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产品目录

产品展示/Products

  • VildagliptinVildagliptin,NVP-LAF 237,LAF237

    产品名称: VildagliptinVildagliptin,NVP-LAF 237,LAF237

    产品简介:vildagliptin is a cyanopyrrolidine-based, orally bioavailable inhibitor of dipeptidyl peptidase 4 (dpp-4), with hypoglycemic activity. vildagliptin´s cyan..

    产品型号:T1502 原产地:美洲价格: ¥0.0

  • Buparlisib HydrochlorideBuparlisib Hydrochloride,BKM120 Hydrochloride,NVP-BKM120 Hydrochloride

    产品名称: Buparlisib HydrochlorideBuparlisib Hydrochloride,BKM120 Hydrochloride,NVP-BKM120 Hydrochloride

    产品简介:buparlisib hydrochloride is an inhibitor of pan-class i pi3k (ic50: 52 nm/166 nm/116 nm/262 nm for p110α/p110β/p110δ/p110γ, respectively)...

    产品型号:T16365 原产地:美洲价格: ¥0.0

  • Infigratinib phosphateInfigratinib phosphate,BGJ-398 phosphate,NVP-BGJ398 phosphate

    产品名称: Infigratinib phosphateInfigratinib phosphate,BGJ-398 phosphate,NVP-BGJ398 phosphate

    产品简介:infigratinib phosphate is an effective inhibitor of the fgfr family (ic50: 0.9 nm, 1.4 nm, 1 nm, and 60 nm for fgfr1, fgfr2, fgfr3, and fgfr4, respectively)...

    产品型号:T16364 原产地:美洲价格: ¥0.0

  • NVP-2NVP-2

    产品名称: NVP-2NVP-2

    产品简介:nvp-2 is an effective and selective atp-competitive cyclin-dependent kinase 9 (cdk9) probe. nvp-2 induces cell apoptosis. nvp-2 inhibits cdk9/cyct activity (ic5..

    产品型号:T16363 原产地:美洲价格: ¥0.0

  • NVP 231NVP 231

    产品名称: NVP 231NVP 231

    产品简介:nvp-231 is a potent, specific and reversible cerk inhibitor(ic50=12±2 nm) that competitively inhibits ceramide binding to cerk...

    产品型号:T1933 原产地:美洲价格: ¥0.0

  • BuparlisibBuparlisib,BKM120,NVP-BKM120

    产品名称: BuparlisibBuparlisib,BKM120,NVP-BKM120

    产品简介:buparlisib is an orally bioavailable specific oral inhibitor of the pan-class i pi3k (ic50s: 52/166/116/nm for p110α, p110β, and p110δ)...

    产品型号:T1827 原产地:美洲价格: ¥0.0

  • SonidegibSonidegib,NVP-LDE225,Erismodegib

    产品名称: SonidegibSonidegib,NVP-LDE225,Erismodegib

    产品简介:lde225 (nvp-lde225; erismodegib), a smoothened (smo) antagonist, inhibits hedgehog (hh) signaling with ic50 of 1.3 nm (mouse) and 2.5 nm (human), respectively...

    产品型号:T1926 原产地:美洲价格: ¥0.0

  • TAE226TAE226,NVP-TAE 226,

    产品名称: TAE226TAE226,NVP-TAE 226,

    产品简介:nvp-tae226 is an effective fak inhibitor (ic50: 5.5 nm) and most effective to pyk2(ic50: 3.5 nm); 10- to 100-fold less effective against igf-1r, insr, c-met, an..

    产品型号:T1918 原产地:美洲价格: ¥0.0

  • NVP-BHG712 isomerNVP-BHG712 isomer

    产品名称: NVP-BHG712 isomerNVP-BHG712 isomer

    产品简介:nvp-bhg712 isomer shows conserved non-bonded binding to epha2 and ephb4...

