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产品名称: (1R,3S)-THCCA-Asn;化合物 (1R,3S)-THCCA-Asn(1R,3S)-THCCA-Asn
产品简介:(1r,3s)-thcca-asn (4j) is a selective inhibitor of thrombin (ic50: 0.07-0.14 μm) with anti-thrombotic effects...产品型号:T62949 原产地:中国大陆价格: ¥0.0
产品名称: (S, R)-LSN 3318839;化合物(S,R)-LSN 3318839(S, R)-LSN 3318839(Isomer-2764704-18-7);(S, R)-LSN 3318839(Is
产品简介:产品可用于生物细胞实验..产品型号:T63166L 原产地:中国大陆价格: ¥0.0
产品名称: R547;化合物R547Ro 4584820;Ro 4584820
产品简介:r547 (ro 4584820) is a potent atp-competitive inhibitor of cdk1/2/4 with ki of 2 nm/3 nm/1 nm. it is less potent to cdk7 and gsk3α/β, while inactive to other ki..产品型号:T6312 原产地:中国大陆价格: ¥0.0
产品名称: (R)-MALT1-IN-7;化合物 (R)-MALT1-IN-7(R)-MALT1-IN-7
产品简介:(r)-malt1-in-7 (compound 142a) is a potent inhibitor of malt1 protease and has potential for cancer research...产品型号:T63133 原产地:中国大陆价格: ¥0.0
产品名称: AT1R antagonist 2;化合物 AT1R antagonist 2AT1R antagonist 2
产品简介:at1r antagonist 2 is a potent at1r selective ligand with good at1r affinity (ki: 26 nm)...产品型号:T64122 原产地:中国大陆价格: ¥0.0
产品名称: Laniquidar TFA;拉尼喹达三氟乙酸盐Laniquidar TFA(197509-46-9 Free base)|||R101933;Laniquidar TFA(197509-46-9 F
产品简介:laniquidar tfa (r101933) is a novel orally available non-competitive p-glycoprotein (p-gp) inhibitor with an ic50 value of 0.51 μm.laniquidar has limited bioava..产品型号:T64133L 原产地:中国大陆价格: ¥0.0
产品名称: GLP-1R agonist 10;化合物 GLP-1R agonist 10GLP-1R agonist 10
产品简介:glp-1r agonist 10 is a glp-1 agonist (ec50: 0.051 nm)...产品型号:T64007 原产地:中国大陆价格: ¥0.0
产品名称: 5-HT6R/MAO-B modulator 1;化合物 5-HT6R/MAO-B modulator 15-HT6R/MAO-B modulator 1
产品简介:5-ht6r/mao-b modulator 1 is an antagonist of 5-ht6r at gs signaling and an irreversible inhibitor of mao-b that exhibits glial protective activity. 5-ht6r/mao-b..产品型号:T64036 原产地:中国大陆价格: ¥0.0
产品名称: CSF1R-IN-3;化合物CSF1R-IN-3CSF1R-IN-3
产品简介:csf1r-in-3 is an orally effective csf-1r inhibitor with an ic50 value of 2.1 nm. csf1r-in-3 has anti-proliferative activity against colorectal cancer cells. csf..产品型号:T64066 原产地:中国大陆价格: ¥0.0
产品名称: R-BC154 acetate;化合物 R-BC154 acetateR-BC154 acetate
产品简介:r-bc154 acetate, a selective fluorescent antagonist of α9β1 integrin, serves as a high-affinity, activation-dependent probe for investigating α9β1 and α4β1 inte..产品型号:T74072 原产地:中国大陆价格: ¥0.0
产品名称: (R)-V-0219 hydrochloride;化合物 (R)-V-0219 hydrochloride(R)-V-0219 hydrochloride
产品简介:(r)-v-0219 hydrochloride, an enantiomer of v-0219, functions as an orally active positive allosteric modulator (pam) of the glp-1 receptor (glp-1r). it induces ..产品型号:T74264 原产地:中国大陆价格: ¥0.0
产品名称: (R)-Preclamol hydrochloride;化合物 (R)-Preclamol hydrochloride(R)-Preclamol hydrochloride
产品简介:(r)-preclamol hydrochloride ((+)-3-ppp hydrochloride), the r-enantiomer of preclamol hydrochloride, acts as a da agonist, stimulating both autoreceptors and pos..产品型号:T73685 原产地:中国大陆价格: ¥0.0
产品名称: Talarozole;他拉罗唑R115866;R115866|||他拉罗唑
产品简介:talarozole (r115866) is an oral systemic all-trans retinoic acid metabolism blocking agent (ramba). talarozole inhibits both cyp26a1 and cyp26b1 with ic50s of 5..产品型号:T7370 原产地:中国大陆价格: ¥0.0
产品名称: (3R,5R,6S)-Atogepant;化合物 (3R,5R,6S)-Atogepant(3R,5R,6S)-Atogepant
产品简介:atogepant ((3r,5r,6s)-mk-8031) is the enantiomer of itself and serves as a calcitonin gene-related peptide (cgrp) receptor antagonist, primarily utilized in mig..产品型号:T73703 原产地:中国大陆价格: ¥0.0
产品名称: (R)-Lanicemine;化合物 (R)-Lanicemine(R)-Lanicemine
产品简介:(r)-lanicemine ((r)-azd6765), the less active r-enantiomer of lanicemine, is a low-trapping nmda channel blocker, exhibiting a binding affinity (ki) of 0.56-2.1..产品型号:T73682 原产地:中国大陆价格: ¥0.0
产品名称: TGFβR-IN-1;化合物 TGFβR-IN-1TGFβR-IN-1
产品简介:tgfβr-in-1 is a long-acting tumor-activated proagent of a tgfβr inhibitor...产品型号:T74163 原产地:中国大陆价格: ¥0.0
产品名称: (R)-IDHP;化合物 (R)-IDHP(R)-IDHP
产品简介:(r)-idhp, an isomer of idhp and a metabolite of salvia, exhibits vasorelaxant properties by inhibiting calcium (ca 2+) release and inward flow through both volt..产品型号:T74193 原产地:中国大陆价格: ¥0.0
产品名称: S1R agonist 1;化合物 S1R agonist 1S1R agonist 1
产品简介:compound 6b, also known as s1r agonist 1, is a selective agonist for s1r with dissociation constants (ki) of 0.93 nm for s1r and 72 nm for s2r. this compound de..产品型号:T74822 原产地:中国大陆价格: ¥0.0
产品名称: EGFR T790M/L858R-IN-2;化合物 EGFR T790M/L858R-IN-2EGFR T790M/L858R-IN-2
产品简介:egfrt790m/l858r-in-2 is a potent, selective inhibitor of egfrt790m/l858r, exhibiting ic50 values of 3.5 nm for egfrt790m/l858r and 1290 nm for egfr wt. this com..产品型号:T74833 原产地:中国大陆价格: ¥0.0
产品名称: MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan;化合物 MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-ExatecanMC-Gly-
产品简介:mc-gly-gly-phe-gly-(r)-cyclopropane-exatecan is an agent-linker conjugate for antibody-drug conjugates (adcs), incorporating exatecan, a dna topoisomerase i inh..产品型号:T74723 原产地:中国大陆价格: ¥0.0