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产品目录

产品展示/Products

  • 5-HT6/5-HT2A receptor ligand-1;化合物 5-HT6/5-HT2A receptor ligand-15-HT6/5-HT2A receptor ligand-1

    产品名称: 5-HT6/5-HT2A receptor ligand-1;化合物 5-HT6/5-HT2A receptor ligand-15-HT6/5-HT2A receptor ligand-1

    产品简介:5-ht6/5-ht2a receptor ligand-1 (compound 33) is a dual antagonist for the 5-ht6 and 5-ht2a receptors. it exhibits a k i value of 2 nm and 11 nm for the respecti..

    产品型号:T61207 原产地:中国大陆价格: ¥0.0

  • PDE4-IN-11;化合物 PDE4-IN-11PDE4-IN-11

    产品名称: PDE4-IN-11;化合物 PDE4-IN-11PDE4-IN-11

    产品简介:pde4-in-11 is a potent phosphodiesterase isoenzyme 4 (pde4) inhibitor, exhibiting remarkable bronchodilatory and anti-inflammatory characteristics. it is specif..

    产品型号:T61208 原产地:中国大陆价格: ¥0.0

  • HDAC-IN-27;化合物 HDAC-IN-27HDAC-IN-27

    产品名称: HDAC-IN-27;化合物 HDAC-IN-27HDAC-IN-27

    产品简介:hdac-in-27 是一种有效的口服活性 hdac i 类选择性抑制剂,对 hdac1-3 的 ic 50 值范围为 0.43 至 3.01 nm。抗急性髓系白血病 (aml) 活性。..

    产品型号:T61209 原产地:中国大陆价格: ¥0.0

  • R-PSOP;化合物 R-PSOPR-PSOP

    产品名称: R-PSOP;化合物 R-PSOPR-PSOP

    产品简介:r-psop is a potent and selective nonpeptidic nmur2 antagonist, exhibiting binding affinity to human and rat nmur2 with ki values of 52 nm and 32 nm, respectivel..

    产品型号:T61210 原产地:中国大陆价格: ¥0.0

  • 5-LOX-IN-1;化合物5-LOX-IN-15-LOX-IN-1

    产品名称: 5-LOX-IN-1;化合物5-LOX-IN-15-LOX-IN-1

    产品简介:5-lox-in-1 is a 5-lipoxygenase (5-lox) inhibitor (ic50: 2.3 μm).5-lox-in-1 can be used for cancer research...

    产品型号:T61211 原产地:中国大陆价格: ¥0.0

  • Steroid sulfatase-IN-2;化合物 Steroid sulfatase-IN-2Steroid sulfatase-IN-2

    产品名称: Steroid sulfatase-IN-2;化合物 Steroid sulfatase-IN-2Steroid sulfatase-IN-2

    产品简介:steroid sulfatase-in-2 is an active inhibitor of steroid sulfatase (sts), demonstrating an ic50 value of 109.5 nm. its potential application lies in hormone-dep..

    产品型号:T61212 原产地:中国大陆价格: ¥0.0

  • PF-03654764;化合物PF-03654764PF-03654764

    产品名称: PF-03654764;化合物PF-03654764PF-03654764

    产品简介:pf-03654764 is an orally active, potent, and selective histamine h3 receptor antagonist that inhibits human h3 and rat h3 with ki values of 1.2 nm and 7.9 nm, r..

    产品型号:T61213 原产地:中国大陆价格: ¥0.0

  • EWP 815;化合物EWP 815EWP 815

    产品名称: EWP 815;化合物EWP 815EWP 815

    产品简介:ewp 815 is a disulfiram analogue that functions as a powerful inhibitor of ins(1,4) p 2 phosphatase, ins(1,4,5) p 3 5-phosphatase, and dopamine β-hydroxylase ac..

    产品型号:T61214 原产地:中国大陆价格: ¥0.0

  • Alinidine hydrobromide;化合物 Alinidine hydrobromideAlinidine hydrobromide

    产品名称: Alinidine hydrobromide;化合物 Alinidine hydrobromideAlinidine hydrobromide

    产品简介:alinidine hydrobromide, a specific bradycardic agent, diminishes the slope of the diastolic depolarization in sinoatrial tissue and purkinje fibers [1]...

