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产品名称: SR-3677Inhibitor,Rho-associated protein kinase,Autophagy,SR 3677,Rho-kinase,SR3677,ROCK,ROK,SR-3677,
产品简介:sr-3677 is an effective and specific inhibitor of rock2 (ic50: 3 nm)...产品型号:TQ0187 原产地:中国大陆价格: ¥0.0
产品名称: ValrubicinInhibitor,AD 32,AD32,Valrubicin,inhibit,PKC,Antibiotic,Protein kinase C
产品简介:valrubicin (ad 32) inhibits tpa- and pdbu-induced pkc activation (ic50s: 0.85 and 1.25 μm) and has antitumor and anti-inflammatory activity...产品型号:T7604 原产地:中国大陆价格: ¥0.0
产品名称: Aurora kinase inhibitor-2inhibit,Aurora-A,Aurora kinase inhibitor2,Aurora Kinase,ATP-competitive,Aur
产品简介:aurora kinase inhibitor ii is a cell-permeable anilinoquinazoline that inhibit the activity of aurora a (ic50 = 0.39 m)...产品型号:T9040 原产地:中国大陆价格: ¥0.0
产品名称: HS-1371HS-1371,Inhibitor,Receptor-interacting protein kinases,RIPK,inhibit,HS 1371,RIP kinase,HS1371
产品简介:hs-1371 is a novel kinase inhibitor of receptor-interacting protein kinase 3 (rip3) with an ic50 of 20.8 nm...产品型号:T6815 原产地:中国大陆价格: ¥0.0
产品名称: EMD638683inhibit,EMD-638683,EMD638683,Serum and glucocorticoid-regulated kinase,EMD 638683,Inhibitor
产品简介:emd638683,a novel sgk inhibitor with antihypertensive potency(with an ic50 of 3 μm)...产品型号:T6635 原产地:中国大陆价格: ¥0.0
产品名称: GRK5-IN-2metabolic,bicyclic,insulin,kinase,inhibit,Inhibitor,disease,pyridine-based,GRK5 IN 2,GRK-5-
产品简介:grk5-in-2, a pyridine-based bicyclic compound, is a potent g-protein-coupled receptor kinase 5 (grk5) inhibitor. it regulates the expression and/or release of i..产品型号:T9609 原产地:中国大陆价格: ¥0.0
产品名称: AMG-47aInhibitor,signal,kinases,AMG 47a,JAK,Janus kinase,AMG-47a,transduction,Src,VEGFR,cytoplamic,p
产品简介:amg-47a is a potent inhibitor of lck and t cell proliferation. amg-47a could promote the degradation of the kras oncoprotein. amg-47a selectively reduced the le..产品型号:T7123 原产地:中国大陆价格: ¥0.0
产品名称: SKI VPI3K,SKI V,Inhibitor,Apoptosis,GST-hSK,sphingosine,second,mitogenic,Phosphoinositide 3-kinase,S
产品简介:ski v is a potent and noncompetitive non-lipid sphingosine kinase (sphk; sk) inhibitor (gst-hsk,ic50 : 2 μm), and is a pi3k inhibitor(hpi3k,ic50 : 6 μm), induce..产品型号:T8461 原产地:中国大陆价格: ¥0.0
产品名称: PHA-767491 hydrochloridePHA767491,PHA 767491,inhibit,CAY-10572,Cyclin dependent kinase,CDK,CAY 10572
产品简介:pha-767491 is an effective atp-competitive dual cdc7/cdk9 inhibitor (ic50: 10/34 nm). it has ~20-fold selectivity against gsk3-β and cdk1/2, 50-fold selectivity..产品型号:T6940 原产地:中国大陆价格: ¥0.0
产品名称: CCT129202inhibit,CCT-129202,CCT 129202,Inhibitor,CCT129202,Aurora Kinase
产品简介:cct129202 is an atp-competitive pan-aurora inhibitor for aurora a, aurora b and aurora c with ic50 of 0.042 μm, 0.198 μm and 0.227 μm, respectively. it is less ..产品型号:T6435 原产地:中国大陆价格: ¥0.0