    产品型号:T19487 原产地:美洲价格: ¥0.0

  • InfigratinibInfigratinib,NVP-BGJ398,BGJ-398

    产品名称: InfigratinibInfigratinib,NVP-BGJ398,BGJ-398

    产品简介:infigratinib (bgj398) is an orally bioavailable pan fgfr inhibitor (ic50: 0.9/1.4/1 nm for fgfr1/2/3), >40-fold selective for fgfr versus fgfr4 and vegfr2...

    产品型号:T1975 原产地:美洲价格: ¥0.0

  • NVP-BVU972NVP-BVU972

    产品名称: NVP-BVU972NVP-BVU972

    产品简介:nvp-bvu972 is a selective and potent met inhibitor with ic50 of 14 nm...

    产品型号:T2680 原产地:美洲价格: ¥0.0

  • PanobinostatPanobinostat,NVP-LBH589,LBH589

    产品名称: PanobinostatPanobinostat,NVP-LBH589,LBH589

    产品简介:panobinostat is a potent inhibitor of all hdacs (kis: 0.6-31 nm for hdac1-11)...

    产品型号:T2383 原产地:美洲价格: ¥0.0

  • TAE684TAE684,NVP-TAE 684,

    产品名称: TAE684TAE684,NVP-TAE 684,

    产品简介:nvp-tae 684 is a excellently effective and specific alk inhibitor(ic50=3 nm)...

    产品型号:T2251 原产地:美洲价格: ¥0.0

  • DactolisibDactolisib,NVP-BEZ235,BEZ235

    产品名称: DactolisibDactolisib,NVP-BEZ235,BEZ235

    产品简介:dactolisib is an orally bioavailable inhibitor of pi3k and mtor (ic50s: 4 nm/5 nm/7 nm/75 nm, and 20.7 nm for p110α/p110γ/p110δ/p110β and mtor)...

    产品型号:T2235 原产地:美洲价格: ¥0.0

  • AEE788AEE788,NVP-AEE 788,

    产品名称: AEE788AEE788,NVP-AEE 788,

    产品简介:aee788 has been used in trials studying the treatment of cancer, glioblastoma multiforme, and brain and central nervous system tumors...

    产品型号:T2116 原产地:美洲价格: ¥0.0

  • NVP-BEP800NVP-BEP800,VER-82576,

    产品名称: NVP-BEP800NVP-BEP800,VER-82576,

    产品简介:nvp-bep800, a synthetic hsp90β inhibitor (ic50: 58 nm), exhibits >70-fold selectivity against hsp90 family members trap-1 and grp94...

    产品型号:T2114 原产地:美洲价格: ¥0.0

  • NVP-BSK805NVP-BSK805,BSK 805,NVP-BSK805 2HCl

    产品名称: NVP-BSK805NVP-BSK805,BSK 805,NVP-BSK805 2HCl

    产品简介:nvp-bsk805 is an atp-competitive jak2 inhibitor...

    产品型号:T5049 原产地:美洲价格: ¥0.0

  • NVP-AEW541NVP-AEW541,AEW541,

    产品名称: NVP-AEW541NVP-AEW541,AEW541,

    产品简介:nvp-aew541, a potent inhibitor of igf-1r(ic50=150 nm) and insr(ic50=140 nm), exhibits excellent efficiency and specificity for igf-1r in a cell-based assay...

    产品型号:T6080 原产地:美洲价格: ¥0.0

  • NVP-ADW742NVP-ADW742,ADW,GSK 552602A

    产品名称: NVP-ADW742NVP-ADW742,ADW,GSK 552602A

    产品简介:nvp-adw742 is an igf-1r inhibitor with ic50 of 0.17 μm, >16-fold more potent against igf-1r than insr; little activity to her2, pdgfr, vegfr-2, bcr-abl and ..

    产品型号:T6079 原产地:美洲价格: ¥0.0

  • BGT226BGT226,BGT226 maleate,NVP-BGT226 (maleate)

    产品名称: BGT226BGT226,BGT226 maleate,NVP-BGT226 (maleate)

    产品简介:bgt226 (nvp-bgt226) is a class i pi3k/mtor inhibitor for pi3kα/β/γ (ic50: 4/63/38 nm) ...

    产品型号:T6072 原产地:美洲价格: ¥0.0

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