号:T7971 原产地:中国大陆价格: ¥0.0
产品名称: PI3Kα/HDAC6-IN-1;化合物 PI3Kα/HDAC6-IN-1PI3Kα/HDAC6-IN-1
产品简介:pi3kα/hdac6-in-1 (compound 21j) is a dual inhibitor of pi3kα and hdac6, exhibiting ic50 values of 2.9 nm and 26 nm, respectively. it effectively hinders akt(ser..产品型号:T79710 原产地:中国大陆价格: ¥0.0
产品名称: TPH1-IN-1;化合物 TPH1-IN-1TPH1-IN-1
产品简介:tph1-in-1 (compound 40) is a xanthine derivative that serves as an inhibitor of tryptophan hydroxylase tph1, with an ic50 of 110.1 nm. demonstrating robust in v..产品型号:T79712 原产地:中国大陆价格: ¥0.0
产品名称: JMJD3/HDAC-IN-1;化合物 JMJD3/HDAC-IN-1JMJD3/HDAC-IN-1
产品简介:compound a5b, also known as jmjd3/hdac-in-1, is a dual inhibitor that targets both jmjd3 (jumonji domain-containing protein demethylase 3) and hadc1 (histone de..产品型号:T79713 原产地:中国大陆价格: ¥0.0
产品名称: VHL-IN-1;化合物 VHL-IN-1VHL-IN-1
产品简介:vhl-in-1 (compound 30), a ubiquitin e3 ligase von hippel-lindau (vhl) inhibitor with a dissociation constant (kd) of 37 nm, potently stabilizes hif-1α and enhan..产品型号:T79720 原产地:中国大陆价格: ¥0.0
产品名称: DDR1/2 inhibitor-2;化合物 DDR1/2 inhibitor-2DDR1/2 inhibitor-2
产品简介:ddr1/2 inhibitor-2 (example 31) serves as an inhibitor of ddr1/ddr2, exhibiting ic50 values below 100 nm. it is applicable in cancer and fibrotic disease resear..产品型号:T79811 原产地:中国大陆价格: ¥0.0
产品名称: S1P1 agonist 6;化合物 S1P1 agonist 6S1P1 agonist 6
产品简介:compound i (s1p1 agonist 6) is an s1p1 agonist that mitigates autoimmune activity by inhibiting lymphocyte trafficking and has potential as an immunosuppressive..产品型号:T79816 原产地:中国大陆价格: ¥0.0
产品名称: S1P1 agonist 6 hemicalcium;化合物 S1P1 agonist 6 hemicalciumS1P1 agonist 6 hemicalcium
产品简介:compound i (s1p1 agonist 6 hemicalcium) is an s1p1 agonist that diminishes autoimmune activity by inhibiting lymphocyte trafficking, and serves as an immunosupp..产品型号:T79817 原产地:中国大陆价格: ¥0.0
产品名称: Sigma-1 receptor antagonist 5;化合物 Sigma-1 receptor antagonist 5Sigma-1 receptor antagonist 5
产品简介:sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptors ..产品型号:T78734 原产地:中国大陆价格: ¥0.0
产品名称: DGKα&ζ-IN-1;化合物 DGKα&ζ-IN-1DGKα&ζ-IN-1
产品简介:dgkα&ζ-in-1 (compound ii) is an inhibitor targeting dgk that potentiates t-cell function and exhibits a synergistic interaction with pd-1, offering therapeutic ..产品型号:T79824 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC MLKL Degrader-1;化合物 PROTAC MLKL Degrader-1PROTAC MLKL Degrader-1
产品简介:protac mlkl degrader-1 (compound 36) is a selective protac degrader targeting mlkl, achieving a degradation maximum (d max) over 90%. the compound encompasses m..产品型号:T79831 原产地:中国大陆价格: ¥0.0
产品名称: CRM1-IN-1;化合物 CRM1-IN-1CRM1-IN-1
产品简介:crm1-in-1 (compound kl1), a noncovalent inhibitor of crm1, promotes nuclear degradation of crm1 with an ic50 of 0.27 μm, inhibits crm1-mediated nuclear export, ..产品型号:T79654 原产地:中国大陆价格: ¥0.0