产品名称: GSK1838705ACD246,Anaplastic lymphoma kinase,inhibit,Cluster of differentiation 246,Anaplastic lympho
产品简介:gsk1838705a is an effective igf-1r inhibitor (ic50: 2.0 nm), modestly potent to ir (ic50: 1.6 nm) and alk (ic50: 0.5 nm), respectively, and little inhibition to..产品型号:T3079 原产地:中国大陆价格: ¥0.0
产品名称: Brepocitinibinhibit,Janus kinase,PF06700841,JAK,Brepocitinib,Inhibitor,PF 06700841
产品简介:brepocitinib is a potent dual jak1/tyk2 inhibitor (ic50s: 17 nm/23 nm). brepocitinib also inhibits jak2/3 (ic50s: 77 nm/6.49 μm)...产品型号:TQ0010 原产地:中国大陆价格: ¥0.0
产品名称: SU6656PTK2 protein tyrosine kinase 2,Focal adhesion kinase,FAK,Akt,SU-6656,PTK2,Inhibitor,Protein ki
产品简介:su 6656 is a selective inhibitor of src family kinases, with ic50 of 280 nm, 20 nm, 130 nm, and 170 nm for src, yes, lyn, and fyn, respectively...产品型号:T6997 原产地:中国大陆价格: ¥0.0
产品名称: ON123300Platelet-derived growth factor receptor,AMP-activated protein kinase,ON-123300,ON 123300,FGF
产品简介:on123300 is a potent and multi-targeted kinase inhibitor for cdk4/ark5/pdgfrβ/fgfr1/ret/fyn (ic50: 3.9/5/26/26/9.2/11 nm)...产品型号:T6920 原产地:中国大陆价格: ¥0.0
产品名称: HQ461cyclin K degrader,Cyclin dependent kinase,molecular glue,HQ461,HQ 461,HQ-461,CDK12 substrate ph
产品简介:hq461 is a molecular glue that promotes cdk12-ddb1 interaction to trigger cyclin k degradation, resulting in decreased cdk12 substrate phosphorylation, downregu..产品型号:T9849 原产地:中国大陆价格: ¥0.0
产品名称: CDK-IN-2Inhibitor,CDK IN 2,inhibit,CDK,Cyclin dependent kinase,CDKIN2
产品简介:cdk-in-2 is a potent and specific cdk9 inhibitor (ic50: <8 nm)...产品型号:TQ0078 原产地:中国大陆价格: ¥0.0
产品名称: LY2857785Cyclin dependent kinase,LY 2857785,CDK,Apoptosis,LY2857785,Inhibitor,inhibit,LY-2857785
产品简介:ly2857785 is a type i competitive and reversible atp kinase inhibitor against cdk7/cdk8/cdk9 (ic50s: 246 nm/16 nm/11 nm)...产品型号:TQ0060 原产地:中国大陆价格: ¥0.0
产品名称: PNU112455A hydrochlorideanticooperative,Cyclin dependent kinase,PNU112455A hydrochloride,Alzheimer’s
产品简介:pnu 112455a is an atp site competetive inhibitor of cdk2 and cdk5,binds to the atp site of cdk2 and cdk5 with kms of 3.6 and 3.2 μm, respectively...产品型号:T8230 原产地:中国大陆价格: ¥0.0
产品名称: (E)-Akt inhibitor-IVbreast,PKB,(E) Akt inhibitor IV,PI3K,Inhibitor,Protein kinase B,Akt,inhibit,(E)A
产品简介:(e)-akt inhibitor-iv? ((e)-aktiv) is an inhibitor of pi3k-akt...产品型号:T9393 原产地:中国大陆价格: ¥0.0
产品名称: LJI308viability,Ribosomal S6 Kinase (RSK),LJI-308,stimulation,phosphorylation,LJI308,inhibit,mutatio
产品简介:lji308 is a potent, and pan-rsk (p90 ribosomal s6 kinase) inhibitor with ic50 of 6 nm, 4 nm, and 13 nm for rsk1, rsk2, and rsk3, respectively...产品型号:T6878 原产地:中国大陆价格: ¥0.0