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产品名称: Laninamivir;化合物LaninamivirR 125489;(4S,5R,6R)-5-乙酰氨基-4-胍基-6-((1R,2R)-2,3-二羟基-1-甲氧基丙基)-5,6-二氢-4H-吡喃-2
产品简介:laninamivir (r 125489) is an effective inhibitor of influenza neuraminidase (na) (ic50s: 0.90 nm, 1.83 nm, and 3.12 nm for avian h12n5 na (n5), ph1n1 n1 na (p09..产品型号:T15707 原产地:中国大陆价格: ¥0.0
产品名称: Indibulin;化合物IndibulinZIO 301|||D 24851;2-(1-(4-氯苄基)-1H-吲哚-3-基)-2-氧代-N-(吡啶-4-基)乙酰胺|||ZIO 301|||D 248
产品简介:indibulin (d 24851) is a synthetic small molecule with antimitotic and potential antineoplastic activities.indibulin an orally applicable inhibitor of tubulin a..产品型号:T15576 原产地:中国大陆价格: ¥0.0
产品名称: INDY;化合物INDY1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2-ylidene)propan-2-one;1-(3-ethyl-5-hydroxy-1,3-be
产品简介:indy is an atp-competitive inhibitor of dyrk1a and dyrk1b with ic50s of 0.24 μm and 0.23 μm and a ki of 0.18 μm for dyrk1a atp pocket, respectively...产品型号:T15579 原产地:中国大陆价格: ¥0.0
产品名称: IRL-1620 acetate;化合物IRL-1620 acetateIRL-1620 acetate(142569-99-1 free base);IRL-1620 acetate(142569-
产品简介:irl-1620 acetate is an effective and selective agonist of endothelin b receptor (etb) with a ki of 16 pm which is more selective than eta with a ki of 19 μm. ..产品型号:T15595L 原产地:中国大陆价格: ¥0.0
产品名称: IU1-47;化合物IU1-47IU1-47
产品简介:iu1-47 is an effective and specific usp14 inhibitor (ic50: 0.6 μm). iu1-47 causes tau elimination in cultured neurons. iu1-47 inhibits isot/usp5 (ic50: 20 μm)...产品型号:T15604 原产地:中国大陆价格: ¥0.0
产品名称: JAK1-IN-4;化合物 T15606JAK1-IN-4
产品简介:jak1-in-4 is a selective jak1 inhibitor (ic50s: 85 nm, 12.8 μm and >30 μm for jak1, jak2, and jak3, respectively). jak1-in-4 inhibits stat3 phosphorylation in n..产品型号:T15606 原产地:中国大陆价格: ¥0.0
产品名称: GSK3186899;化合物GSK31868993,3,3-trifluoro-N-[4-[[3-[(2R)-2-methylmorpholin-4-yl]-1H-pyrazolo[3,4-d]pyr
产品简介:gsk3186899 is an inhibitor of cdc2-related kinase 12 with an ec50 of 1.4 μm for l. donovani...产品型号:T15438 原产地:中国大陆价格: ¥0.0
产品名称: Hydroxy-Amino-bis(PEG1-C2-Boc);化合物 T15508Hydroxy-Amino-bis(PEG1-C2-Boc)
产品简介:hydroxy-amino-bis(peg1-c2-boc) is an alkyl/ether-based linker used for the synthesis of protacs[1]...产品型号:T15508 原产地:中国大陆价格: ¥0.0
产品名称: Hydroxy-PEG1-acid;化合物 T15510Hydroxy-PEG1-acid
产品简介:hydroxy-peg1-acid is a non-cleavable 1-unit polyethylene glycol (peg) linker utilized for the synthesis of antibody-drug conjugates (adcs)[1]...产品型号:T15510 原产地:中国大陆价格: ¥0.0
产品名称: Hydroxy-PEG1-C2-methyl ester;化合物 T15511Methyl 3-(2-hydroxyethoxy)propanoate;Methyl 3-(2-hydroxyethox
