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产品名称: PROTAC CDK12/13 Degrader-1;化合物 PROTAC CDK12/13 Degrader-1PROTAC CDK12/13 Degrader-1
产品简介:protac cdk12/13 degrader-1 (7f) is a potent and selective dual degrader of the cell cycle protein-dependent kinases cdk12 (dc50: 2.2 nm) and cdk13 (dc50: 2.1 nm..产品型号:T64284 原产地:中国大陆价格: ¥0.0
产品名称: Protease-Activated Receptor-1 antagonist 2;化合物 Protease-Activated Receptor-1 antagonist?2Protease-Ac
产品简介:protease-activated receptor-1 antagonist 2 is a selective, orally active protease-activated receptor-1 (par-1) antagonist (ic50: 7 nm). it has shown good pharma..产品型号:T64285 原产地:中国大陆价格: ¥0.0
产品名称: Quinidine polygalacturonate;化合物 Quinidine polygalacturonateQuinidine polygalacturonate
产品简介:quinidine polygalacturonate is a potent, selective, orally active inhibitor of cytochrome p450db (cytochrome p450db) and a potent k+channel blocker with an ic50..产品型号:T64286 原产地:中国大陆价格: ¥0.0
产品名称: Reteplase;化合物 ReteplaseReteplase
产品简介:reteplase (bm 06.022) is a recombinant plasminogen activator consisting of the kringle 2 and protease domains of human tissue-type fibrinogen activator. retepla..产品型号:T64287 原产地:中国大陆价格: ¥0.0
产品名称: RG7800 hydrochloride;化合物 RG7800 hydrochlorideRG7800 hydrochloride
产品简介:rg7800 hydrochloride is an orally active smn2 splicing modulator that acts on smn2 splicing (ec1.5x: 23 nm) and smn proteins (ec1.5x: 87 nm)...产品型号:T64288 原产地:中国大陆价格: ¥0.0
产品名称: Rucaparib camsylate;化合物 Rucaparib camsylateRucaparib camsylate
产品简介:rucaparib (ag014699) camsylate is an orally active inhibitor of parp proteins (parp-1, parp-2 and parp-3) with a ki=1.4 nm for parp-1. rucaparib camsylate is an..产品型号:T64289 原产地:中国大陆价格: ¥0.0
产品名称: SCO-792;化合物 SCO-792SCO-792
产品简介:sco-792 is a potent, reversible, orally active inhibitor of enteropeptidase, which slowly dissociates from enteropeptidase in vitro and inhibits protein digesti..产品型号:T64290 原产地:中国大陆价格: ¥0.0
产品名称: sEH inhibitor-1;化合物 sEH inhibitor-1sEH inhibitor-1
产品简介:seh inhibitor-1 (compound tcpu) is a potent, orally active inhibitor of soluble epoxide hydrolase (seh) with ic50 values of 0.4 and 5.3 nm for human and murine ..产品型号:T64291 原产地:中国大陆价格: ¥0.0
产品名称: Simvastatin acid calcium hydrate;化合物 Simvastatin acid calcium hydrateSimvastatin acid calcium hydrat
产品简介:simvastatin acid (tenivastatin) calcium hydrate is an orally active inhibitor of hmg-coa reductase (hmgcr). simvastatin acid calcium hydrate also inhibits indox..产品型号:T64292 原产地:中国大陆价格: ¥0.0
产品名称: SLN124;化合物 SLN124SLN124
产品简介:sln124 is a galnac-sirna that targets transmembrane serine protease 6 (tmprss6) and consists of a trimeric galnac ligand bound to tmprss6-sirna. sln124 has the ..产品型号:T64293 原产地:中国大陆价格: ¥0.0
产品名称: Succinic acid sodium;化合物 Succinic acid sodiumSuccinic acid sodium
产品简介:succinic acid sodium is an orally active anxiolytic. succinic acid sodium down-regulates the expression of kcnmb1 (potassium channel subunit β1) and tet1 (10-11..产品型号:T64294 原产地:中国大陆价格: ¥0.0
产品名称: TIY-7;化合物 TIY-7TIY-7
产品简介:tiy-7 is a selective, orally active inhibitor of the promyosin receptor kinase (trk) enzyme. tiy-7 exhibited anti-tumour effects in a mouse xenograft model...产品型号:T64296 原产地:中国大陆价格: ¥0.0
产品名称: Turoctocog alfa;化合物 Turoctocog alfaTuroctocog alfa
产品简介:turoctocog alfa is a recombinant coagulation factor viii (fviii) derived from chinese hamster ovary (cho) cells. turoctocog alfa can be used in the study of hae..产品型号:T64298 原产地:中国大陆价格: ¥0.0
产品名称: Valacyclovir hydrochloride hydrate;化合物 Valacyclovir hydrochloride hydrateValacyclovir hydrochloride
产品简介:valacyclovir hydrochloride hydrate is a potent antiviral agent, a prodrug that is rapidly converted to acyclovir in vivo. valacyclovir hydrochloride hydrate can..产品型号:T64299 原产地:中国大陆价格: ¥0.0
产品名称: Vimirogant hydrochloride;化合物 Vimirogant hydrochlorideVimirogant hydrochloride
产品简介:vimirogant (vtp-43742) hydrochloride is an orally active, selective rorγt inhibitor (ic50: 17 nm, ki: 3.5 nm) that is more than 1000 times more selective than r..产品型号:T64300 原产地:中国大陆价格: ¥0.0
产品名称: VU6028418;化合物 VU6028418VU6028418
产品简介:vu6028418 is a highly selective, potent, orally active m4machr antagonist that acts on hm4 (ic50: 4.1 nm)...产品型号:T64301 原产地:中国大陆价格: ¥0.0
产品名称: DX3-235;化合物 DX3-235DX3-235
产品简介:dx3-235 is an inhibitor of oxidative phosphorylation (oxphos). in galactose-containing media, dx3-235 inhibits complex i function and atp production by nanomola..产品型号:T64108 原产地:中国大陆价格: ¥0.0
产品名称: COX-2-IN-28;化合物 COX-2-IN-28COX-2-IN-28
产品简介:cox-2-in-28 is a potent and selective cox-2 inhibitor capable of acting on cox-2 (ic50: 0.054 μm), 15-lox (ic50: 2.14 μm) and cox-1 (ic50: 13.21 μm)...产品型号:T64109 原产地:中国大陆价格: ¥0.0
产品名称: Debio 0617B;化合物 Debio 0617BDebio 0617B
产品简介:debio 0617b is a multi-kinase inhibitor that reduces maintenance and self-renewal of primary human aml cd34+ stem/progenitor cells. debio 0617b targets key kina..产品型号:T64110 原产地:中国大陆价格: ¥0.0
产品名称: Antitumor agent-76;化合物 Antitumor agent-76Antitumor agent-76
产品简介:antitumor agent-76 is a water-soluble, orally active, rapid-release prodrug of triptolide that exhibits anticancer effects...产品型号:T64111 原产地:中国大陆价格: ¥0.0