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产品名称: PDE4B-IN-3;化合物 PDE4B-IN-3PDE4B-IN-3
产品简介:pde4b-in-3 is a potent inhibitor of pde4b (ic50: 0.94 μm) and exhibits anti-inflammatory effects...产品型号:T64005 原产地:中国大陆价格: ¥0.0
产品名称: BRD4-BD1/2-IN-2;化合物 BRD4-BD1/2-IN-2BRD4-BD1/2-IN-2
产品简介:brd4-bd1/2-in-2 is a potent inhibitor of brd4-bd2, capable of acting on both brd4 bd2 (ic50<0.5 nm) and brd4 bd1 (ic50<300 nm)...产品型号:T63707 原产地:中国大陆价格: ¥0.0
产品名称: GPX4-IN-3;化合物 GPX4-IN-3GPX4-IN-3
产品简介:gpx4-in-3 (26a) is a potent inhibitor of glutathione peroxidase 4 (gpx4), selectively inducing ferroptosis. it demonstrates a 71.7% inhibition rate of gpx4 at a..产品型号:T63729 原产地:中国大陆价格: ¥0.0
产品名称: FTO-IN-4;化合物 FTO-IN-4FTO-IN-4
产品简介:fto-in-4 is a potent and selective inhibitor of adiposity and obesity-associated protein (fto)...产品型号:T63740 原产地:中国大陆价格: ¥0.0
产品名称: Autophagy inducer 4;化合物 Autophagy inducer 4Autophagy inducer 4
产品简介:autophagy inducer 4 is a mannich base derivative based on magnolol and can be used as an anticancer agent. autophagy inducer 4 induces autophagy and thus inhibi..产品型号:T63744 原产地:中国大陆价格: ¥0.0
产品名称: rel-MDM2/4-p53-IN-2;化合物 rel-MDM2/4-p53-IN-2rel-MDM2/4-p53-IN-2
产品简介:rel-mdm2/4-p53-in-2 (2q) is a potent dual mdm2/mdm4 inhibitor and p53 activator that acts on both the mdm2-p53 complex (ic50: 70.7 nm) and the mdm4-p53 complex ..产品型号:T63748 原产地:中国大陆价格: ¥0.0
产品名称: Allopurinol Sodium;1H-吡唑并[3,4-D]嘧啶-4-醇单钠盐Allopurinol sodium salt|||Sodium allopurinol;1H-吡唑并[3,4-D]嘧
产品简介:allopurinol sodium is a xanthine oxidase inhibitor with an ic50 of 7.82±0.12 μm...产品型号:T6376 原产地:中国大陆价格: ¥0.0
产品名称: 4BAB;化合物 4BAB4BAB
产品简介:4bab (compound 29) is an irreversible inhibitor of glyoxalase i (glo1) and exhibits anticancer activity...产品型号:T63944 原产地:中国大陆价格: ¥0.0
产品名称: CYP3A4-IN-1;化合物 CYP3A4-IN-1CYP3A4-IN-1
产品简介:cyp3a4-in-1 is a potent inhibitor of cytochrome p450 3a4 (cyp3a4) (ic50: 0.085 μm)...产品型号:T63954 原产地:中国大陆价格: ¥0.0
产品名称: DPP-4/GPR119 modulator 2;化合物 DPP-4/GPR119 modulator 2DPP-4/GPR119 modulator 2
产品简介:dpp-4/gpr119 modulator 2 is an inhibitor of dipeptidyl peptidase iv (dpp-iv) (ic50: 0.22 μm) and an agonist of gpr119 (ec50: 0.95 μm)...产品型号:T63964 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/mTOR Inhibitor-4;化合物 PI3K/mTOR Inhibitor-4PI3K/mTOR Inhibitor-4
产品简介:pi3k/mtor inhibitor-4 is an orally active pan-i pi3k/mtor inhibitor. pi3k/mtor inhibitor-4 is an enzyme inhibitor that acts on pi3kα (ic50: 0.63 nm), pi3kγ (ic5..产品型号:T63770 原产地:中国大陆价格: ¥0.0
产品名称: PDE1-IN-4;化合物 PDE1-IN-4PDE1-IN-4
产品简介:pde1-in-4 is a potent and selective inhibitor of pde1 (phosphodiesterase-1), acting on pde1c (ic50: 10 nm), pde1a (ic50: 145 nm) and pde1b (ic50: 354 nm). pde1-..产品型号:T63776 原产地:中国大陆价格: ¥0.0
产品名称: AMG 517化合物AMG517AMG517|||N-[4-[[6-[4-(三氟甲基)苯基]-4-嘧啶基]氧基]-2-苯并噻唑基]乙酰胺|||AMG-517
产品简介:amg 517 is an effective and specific trpv1 antagonist, antagonizes proton (ic50: 0.76 nm), capsaicin (ic50: 0.62 nm), and heat activation (ic50: 1.3 nm) of trpv..产品型号:T6379 原产地:中国大陆价格: ¥0.0
产品名称: GID4 Ligand 1;化合物 GID4 Ligand 1GID4 Ligand 1
产品简介:gid4 ligand 1 is a cell-permeable, highly selective gid4 binder with an ic50 value of 5.4 μm and a kd value of 5.6 μm. gid4 ligand 1 is capable of binding gid4 ..产品型号:T63799 原产地:中国大陆价格: ¥0.0
产品名称: Phosphatidylinositol 4,5-bisphosphate;化合物 Phosphatidylinositol 4,5-bisphosphatePhosphatidylinositol
产品简介:phosphatidylinositol 4,5-bisphosphate (l-alpha-phosphatidylinositol-4,5-bisphosphate), serving as a critical phospholipid in cell membranes, functions as a subs..产品型号:T73812 原产地:中国大陆价格: ¥0.0
产品名称: Bosentan-d4;化合物 Bosentan-d4Bosentan-d4
产品简介:bosentan-d4, the deuterium-labeled variant of bosentan, serves as a competitive dual antagonist against endothelin-1 (et) by targeting both et a and et b recept..产品型号:T73820 原产地:中国大陆价格: ¥0.0
产品名称: BRD4 Inhibitor-16;化合物 BRD4 Inhibitor-16BRD4 Inhibitor-16
产品简介:brd4 inhibitor-16 (compound 4) is a potent inhibitor of bromodomain 4 (brd4), whose overexpression is closely correlated with various human cancers through the ..产品型号:T73830 原产地:中国大陆价格: ¥0.0
产品名称: Verucerfont;化合物VerucerfontNBI77860|||GSK561679;NBI77860|||3-(4-甲氧基-2-甲基苯基)-2,5-二甲基-N-[(1S)-1-(3-甲基-1
产品简介:verucerfont (nbi77860) is an antagonist of corticotropin-releasing factor receptor 1 (crf1) ...产品型号:T7361 原产地:中国大陆价格: ¥0.0
产品名称: WDR5-IN-4 TFA;WDR5-IN-4 TFAWDR5-IN-4 TFA
产品简介:wdr5-in-4 tfa is an inhibitor of the win site of chromatin-associated wd repeat-containing protein 5 ( wdr5 ), with a k d of 0.1 nm. wdr5-in-4 tfa displaces wdr..产品型号:T73724 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC AR Degrader-4 TFA;化合物 PROTAC AR Degrader-4 TFAPROTAC AR Degrader-4 TFA
产品简介:protac ar degrader-4, an androgen receptor (ar) degrader, incorporates an iap ligand binding group, a linker, and an ar binding group. it represents a class of ..产品型号:T73726 原产地:中国大陆价格: ¥0.0