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产品名称: AZD8931 diFuMaric acid化合物AZD8931 diFuMaric acid4-[[4-[(3-氯-2-氟苯基)氨基]-7-甲氧基-6-喹唑啉基]氧基]-N-甲基-1-哌啶乙酰胺二富
产品简介:azd8931 is a reversible and atp competitive inhibitor of egfr, erbb2 and erbb3 (ic50 of 4 nm, 3 nm and 4 nm, respectively)...产品型号:T8751 原产地:中国大陆价格: ¥0.0
产品名称: MID-1;化合物MID-1MID-1
产品简介:mid-1 is an inhibitor of mg53-irs-1 (mitsugumin 53-insulin receptor substrate-1) interaction. it disrupts molecular association of mg53 with irs-1 and abolishes..产品型号:T8773 原产地:中国大陆价格: ¥0.0
产品名称: SMBA1;化合物 T8792SMBA1
产品简介:smba1 is a bax activator and a potent bax agonist (ki : 43.3 nm) that induces cell cycle arrest and apoptosis in malignant glioma cells.smba1 has shown antitumo..产品型号:T8792 原产地:中国大陆价格: ¥0.0
产品名称: 1-Methylhistamine dihydrochloride;1-甲基组胺二对甲苯磺酸盐1-Methylhistamine dihydrochloride
产品简介:1-methylhistamine dihydrochloride is a major metabolite of histamine by histamine n-methyltransferase in the pathway of histidine metabolism. it has been used a..产品型号:T8790 原产地:中国大陆价格: ¥0.0
产品名称: TIE-2/VEGFR-2 kinase-IN-1;化合物 T8817TIE-2/VEGFR-2 kinase-IN-1
产品简介:tie-2/vegfr-2 kinase-in-1 is used for the synthesis of tie-2 and/or vegfr-2 inhibitors that can be used for the study of diseases associated with inappropriate ..产品型号:T8817 原产地:中国大陆价格: ¥0.0
产品名称: TC-G 1005化合物TC-G 1005(4-环丙基-3,4-二氢-1(2H)-喹喔啉基)[4-(2,5-二甲基苯氧基)-3-吡啶基]甲酮
产品简介:tc-g 1005 is a potent and selective gpba agonist (ec50 :0.72 nm; htgr5). selective for tgr5 over fxr (farnesoid x receptor). increases plasma glp-1 levels and r..产品型号:T8818 原产地:中国大陆价格: ¥0.0
产品名称: met-kinase-in-2;化合物 T87951,6-Naphthyridin-4(1H)-one, 5-[[3-fluoro-4-[[7-(2-hydroxy-2-methylpropoxy)-
产品简介:met kinase-in-2, a selective and potent met kinase inhibitor, demonstrates oral bioavailability and exhibits an ic50 value of 7.4 nm. it also possesses antitumo..产品型号:T8795 原产地:中国大陆价格: ¥0.0
产品名称: IMT1;化合物LDC195943(IMT1)Propanamide, N,N-dimethyl-2-[[4-(2-methylphenyl)-2-oxo-2H-1-benzopyran-7-yl]o
产品简介:imt1 (propanamide, n,n-dimethyl-2-[[4-(2-methylphenyl)-2-oxo-2h-1-benzopyran-7-yl]oxy]-) has anticancer activity...产品型号:T8841 原产地:中国大陆价格: ¥0.0
产品名称: yGsy2p-IN-1;化合物yGsy2p-IN-1yGsy2p-IN-1
产品简介:ygsy2p-in-1 is a potent yeast glycogen synthase 2 (ygsy2p) and human glycogen synthase 1 (hgys1) inhibitor. ygsy2p-in-h23 a pyrazole inhibitor,and is used for g..产品型号:T8703 原产地:中国大陆价格: ¥0.0
产品名称: Teriparatide acetate;醋酸立特帕肽hPTH 1-34 (acetate salt)|||Parathar acetate|||Forteo;hPTH 1-34 (acetate s
产品简介:teriparatide acetate (forteo) is a pht agonist, with an ic50 of 2 nm in hek293 cells.teriparatide acetate is a recombinant form of parathyroid hormone. it is an..产品型号:T21460 原产地:中国大陆价格: ¥0.0
产品名称: BPR1K871;化合物 T10592DBPR114;DBPR114
产品简介:bpr1k871, a preclinical development candidate for anti-cancer therapy [1], is a potent, selective dual inhibitor targeting flt3 and aurka, with ic50 values of 1..产品型号:T10592 原产地:中国大陆价格: ¥0.0
产品名称: BPR1M97;化合物BPR1M97BPR1M97
产品简介:bpr1m97 is a mu opioid receptor (mop) and neuropeptide-orphin fq (nop) receptor agonist with blood-brain barrier permeability and potency, with kis values of 1...产品型号:T10593 原产地:中国大陆价格: ¥0.0
产品名称: BRCA1-IN-1;化合物 T10600BRCA1-IN-1
产品简介:brca1-in-1 is a novel small-molecule-like inhibitor of brca1 (ic50: 0.53 μm; ki: 0.71 μm)...产品型号:T10600 原产地:中国大陆价格: ¥0.0
产品名称: BRCA1-IN-2;BRCA1 抑制剂2BRCA1-IN-2
产品简介:brca1-in-2 is a cell membrane-crossing brca1 protein-protein interaction (ppi) inhibitor with antitumor activity that acts by disrupting the interaction of brca..产品型号:T10601 原产地:中国大陆价格: ¥0.0
产品名称: BRM/BRG1 ATP Inhibitor-1;化合物BRM/BRG1 ATP Inhibitor-1BRM/BRG1 ATP Inhibitor-1
产品简介:brm/brg1 atp inhibitor-1 is an allosteric dual brahma homolog (brm)/swi/snf related matrix-associated actin-dependent regulator of chromatin subfamily a member ..产品型号:T10616 原产地:中国大陆价格: ¥0.0
产品名称: Bromodomain IN-1;化合物 T10620Bromodomain IN-1
产品简介:bromodomain in-1 is an inhibitor of bromodomain...产品型号:T10620 原产地:中国大陆价格: ¥0.0
产品名称: Asparagusic acid芦笋酸1,2-二噻戊环-4-羧酸|||芦笋酸
产品简介:asparagusic acid is unique to asparagus. it is responsible for the odorous urine excreted after eating asparagus. its derivatives ihydroasparagusic acid have an..产品型号:T10388 原产地:中国大陆价格: ¥0.0
产品名称: ATM Inhibitor-1;化合物 T10396ATM Inhibitor-1
产品简介:atm inhibitor-1 is a highly potent, selective and orally active atm inhibito (ic50: 0.7 nm) anti-tumor activity. it shows weak activity against mtor (ic50, 21 μ..产品型号:T10396 原产地:中国大陆价格: ¥0.0
产品名称: ATP synthase inhibitor 1;化合物ATP synthase inhibitor 1ATP synthase inhibitor 1
产品简介:atp synthase inhibitor 1 is an inhibitor of the c subunit of the f1/fo-atp synthase complex. it inhibits mitochondrial permeability transition pore (mptp) openi..产品型号:T10404 原产地:中国大陆价格: ¥0.0
产品名称: Tuvusertib;化合物TuvusertibM1774|||ATR inhibitor 1;M1774|||ATR inhibitor 1
产品简介:tuvusertib (m1774) is an orally available ataxia telangiectasia and rad3-related (atr) kinase inhibitor (ki< 1 ?μ) with selective and potentially antitumor acti..产品型号:T10406 原产地:中国大陆价格: ¥0.0