产品简介:hydroxy-peg1-c2-methyl ester is a polyethylene glycol (peg) derived linker widely employed for the production of protacs - proteolysis targeting chimeras. [1]..产品型号:T15511 原产地:中国大陆价格: ¥0.0
产品名称: Hydroxy-PEG1-(CH2)2-Boc;化合物 T15512Hydroxy-PEG1-(CH2)2-Boc
产品简介:hydroxy-peg1-(ch2)2-boc is a polyethylene glycol (peg)-based linker used in the synthesis of proteolysis-targeting chimeric molecules (protacs)[1]...产品型号:T15512 原产地:中国大陆价格: ¥0.0
产品名称: Hydroxy-PEG1-CH2-Boc;化合物 T15513Hydroxy-PEG1-CH2-Boc
产品简介:hydroxy-peg1-ch2-boc is a peg-based linker for protacs which joins two essential ligands, crucial for forming protac molecules. this linker enables selective pr..产品型号:T15513 原产地:中国大陆价格: ¥0.0
产品名称: Hydroxy-PEG5-Boc1-羟基-3,6,9,12,15-五氧杂十八烷-18-羧酸叔丁酯1-羟基-3,6,9,12,15-五氧杂十八烷-18-羧酸叔丁酯
产品简介:hydroxy-peg6-boc is a peg-based protac linker that can be used in protac synthesis[1]...产品型号:T15534 原产地:中国大陆价格: ¥0.0
产品名称: GPR120 Agonist 3;化合物GPR120 Agonist 3FFAR|||GPR120-IN-1|||GPR120-IN-1|||GPR120 Agonist 3|||GPR120 Ago
产品简介:gpr120 agonist 3 (gpr120-in-1) is a selective agonist of gpr120 ( logec50: -7.62)...产品型号:T15413 原产地:中国大陆价格: ¥0.0
产品名称: GR148672X化合物GR148672X4,4,4-三氟-1-(2-噻吩基)-1,2,3-丁三酮 2-[(3-甲基苯基)腙]
产品简介:gr148672x is an inhibitor of triacyglycerol hydrolase (tgh) (ic50: 4 nm)...产品型号:T15416 原产地:中国大陆价格: ¥0.0
产品名称: KDM5-IN-1;化合物KDM5-IN-1KDM5-IN-1
产品简介:kdm5-in-1 is an effective and selective inhibitor of kdm5 with an ic50 of 15.1 nm...产品型号:T15649 原产地:中国大陆价格: ¥0.0
产品名称: KDM5A-IN-1;KDM5A抑制剂1KDM5A-IN-1
产品简介:kdm5a-in-1 is an orally available, potent and selective inhibitor of the pan-histidine lysine demethylase 5 kdm5, inhibiting kdm5a, kdm5b, and kdm5c with ic50 v..产品型号:T15650 原产地:中国大陆价格: ¥0.0
产品名称: Ketohexokinase inhibitor 1;化合物Ketohexokinase inhibitor 1PF-06835919;PF-06835919
产品简介:ketohexokinase inhibitor 1 is a ketohexokinase inhibitor (ic50s: 8.4 nm and 66 nm for khk-c and khk-a, respectively)...产品型号:T15654 原产地:中国大陆价格: ¥0.0
产品名称: KHK-IN-1 hydrochloride;化合物 T15659KHK-IN-1 hydrochloride
产品简介:khk-in-1 hydrochloride is a potent inhibitor of ketohexokinase (khk) (ic50: 12 nm). in the atp-binding region of khk, khk-in-1 hydrochloride interacts with asp-..产品型号:T15659 原产地:中国大陆价格: ¥0.0
产品名称: KHK-IN-1;化合物KHK-IN-1KHK-IN-8|||Ketohexokinase inhibitor 8;KHK-IN-8|||Ketohexokinase inhibitor 8
产品简介:khk-in-1 (khk-in-8) is a selective and cell membrane permeable inhibitor of ketohexokinase (khk, ic50=12 nm; f=34%). khk-in-1 inhibits f1p production in hepg2 c..产品型号:T15660 原产地:中国大陆价格: ¥0.0