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产品名称: pan-HER-IN-1;化合物 pan-HER-IN-1pan-HER-IN-1
产品简介:pan-her-in-1 (compound c5) is an irreversible, orally active pan- her inhibitor. pan-her-in-1 exhibits ic 50s of 0.38, 1.6, 2.2 and 3.5 nm for egfr, her4, egfr ..产品型号:T62047 原产地:中国大陆价格: ¥0.0
产品名称: Topo I-IN-1;化合物 Topo I-IN-1Topo I-IN-1
产品简介:topo i-in-1 (compound 14d) is a potent topo i inhibitor. topo i-in-1 exhibits antitumor activity and dna intercalative capability. topo i-in-1 can induce cell a..产品型号:T62048 原产地:中国大陆价格: ¥0.0
产品名称: CTX-712;化合物 CTX-712CTX-712
产品简介:ctx-712 is a potent inhibitor of cdc2-like kinase ( clk ). ctx-712 inhibits inhibits cancer survival and cancer cell growth...产品型号:T62049 原产地:中国大陆价格: ¥0.0
产品名称: AT7519;化合物AT7519AT7519
产品简介:at7519 is a cdk1/2/4/6/9 inhibitor (ic50: 10-210 nm). it is less effective to cdk3 and little active to cdk7...产品型号:T6205 原产地:中国大陆价格: ¥0.0
产品名称: Orexin receptor antagonist 4;化合物 Orexin receptor antagonist 4Orexin receptor antagonist 4
产品简介:orexin receptor antagonist 4 is potent and selective orexin 2 receptor (ox2r) antagonist. orexin receptor antagonist 4 shows ic50 of 4.27 nm and 295 nm for ox2r..产品型号:T62050 原产地:中国大陆价格: ¥0.0
产品名称: (R)-(+)-Dimethindene maleate;化合物 (R)-(+)-Dimethindene maleate(R)-(+)-Dimethindene maleate
产品简介:(r)-(+)-dimethindene maleate is an orally active h 1 -receptor blocker...产品型号:T62051 原产地:中国大陆价格: ¥0.0
产品名称: AMPK activator 6;化合物 AMPK activator 6AMPK activator 6
产品简介:ampk activator 6 (compound gc) activates the ampk pathway and reduces lipid content in hepg2 and 3t3-l1 cells. ampk activator 6 significantly suppresses the inc..产品型号:T62052 原产地:中国大陆价格: ¥0.0
产品名称: Lorpucitinib;化合物LorpucitinibJNJ-64251330;JNJ-64251330
产品简介:lorpucitinib (jnj-64251330) is an orally available, selective and potent jak kinase inhibitor for the study of inflammatory and gastrointestinal disorders assoc..产品型号:T62053 原产地:中国大陆价格: ¥0.0
产品名称: D4R antagonis-2;化合物 D4R antagonis-2D4R antagonis-2
产品简介:d4r antagonist-2 is a potent and selective d4r antagonist (ic50= 6.52 μm). d4r antagonist-2 displays favorable in vitro pk parameters and exhibits good brain pe..产品型号:T62054 原产地:中国大陆价格: ¥0.0
产品名称: NVS-BET-1;化合物 NVS-BET-1NVS-BET-1
产品简介:nvs-bet-1 is a bet bromodomain inhibitor. nvs-bet-1 can regulate keratinocyte plasticity...产品型号:T62055 原产地:中国大陆价格: ¥0.0
产品名称: (E/Z)-Zotiraciclib hydrochloride;化合物 (E/Z)-Zotiraciclib hydrochloride(E/Z)-Zotiraciclib hydrochlorid
产品简介:(e/z)-zotiraciclib ((e/z)-tg02) hydrochloride is a potent inhibitor of cdk2, jak2, and flt3...产品型号:T62056 原产地:中国大陆价格: ¥0.0
产品名称: TLR9-IN-1;化合物 TLR9-IN-1TLR9-IN-1
产品简介:tlr9-in-1 is a selective and potent tlr9 inhibitor that acts on human tlr9 (ic50: 7 nm). tlr9-in-1 can be used in the study of adverse immune response-related d..产品型号:T62254 原产地:中国大陆价格: ¥0.0
产品名称: 20S Proteasome-IN-4;化合物 20S Proteasome-IN-420S Proteasome-IN-4
产品简介:20s proteasome-in-4 (compound 7) is an orally active inhibitor of the 20s proteasome, selectively targeting the parasite form and demonstrating brain penetratio..产品型号:T62255 原产地:中国大陆价格: ¥0.0
产品名称: HBV-IN-11;化合物 HBV-IN-11HBV-IN-11
产品简介:hbv-in-11 is a potent inhibitor of hbsag secretion (ec50: 0.46 μm)...产品型号:T62256 原产地:中国大陆价格: ¥0.0
产品名称: Ten01;化合物 Ten01Ten01
产品简介:ten01 exhibits a 5.0 nm inhibition of jak1 kinase...产品型号:T62257 原产地:中国大陆价格: ¥0.0
产品名称: Bestatin trifluoroacetate;化合物 Bestatin trifluoroacetateBestatin trifluoroacetate
产品简介:bestatin trifluoroacetate (ubenimex trifluoroacetate) is a cd13 (aminopeptidase n)/apn and leukotriene a4 hydrolase inhibitor that is often used in cancer resea..产品型号:T62258 原产地:中国大陆价格: ¥0.0
产品名称: COX-2-IN-21;化合物 COX-2-IN-21COX-2-IN-21
产品简介:cox-2-in-21 (compound 5c) is an orally active, selective cox-2 inhibitor (ic50: 0.039 μm). cox-2-in-21 has good anti-inflammatory potential...产品型号:T62259 原产地:中国大陆价格: ¥0.0
产品名称: FLT3-IN-11;化合物 FLT3-IN-11FLT3-IN-11
产品简介:flt3-in-11 (compound 30) is an orally active, potent and selective inhibitor of flt3 kinase, acting on wild-type flt3 (ic50: 7.22 nm) and flt3-d835y (ic50: 4.95..产品型号:T62260 原产地:中国大陆价格: ¥0.0
产品名称: GPR84 antagonist 1;化合物 GPR84 antagonist 1GPR84 antagonist 1
产品简介:gpr84 antagonist 1 is a highly selective, high-affinity competitive antagonist of human gpr84...产品型号:T62261 原产地:中国大陆价格: ¥0.0
产品名称: Neuroinflammatory-IN-2;化合物 Neuroinflammatory-IN-2Neuroinflammatory-IN-2
产品简介:neuroinflammatory-in-2 (compound 7i) is a potent anti-neuroinflammatory agent, capable of acting on mao-b (ic50: 10.30 μm). neuroinflammatory-in-2 inhibits 96.3..产品型号:T62262 原产地:中国大陆价格: ¥0.0