    产品型号:T61215 原产地:中国大陆价格: ¥0.0

  • Dichlorphenamide disodium;化合物 Dichlorphenamide disodiumDichlorphenamide disodium

    产品名称: Dichlorphenamide disodium;化合物 Dichlorphenamide disodiumDichlorphenamide disodium

    产品简介:dichlorphenamide disodium is a specific, orally active carbonic anhydrase inhibitor. it effectively reduces intraocular pressure by impeding the secretion of aq..

    产品型号:T61216 原产地:中国大陆价格: ¥0.0

  • RSV-IN-3;化合物 RSV-IN-3RSV-IN-3

    产品名称: RSV-IN-3;化合物 RSV-IN-3RSV-IN-3

    产品简介:rsv-in-3 (compound 1) serves as a dual inhibitor targeting both the respiratory syncytial virus (rsv) and influenza virus a (iav), demonstrating anti-rsv effica..

    产品型号:T61217 原产地:中国大陆价格: ¥0.0

  • L-I-OddU;化合物 L-I-OddUL-I-OddU

    产品名称: L-I-OddU;化合物 L-I-OddUL-I-OddU

    产品简介:l-i-oddu, a potent and selective anti-epstein-barr virus (ebv) agent, is a l-5´-halo-dioxolane nucleoside analogue. it demonstrates antiviral activity by ..

    产品型号:T61080 原产地:中国大陆价格: ¥0.0

  • DFPM;化合物 DFPMDFPM

    产品名称: DFPM;化合物 DFPMDFPM

    产品简介:dfpm, a chemical compound, acts as an activator of the plant resistance protein signaling in roots, thereby causing inhibition of root growth. it also reduces t..

    产品型号:T61081 原产地:中国大陆价格: ¥0.0

  • CYP1B1-IN-2;化合物 CYP1B1-IN-2CYP1B1-IN-2

    产品名称: CYP1B1-IN-2;化合物 CYP1B1-IN-2CYP1B1-IN-2

    产品简介:cyp1b1-in-2 (compound 9j) is a highly potent and selective inhibitor of cyp1b1, a cytochrome p450 enzyme. it exhibits an ic50 value of 0.52 nm [1]...

    产品型号:T61082 原产地:中国大陆价格: ¥0.0

  • DN-F01;化合物 DN-F01DN-F01

    产品名称: DN-F01;化合物 DN-F01DN-F01

    产品简介:dn-f01 exhibits a potent calcium-dependent inhibitory effect on cardiac myofibrillar atpase activity, with an ic50 of 11 ± 4 nmol/l...

    产品型号:T61083 原产地:中国大陆价格: ¥0.0

  • Tubulin polymerization-IN-37;化合物 Tubulin polymerization-IN-37Tubulin polymerization-IN-37

    产品名称: Tubulin polymerization-IN-37;化合物 Tubulin polymerization-IN-37Tubulin polymerization-IN-37

    产品简介:tubulin polymerization-in-37 is a potent inhibitor (ic50: 2.3 μμ) of tubulin polymerization by binding specifically to the colchicine site of tubulin and preven..

    产品型号:T61084 原产地:中国大陆价格: ¥0.0

  • TGP-377/421;化合物TGP-377/421Targapre-miR-377/421;Targapre-miR-377/421

    产品名称: TGP-377/421;化合物TGP-377/421Targapre-miR-377/421;Targapre-miR-377/421

    产品简介:tgp-377/421 (targapre-mir-377/421) is a potent mir-377 and mir-421 dual inhibitor that inhibits mir-377 and mir-421 by binding to their functional sites...

    产品型号:T61085 原产地:中国大陆价格: ¥0.0

  • HN37;化合物 HN37HN37

    产品名称: HN37;化合物 HN37HN37

    产品简介:hn37 as a potent and chemically stable antiepileptic drug candidate, with an ec 50 of 37 nm for kcnq2 [1]...

    产品型号:T61086 原产地:中国大陆价格: ¥0.0

  • THK-5105;化合物 THK-5105THK-5105

    产品名称: THK-5105;化合物 THK-5105THK-5105

    产品简介:thk-5105, an arylquinoline derivative, demonstrates a high binding affinity for tau fibrils, protein aggregates, and tau-rich alzheimer´s disease (ad) bra..

    产品型号:T61087 原产地:中国大陆价格: ¥0.0

  • Propiomazine;化合物 PropiomazinePropiomazine

    产品名称: Propiomazine;化合物 PropiomazinePropiomazine

    产品简介:propiomazine is an orally active antihistamine agent that possesses sedative properties. it finds utility in insomnia research [1] [2]...

    产品型号:T61088 原产地:中国大陆价格: ¥0.0

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