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产品名称: EtrasimodEtrasimod,APD-334,LPL Receptor,Inhibitor,inhibit,APD 334,Lysophospholipid Receptor
产品简介:etrasimod is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (s1p1) receptor (ic50: 1.88 nm in cho cells)...产品型号:TQ0227 原产地:中国大陆价格: ¥0.0
产品名称: MK-571 sodiumMRP4,Lysophospholipid Receptor,human mast cells,LAD2,MK 571 sodium,MRP1,Leukotriene Rec
产品简介:mk-571 is a selective, orally active antagonist of the cyslt1 receptor. mk571 is a multidrug resistance protein-2 (abcc2, mrp2) inhibitor used to demonstrate th..产品型号:T3148 原产地:中国大陆价格: ¥0.0
产品名称: Angiotensin I/II (1-5)Angiotensin I/II (15),inhibit,Angiotensin Receptor,Inhibitor,Angiotensin I/II
产品简介:angiotensin i/ii (1-5) is a peptide (asp-arg-val-tyr-ile) that contains the amino acids 1-5 and is converted from angiotensin i/ii...产品型号:TP1528 原产地:中国大陆价格: ¥0.0
产品名称: GW 405833GW405833,GW 405833,Cannabinoid Receptor,GW-405833,L768242,anti-inflammatory,Inhibitor,L 768
产品简介:gw 405833 is an agonist of cannabinoid-2 (cb(2)) receptor-selective..产品型号:T7705 原产地:中国大陆价格: ¥0.0
产品名称: GSK163090Dopamine Receptor,5-HT1A,GSK163090,Inhibitor,5-hydroxytryptamine Receptor,antidepressant,an
产品简介:gsk163090 is a specific and orally active 5-ht1a/b/d receptor antagonist (pkis: 9.4/8.5/9.7, and 6.3/6.7 for 5-ht1a/b/d, and dopamine d2/d3)...产品型号:TQ0311 原产地:中国大陆价格: ¥0.0
产品名称: GolvatinibE7050,Golvatinib,c-Met/HGFR,VEGFR,Inhibitor,Vascular endothelial growth factor receptor,E
产品简介:golvatinib is an orally bioavailable dual kinase inhibitor of c-met (hepatocyte growth factor receptor) and vegfr-2 (vascular endothelial growth factor receptor..产品型号:T6517 原产地:中国大陆价格: ¥0.0
产品名称: GSK5182inhibit,GSK-5182,GSK5182,Reactive Oxygen Species,GSK 5182,Estrogen Receptor/ERR,Inhibitor
产品简介:gsk5182 is a highly selective inverse estrogen-related receptor γ agonist (ic50 : 79 nm)..产品型号:T8370 原产地:中国大陆价格: ¥0.0
产品名称: Rotigotine-Rotigotine,dopamine,5-HT1A,Adrenergic Receptor,receptor,N0923,Serotonin Receptor,N 0923,5
产品简介:rotigotine is a non-ergot dopamine receptor agonist used in the therapy of parkinson disease and restless leg syndrome. administered as a once-daily transdermal..产品型号:T6647 原产地:中国大陆价格: ¥0.0
产品名称: SenktideSenktide,Inhibitor,inhibit,Tachykinin receptor,NK receptor,Neurokinin Receptor
产品简介:senktide is an agonist of tachykinin nk3 receptor...产品型号:T7633 原产地:中国大陆价格: ¥0.0
产品名称: FICZinhibit,Inhibitor,Aryl Hydrocarbon Receptor,AhR,FICZ
产品简介:ficz is a potent aryl agonist for the hydrocarbon receptor (ahr, kd: 70 pm)...产品型号:TQ0257 原产地:中国大陆价格: ¥0.0
产品名称: RevefenacinRevefenacin,TD4208,TD 4208,inhibit,Muscarinic acetylcholine receptor,Inhibitor,mAChR,GSK
产品简介:revefenacin is a machr antagonist has a high affinity on m3 receptor( ki : 0.18 nm),and potentially useful for the treatment of respiratory disease...产品型号:T7392 原产地:中国大陆价格: ¥0.0
产品名称: CB2 receptor agonist 2
产品简介:cb2 receptor agonist 2 is a potent and selective agonist for the cb2 (cannabinoid type 2) receptor, ki = 8.5 nm. cb2 receptor agonist 2 has high affinity and se..产品型号:T22009 原产地:中国大陆价格: ¥0.0
产品名称: N-Formyl-Met-Leu-PheTNF Receptor,TNFR,Inhibitor,NFormylMetLeuPhe,Tumor Necrosis Factor Receptor,inhi
产品简介:n-formyl-met-leu-phe (fmlf) is a synthetic peptide that acts as an agonist at formyl peptide receptors (fpr; ki = 0.8 pm)...产品型号:T7091 原产地:中国大陆价格: ¥0.0
产品名称: LY2828360Inhibitor,LY2828360,inhibit,LY-2828360,LY 2828360,Cannabinoid Receptor
产品简介:ly2828360 is a cannabinoid (cb) receptor 2 agonist (ki = 40.3 nm). it selectively activates cb2 over cb1 in a gtpγs binding assay (ec50s = 20.1 and >100,000 nm,..产品型号:T7316 原产地:中国大陆价格: ¥0.0
产品名称: VUF 101665-HT3A,VUF 10166,VUF10166,VUF-10166,neurotransmission,5-HT3AB,inhibit,5-HT3 receptor ligand
产品简介:vuf10166 is a novel, potent and competitive antagonist for 5-ht3a receptor with ki of 0.04 nm, its affinity at 5-ht3ab receptor is significantly lower...产品型号:T6728 原产地:中国大陆价格: ¥0.0
产品名称: Cyproheptadine hydrochlorideInhibitor,antihistamine,thromboprotective,Cyproheptadine,5-HT Receptor,5
产品简介:cyproheptadine hcl is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist...产品型号:T6814 原产地:中国大陆价格: ¥0.0
产品名称: NorepinephrineAutophagy,L-Noradrenaline,Beta Receptor,inhibit,Levarterenol,Norepinephrine,Inhibitor,
产品简介:norepinephrine can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. it can up-regulate the expression of vascula..产品型号:T7044 原产地:中国大陆价格: ¥0.0
产品名称: RN-1734RN1734,Inhibitor,RN-1734,Transient receptor potential channels,TRP Channel,inhibit,RN 1734
产品简介:rn-1734 is selective trpv4 channel antagonist(ic50 of 2.3 μm,5.9 μm,3.2 μm for htrpv4, mtrpv4 and rtrpv4,respectively)..产品型号:T7572 原产地:中国大陆价格: ¥0.0
产品名称: SSD114 hydrochlorideSSD114,Gamma-aminobutyric acid Receptor,Inhibitor,SSD 114,SSD-114,SSD114 hydroch
产品简介:ssd114 hydrochloride is a gabab receptor positive allosteric modulator...产品型号:T8664 原产地:中国大陆价格: ¥0.0
产品名称: Linoleoyl Ethanolamidefood,intake,Cannabinoid Receptor,feeding,Linoleic acid monoethanolamide,ananda
产品简介:linoleoyl ethanolamide is an endocannabinoid agent. it acts by binding to trpv1 increasing erk phosphorylation and ap-1 dependent transcription in cb-receptor i..产品型号:T8425 原产地:中国大陆价格: ¥0.0