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产品名称: (R)-GSK-3685032;(R)-GSK-3685032(R)-GSK-3685032
产品简介:(r)-gsk-3685032 is the r-enantiomer of gsk-3685032. gsk-3685032 is a first-in-class, non-time-dependent, non-covalent, reversible, selective dnmt1 inhibitor wit..产品型号:T39648 原产地:中国大陆价格: ¥0.0
产品名称: GSK872 HCl(1346546-69-7 free base);化合物GSK872 HClGSK2399872A;GSK2399872A
产品简介:gsk872 hcl(1346546-69-7 free base) (gsk2399872a) is an effective and specific rip3 kinase inhibitor. it binds rip3 kinase domain with high affinity (ic50: 1.8 n..产品型号:T4074L 原产地:中国大陆价格: ¥0.0
产品名称: Umeclidinium bromide;芜地溴铵GSK573719A;芜地溴铵|||GSK573719A
产品简介:umeclidinium bromide (gsk573719a) is a novel machr antagonist...产品型号:T4997 原产地:中国大陆价格: ¥0.0
产品名称: GSK1904529A;化合物GSK1904529AGSK 4529;GSK 4529
产品简介:gsk1904529a (gsk 4529) is a specific inhibitor of igf-1r (ic50=27 nm) and ir(ic50=25 nm) ...产品型号:T6003 原产地:中国大陆价格: ¥0.0
产品名称: GSK1324726A;化合物GSK1324726AI-BET726;I-BET726
产品简介:gsk1324726a (i-bet726) is a greatly specific inhibitor of bet family proteins for brd2(ic50=41 nm), brd3(ic50=31 nm), and brd4 (ic50=22 nm)...产品型号:T6021 原产地:中国大陆价格: ¥0.0
产品名称: GSK2646264;化合物 GSK2646264GSK2646264
产品简介:gsk2646264 (compound 44) is a highly effective and specific inhibitor of spleen tyrosine kinase (syk) with a pic50 of 7.1. in addition to targeting syk, gsk2646..产品型号:T61527 原产地:中国大陆价格: ¥0.0
产品名称: GSK-690693;化合物GSK690693GSK690693;GSK690693
产品简介:gsk-690693 is a pan-akt inhibitor targeting akt1/2/3 with ic50 of 2 nm/13 nm/9 nm, also sensitive to the agc kinase family: pka, prkx and pkc isozymes. phase 1...产品型号:T6285 原产地:中国大陆价格: ¥0.0
产品名称: GSK2945 hydrochloride;化合物 GSK2945 hydrochlorideGSK2945 hydrochloride
产品简介:gsk2945 hydrochloride is a tertiary amine and a highly specific antagonist of rev-erbα/rev-erbα (mouse/human reverse erythropoietic virus α) with an ec50 value ..产品型号:T62852 原产地:中国大陆价格: ¥0.0
产品名称: GSK461364;化合物GSK461364GSK461364A;GSK461364A
产品简介:gsk461364 (gsk461364a)(ki=2.2 nm) inhibits purified plk1 .the specificity of gsk461364 for plk1 is more than 1000-fold over plk2/3...产品型号:T6282 原产地:中国大陆价格: ¥0.0
产品名称: AChE/BACE1/GSK3β-IN-1;化合物 AChE/BACE1/GSK3β-IN-1AChE/BACE1/GSK3β-IN-1
产品简介:ache/bace1/gsk3β-in-1 is an orally active, blood-brain barrier-transparent, moderately bioavailable triple inhibitor of ache/bace1/gsk3β. ache/bace1/gsk3β-in-1 ..产品型号:T62719 原产地:中国大陆价格: ¥0.0
产品名称: GSK-3β inhibitor 7;化合物 GSK-3β inhibitor 7GSK-3β inhibitor 7
产品简介:gsk-3β inhibitor 7 is a gsk-3β inhibitor (ic50: 5.25 μm). gsk-3β inhibitor 7 acts by inserting into the atp-binding binding pocket of gsk-3β and forming hydroge..产品型号:T63866 原产地:中国大陆价格: ¥0.0
产品名称: GSK5852;化合物 GSK5852GSK5852
产品简介:gsk5852 (gsk2485852) is an hcv ns5b rdrp polymerase inhibitor. gsk5852 inhibits ns5b (ic50: 50 nm). gsk5852 exhibits antiviral effects against hepatitis c virus..产品型号:T63936 原产地:中国大陆价格: ¥0.0
产品名称: CDK9/10/GSK3β-IN-1;化合物 CDK9/10/GSK3β-IN-1CDK9/10/GSK3β-IN-1
产品简介:cdk9/10/gsk3β-in-1 is a kinase inhibitor (flavopiridol analogue) that effectively inhibits hsgsk3β, hscdk9/cyclint, hscdk5/p25 and hscdk2/cyclina with ic50 valu..产品型号:T63851 原产地:中国大陆价格: ¥0.0
产品名称: GSK3739936;化合物 GSK3739936GSK3739936
产品简介:gsk3739936 is a potent inhibitor of hiv-1 allosteric integrase (ic50: 11.1 nm, ec50: 1.7 nm). gsk3739936 is also a weak inhibitor of cyp with an ic50 >24.3 μm. ..产品型号:T63977 原产地:中国大陆价格: ¥0.0
产品名称: Verucerfont;化合物VerucerfontNBI77860|||GSK561679;NBI77860|||3-(4-甲氧基-2-甲基苯基)-2,5-二甲基-N-[(1S)-1-(3-甲基-1
产品简介:verucerfont (nbi77860) is an antagonist of corticotropin-releasing factor receptor 1 (crf1) ...产品型号:T7361 原产地:中国大陆价格: ¥0.0
产品名称: GSK2018682;化合物GSK2018682GSK2018682
产品简介:gsk2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pec50s of 7.7 and 7.2,respectively)...产品型号:T7360 原产地:中国大陆价格: ¥0.0
产品名称: Revefenacin;化合物RevefenacinTD-4208|||GSK1160724;TD-4208|||GSK1160724
产品简介:revefenacin (td-4208) is a machr antagonist has a high affinity on m3 receptor( ki : 0.18 nm),and potentially useful for the treatment of respiratory disease...产品型号:T7392 原产地:中国大陆价格: ¥0.0
产品名称: (S,S)-GSK321;化合物 (S,S)-GSK321(S,S)-GSK321
产品简介:(s,s)-gsk321 is a (s,s)-enantiomer of gsk321 [1] ...产品型号:T73929 原产地:中国大陆价格: ¥0.0
产品名称: GSK805;化合物GSK805GSK805
产品简介:gsk805 is a potent, orally bioavailable retinoid-related orphan receptor gamma t (rorγt) inverse agonist that interacts with the receptor´s putative ligan..产品型号:T7388 原产地:中国大陆价格: ¥0.0
产品名称: GSK-2807 free base;化合物 GSK-2807 free baseGSK-2807 free base
产品简介:gsk2807 is a potent and selective, sam-competitive inhibitor of smyd3 (ki = 14 nm). gsk2807 bridges the gap between the sam-binding pocket and the substrate ly..产品型号:T69738 原产地:中国大陆价格: ¥0.0