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产品名称: S1P1 agonist 4;化合物 S1P1 agonist 4S1P1 agonist 4
产品简介:s1p1 agonist 4 exhibits enhanced potency with an ec 50 value of less than 0.05 mg/kg and a predicted human half-life (t1/2) of approximately 5 days, indicating ..产品型号:T61639 原产地:中国大陆价格: ¥0.0
产品名称: Ciproxifan;化合物CiproxifanFUB-359;FUB-359|||环丙基[4-[3-(1H-咪唑-4-基)丙氧基]苯基]甲酮马来酸盐
产品简介:ciproxifan (fub-359) is a highly effective and specific histamin h3-receptor antagonist (ic50: 9.2 nm)...产品型号:T6164 原产地:中国大陆价格: ¥0.0
产品名称: CXCR4 antagonist 9;化合物 CXCR4 antagonist 9CXCR4 antagonist 9
产品简介:cxcr4 antagonist 9 (compound 2) is a potent cxcr4 antagonist displaying an ic50 of 15 nm. it effectively inhibits the cytosolic calcium increase induced by cxcl..产品型号:T61650 原产地:中国大陆价格: ¥0.0
产品名称: O-GlcNAcase-IN-4;化合物 O-GlcNAcase-IN-4O-GlcNAcase-IN-4
产品简介:o-glcnacase-in-4 is an inhibitor of o-glcnacase. it holds potential for researching neurodegenerative diseases and disorders, including alzheimer´s diseas..产品型号:T61662 原产地:中国大陆价格: ¥0.0
产品名称: BChE-IN-4;化合物 BChE-IN-4BChE-IN-4
产品简介:bche-in-4 is a highly potent inhibitor of the enzyme butyrylcholinesterase, capable of crossing the blood-brain barrier. it effectively reduces learning and mem..产品型号:T61669 原产地:中国大陆价格: ¥0.0
产品名称: α-Synuclein inhibitor 4;化合物 α-Synuclein inhibitor 4α-Synuclein inhibitor 4
产品简介:α-synuclein inhibitor 4 (compound 3gh) is a highly effective and blood-brain barrier-permeable inhibitor of α-synuclein aggregation. it displays potent activity..产品型号:T61611 原产地:中国大陆价格: ¥0.0
产品名称: AChE/PDE4-IN-1;化合物 AChE/PDE4-IN-1AChE/PDE4-IN-1
产品简介:ache/pde4-in-1 (compound 12c) is a highly effective and specific dual inhibitor of pde4 and ache, with ic50 values of 0.28 μm and 1.88 μm for ache and pde4d, re..产品型号:T61620 原产地:中国大陆价格: ¥0.0
产品名称: ERK5-IN-4;化合物 ERK5-IN-4ERK5-IN-4
产品简介:erk5-in-4 (compound 34b) is a powerful and specific inhibitor of extracellular signal-related kinase 5 (erk5) activity. it effectively inhibits both the full-le..产品型号:T61628 原产地:中国大陆价格: ¥0.0
产品名称: hCAI/II-IN-4;化合物 hCAI/II-IN-4hCAI/II-IN-4
产品简介:hcai/ii-in-4 (compound 6d) is a powerful inhibitor of both hca i and hca ii enzymes, with ki values of 16.95 nm and 15.22 nm, respectively. it demonstrates inhi..产品型号:T61635 原产地:中国大陆价格: ¥0.0
产品名称: AR antagonist 4;化合物 AR antagonist 4AR antagonist 4
产品简介:ar antagonist 4 (compound 67-b) is an orally active androgen receptor (ar) antagonist that acts on wild-type ar (ic50: 246.6 nm)...产品型号:T62838 原产地:中国大陆价格: ¥0.0
产品名称: IRAK4-IN-13;化合物 IRAK4-IN-13IRAK4-IN-13
产品简介:irak4-in-13 (compound 21) is a selective and potent irak4 inhibitor (ic50: 0.6 nm). irak4-in-13 has a high metabolic clearance, with an intrinsic human liver mi..产品型号:T62850 原产地:中国大陆价格: ¥0.0
产品名称: FLT3/ITD-IN-4;化合物 FLT3/ITD-IN-4FLT3/ITD-IN-4
产品简介:flt3/itd-in-4 (compound 16) is a selective inhibitor of flt3 internal tandem repeat mutations (flt3-itd) (ic50: 2.3 nm). flt3/itd-in-4 can be used to study acut..产品型号:T62863 原产地:中国大陆价格: ¥0.0
产品名称: RdRP-IN-4;化合物 RdRP-IN-4RdRP-IN-4
产品简介:rdrp-in-4 (compound 11q) is an arylbenzohydrazide analogue, an orally active inhibitor of influenza a virus rna-dependent rna polymerase (rdrp) that directly bi..产品型号:T62812 原产地:中国大陆价格: ¥0.0
产品名称: FGFR4-IN-10;化合物 FGFR4-IN-10FGFR4-IN-10
产品简介:fgfr4-in-10 (compound 5a) is a selective and potent inhibitor of fgfr4 (ic50: 70.7 nm).fgfr4-in-10 does not inhibit other fgfr family members (i.e., fgfr1, fgfr..产品型号:T62682 原产地:中国大陆价格: ¥0.0
产品名称: Factor B-IN-4;化合物 Factor B-IN-4Factor B-IN-4
产品简介:factor b-in-4 is a potent inhibitor (ic50: 1 μm) of complement factor b. factor b-in-4 can be used to study inflammatory and immune-related diseases...产品型号:T62688 原产地:中国大陆价格: ¥0.0
产品名称: Antimicrobial agent-4;化合物 Antimicrobial agent-4Antimicrobial agent-4
产品简介:antimicrobial agent-4 (compound 6a) is a potent antimicrobial agent with high activity against microbial pathogens. -4 exhibits a high binding capacity of 10.0 ..产品型号:T62707 原产地:中国大陆价格: ¥0.0
产品名称: Rel-5-(4-Chloro-2-fluorophenyl)-2,3-dimethyl-7-[(2R,4S)-tetrahydro-2-(1-methyl-1H-pyrazol-4-yl)-2H-p
产品简介:rel-5-(4-chloro-2-fluorophenyl)-2,3-dimethyl-7-[(2r,4s)-tetrahydro-2-(1-methyl-1h-pyrazol-4-yl)-2h-pyran-4-yl]pyrido[3,4-b]pyrazine has an ec50 value of ≤ 0.05 ..产品型号:T62750L 原产地:中国大陆价格: ¥0.0
产品名称: Mu opioid receptor antagonist 4;化合物 Mu opioid receptor antagonist 4Mu opioid receptor antagonist 4
产品简介:mu opioid receptor antagonist 4 (compound 31) is a potent and selective mu opioid receptor (mor) antagonist that permeates the blood-brain barrier (ki: 0.38 nm,..产品型号:T62768 原产地:中国大陆价格: ¥0.0
产品名称: CDK4/6-IN-13;化合物 CDK4/6-IN-13CDK4/6-IN-13
产品简介:compounds 10b and 10c, functioning as cdk4/6 inhibitors, demonstrated low nanomolar activity, optimal antiproliferative effects, excellent metabolic properties,..产品型号:T62605 原产地:中国大陆价格: ¥0.0
产品名称: Microtubule inhibitor 4;化合物 Microtubule inhibitor 4Microtubule inhibitor 4
产品简介:microtubule inhibitor 4 (compound 2) is a potent inhibitor of microtubule and inhibits microtubule protein polymerization, ht-29 cells (ic50: 2.1 nm) exhibited ..产品型号:T62642 原产地:中国大陆价格: ¥0.0