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产品名称: mGluR2 modulator 1;化合物 mGluR2 modulator 1mGluR2 modulator 1
产品简介:mglur2 modulator 1 (compound 95) is a potent, blood-brain-barrier permeable modulator of mglur2 (metabotropic glutamate receptor-2) positive transmutation (ec50..产品型号:T62202 原产地:中国大陆价格: ¥0.0
产品名称: CDK9-IN-14;化合物 CDK9-IN-14CDK9-IN-14
产品简介:cdk9-in-14 is a potent, high and low selective cdk9 inhibitor (ic50: 6.92 nm). cdk9-in-14 is a strong inhibitor of mv-4-11 cells and in vivo tumour models with ..产品型号:T62203 原产地:中国大陆价格: ¥0.0
产品名称: Pparδ agonist 7;化合物 Pparδ agonist 7Pparδ agonist 7
产品简介:pparδ agonist 7 is a potent agonist of pparδ. the peroxisome proliferator-activated receptor (ppar) belongs to the intranuclear receptor transcription factor su..产品型号:T62205 原产地:中国大陆价格: ¥0.0
产品名称: Tubulin polymerization-IN-19;化合物 Tubulin polymerization-IN-19Tubulin polymerization-IN-19
产品简介:tubulin aggregation-in-19 (compound 4) is a potent tubulin aggregation inhibitor that has shown potential in breast cancer and drug-resistant colon cancer...产品型号:T62206 原产地:中国大陆价格: ¥0.0
产品名称: KVI-020;化合物 KVI-020KVI-020
产品简介:kvi-020 is a selective, orally active blocker of the atrial potassium channel kv1.5 (ic50: 480 nm). kvi-020 exhibits inhibition of herg (ic50: 15100 nm). kvi-02..产品型号:T62207 原产地:中国大陆价格: ¥0.0
产品名称: Cap-dependent endonuclease-IN-6;化合物 Cap-dependent endonuclease-IN-6Cap-dependent endonuclease-IN-6
产品简介:cap-dependent endonuclease-in-6 (compound 13) is a cap-dependent endonuclease (cen) inhibitor that inhibits influenza virus...产品型号:T62208 原产地:中国大陆价格: ¥0.0
产品名称: HS-276;化合物HS-276HS-276
产品简介:hs-276 is a highly selective, orally active inhibitor of tak1 (ki: 2.5 nm). hs-276 significantly inhibits tak1 (ic50: 8.25 nm), clk2 (ic50: 29 nm), gck (ic50: 2..产品型号:T62209 原产地:中国大陆价格: ¥0.0
产品名称: Antileishmanial agent-10;化合物 Antileishmanial agent-10Antileishmanial agent-10
产品简介:antileishmanial agent-10 (compound 7h) is an antiprotozoal agent...产品型号:T62210 原产地:中国大陆价格: ¥0.0
产品名称: Antifungal agent 33;化合物 Antifungal agent 33Antifungal agent 33
产品简介:antifungal agent 33 (compound 4e) is a potent antifungal agent with significant antifungal activity against candida albicans (mic: 16 μg/ml). (ic50: 0.19 μg/ml)..产品型号:T62211 原产地:中国大陆价格: ¥0.0
产品名称: Antitrypanosomal agent 4;化合物 Antitrypanosomal agent 4Antitrypanosomal agent 4
产品简介:antitrypanosomal agent 4 (compound 19) is a potent antitrypanosomal agent that crosses the blood-brain barrier and shows good resistance to trypanosoma cruzi an..产品型号:T62212 原产地:中国大陆价格: ¥0.0
产品名称: Anagliptin hydrochloride;化合物 Anagliptin hydrochlorideAnagliptin hydrochloride
产品简介:anagliptin (sk-0403) hydrochloride is a potent, highly selective, orally active inhibitor of dipeptidyl peptidase 4 (dpp-4) (ic50: 3.8 nm) with relatively weak ..产品型号:T62213 原产地:中国大陆价格: ¥0.0
产品名称: Tandospirone hydrochloride;化合物 Tandospirone hydrochlorideTandospirone hydrochloride
产品简介:tandospirone (sm-3997) hydrochloride is a potent, selective 5-ht1a receptor partial agonist (ki: 27 nm) that exhibits anxiolytic and antidepressant activity. ta..产品型号:T62215 原产地:中国大陆价格: ¥0.0
产品名称: Influenza virus-IN-5;化合物 Influenza virus-IN-5Influenza virus-IN-5
产品简介:influenza virus-in-5 (compound 5f) is an influenza virus hemagglutinin (ha) inhibitor that acts on the a/h3n2 virus (ec50: 1 nm)...产品型号:T62216 原产地:中国大陆价格: ¥0.0
产品名称: Tubulin polymerization-IN-9;化合物 Tubulin polymerization-IN-9Tubulin polymerization-IN-9
产品简介:tubulin polymerization-in-9 is a potent inhibitor of tubulin (ic50: 1.82 μm). tubulin polymerization-in-9 arrests the cell cycle of k562 cells in g2/m phase and..产品型号:T62217 原产地:中国大陆价格: ¥0.0
产品名称: Parapenzolate bromide;化合物 Parapenzolate bromideParapenzolate bromide
产品简介:parapenzolate bromide is an orally active machr antagonist. parapenzolate bromide is an anticholinergic and antitussive agent...产品型号:T62218 原产地:中国大陆价格: ¥0.0
产品名称: NN-390;化合物 NN-390NN-390
产品简介:nn-390 is a selective, potent hdac6 inhibitor (ic50: 9.8 μm) that crosses the blood-brain barrier. nn-390 has potential for studies in metastatic group 3 neural..产品型号:T62219 原产地:中国大陆价格: ¥0.0
产品名称: PFI-1;化合物PFI1PF-6405761|||PFI 1|||PFI1;PF-6405761|||PFI 1|||PFI1
产品简介:pfi-1 (pf-6405761), a specific bet (bromodomain-containing protein) inhibitor for brd4, is with the ic50 of 0.22 μm in a cell-free assay...产品型号:T6222 原产地:中国大陆价格: ¥0.0
产品名称: DGAT1-IN-3;化合物 DGAT1-IN-3DGAT1-IN-3
产品简介:dgat1-in-3 is a selective, potent, orally active dgat-1 inhibitor that inhibits human dgat-1 (ic50: 38 nm) and rat dgat-1 (ic50: 120 nm).dgat1-in-3 can be used ..产品型号:T62220 原产地:中国大陆价格: ¥0.0
产品名称: NLRP3-IN-8;化合物 NLRP3-IN-8NLRP3-IN-8
产品简介:nlrp3-in-8 (compound 27), an orally active nlrp3 inflammasome inhibitor, directly binds to its target with an ic50 of 1.23 μm for il-1β inhibition. it demonstra..产品型号:T62221 原产地:中国大陆价格: ¥0.0
产品名称: α-Glucosidase-IN-11;化合物 α-Glucosidase-IN-11α-Glucosidase-IN-11
产品简介:α-glucosidase-in-11 is a highly permeable competitive inhibitor of α-glucosidase (ic50: 0.56 μm). α-glucosidase-in-11 binds to the trp residue in α-glucosidase ..产品型号:T62222 原产地:中国大陆价格: ¥0.0