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产品目录

产品展示/Products

  • MPM-1;化合物 MPM-1MPM-1

    产品名称: MPM-1;化合物 MPM-1MPM-1

    产品简介:mpm-1, a mimic of marine eusynstyelamides, serves as an effective anticancer agent. it swiftly induces a necrosis-like death in cancer cells in vitro, facilitat..

    产品型号:T73544 原产地:中国大陆价格: ¥0.0

  • CPUL1;化合物 CPUL1CPUL1

    产品名称: CPUL1;化合物 CPUL1CPUL1

    产品简介:cpul1, a trxr inhibitor, exhibits proliferation-inhibitory and anti-metastatic effects on a549 cells by modulating epithelial-mesenchymal transition (emt) throu..

    产品型号:T73547 原产地:中国大陆价格: ¥0.0

  • PTP1B-IN-1;5-苯基-1,2,5-噻二唑烷-3-酮 1,1-二氧化物PTP1B inhibitor;PTP1B inhibitor|||5-苯基-1,2,5-噻二唑烷-3-酮 1,1-二氧化

    产品名称: PTP1B-IN-1;5-苯基-1,2,5-噻二唑烷-3-酮 1,1-二氧化物PTP1B inhibitor;PTP1B inhibitor|||5-苯基-1,2,5-噻二唑烷-3-酮 1,1-二氧化

    产品简介:ptp1b-in-1 (ptp1b inhibitor) is a potent inhibitor of protein tyrosine phosphatase 1b (ptp1b) (ic50 : 1.6 mm)..

    产品型号:T7356 原产地:中国大陆价格: ¥0.0

  • DRP1i27;化合物 DRP1i27DRP1i27

    产品名称: DRP1i27;化合物 DRP1i27DRP1i27

    产品简介:drp1i27, a potent human dynamin-related protein 1 (drp1) inhibitor, targets the gtpase site of drp1, forming hydrogen bonds with gln34 and asp218. it mitigates ..

    产品型号:T73456 原产地:中国大陆价格: ¥0.0

  • PARL-IN-1;化合物 PARL-IN-1PARL-IN-1

    产品名称: PARL-IN-1;化合物 PARL-IN-1PARL-IN-1

    产品简介:parl-in-1, a potent parl inhibitor, exhibits an ic50 value of 28 nm. it effectively inhibits parl, consequently robustly activating the pink1/parkin pathway and..

    产品型号:T73324 原产地:中国大陆价格: ¥0.0

  • MenA-IN-1;化合物 MenA-IN-1MenA-IN-1

    产品名称: MenA-IN-1;化合物 MenA-IN-1MenA-IN-1

    产品简介:mena in-1, a potent inhibitor of 1,4-dihydroxy-2-naphthoate isoprenyltransferase (mena) from mycobacterium tuberculosis (mtb), exhibits an ic50 value of 13 ?m a..

    产品型号:T73325 原产地:中国大陆价格: ¥0.0

  • NP118809;化合物NP11880939-1B4;39-1B4|||1-【4-(二苯甲基)-1-哌嗪基】-3,3-二苯基-1-丙酮

    产品名称: NP118809;化合物NP11880939-1B4;39-1B4|||1-【4-(二苯甲基)-1-哌嗪基】-3,3-二苯基-1-丙酮

    产品简介:np118809 (39-1b4) is a potent n-type calcium channel blocker(ic50 : 0.11 μm)...

    产品型号:T7334 原产地:中国大陆价格: ¥0.0

  • Quipazine化合物 Quipazine2-(1-哌嗪基)喹啉

    产品名称: Quipazine化合物 Quipazine2-(1-哌嗪基)喹啉

    产品简介:quipazine, a 5-ht (serotonin) agonist, demonstrates affinity for the 5-ht3r receptor in rats with a ki value of 1.4 nm, effectively displacing gr65630. it exhib..

    产品型号:T73341 原产地:中国大陆价格: ¥0.0

  • BAP1-IN-1;化合物 BAP1-IN-1BAP1-IN-1

    产品名称: BAP1-IN-1;化合物 BAP1-IN-1BAP1-IN-1

    产品简介:bap1-in-1 is a catalytic activity inhibitor of brca1 associated protein 1 (bap1), exhibiting an inhibitory concentration (ic50) ranging between 0.1-1 μm...

    产品型号:T73343 原产地:中国大陆价格: ¥0.0

  • Nelotanserin;化合物NelotanserinAPD125;1-[3-(4-溴-1-甲基-1H-吡唑-5-基)-4-甲氧基苯基]-3-(2,4-二氟苯基)脲|||APD125

    产品名称: Nelotanserin;化合物NelotanserinAPD125;1-[3-(4-溴-1-甲基-1H-吡唑-5-基)-4-甲氧基苯基]-3-(2,4-二氟苯基)脲|||APD125

    产品简介:nelotanserin (apd125) is a potent 5-ht2a inverse agonist(ic50 : 1.7 nm), a moderately potent 5-ht2c partial inverse agonist t(ic50 :79 nm )and a weak 5-ht2b inv..

    产品型号:T7350 原产地:中国大陆价格: ¥0.0

  • GY1-22;化合物 GY1-22GY1-22

    产品名称: GY1-22;化合物 GY1-22GY1-22

    产品简介:gy1-22, an inhibitor targeting the dnaja1-mutp53 r175h interaction pocket, holds potential for cancer research applications...

    产品型号:T73505 原产地:中国大陆价格: ¥0.0

  • Pridopidine;4-[3-(甲磺酰基)苯基]-1-丙基哌啶ACR16|||ASP2314|||FR310826;ACR16|||ASP2314|||FR310826|||4-[3-(甲磺酰基)

    产品名称: Pridopidine;4-[3-(甲磺酰基)苯基]-1-丙基哌啶ACR16|||ASP2314|||FR310826;ACR16|||ASP2314|||FR310826|||4-[3-(甲磺酰基)

    产品简介:pridopidine (fr310826), a dopamine (da) stabilizer, acts as a low affinity dopamine d2 receptor (d2r) antagonist, improves motor performance and shows neuroprot..

    产品型号:T7352 原产地:中国大陆价格: ¥0.0

  • TP-030-1;化合物 TP-030-1TP-030-1

    产品名称: TP-030-1;化合物 TP-030-1TP-030-1

    产品简介:tp-030-1, an inhibitor of ripk1, exhibits potent activity against hripk1 (human ripk1) with a ki value of 3.9 nm and against mripk1 (mouse ripk1) with an ic50 v..

    产品型号:T73374 原产地:中国大陆价格: ¥0.0

  • IGUANA-1;化合物 IGUANA-1IGUANA-1

    产品名称: IGUANA-1;化合物 IGUANA-1IGUANA-1

    产品简介:iguana-1, a potent aldh1b1 inhibitor, effectively targets this mitochondrial enzyme involved in promoting colorectal and pancreatic cancer. it exhibits signific..

    产品型号:T73377 原产地:中国大陆价格: ¥0.0

  • TMV-IN-1;化合物 TMV-IN-1TMV-IN-1

    产品名称: TMV-IN-1;化合物 TMV-IN-1TMV-IN-1

    产品简介:tmv-in-1, a chalcone derivative, serves as an inhibitor of the tobacco mosaic virus (tmv), demonstrating effective therapeutic and protective activities, with e..

    产品型号:T73379 原产地:中国大陆价格: ¥0.0

  • Angiotensin (1-7);化合物Angiotensin 1-7Ang-(1-7)|||Angiotensin 1-7|||ASP-ARG-VAL-TYR-ILE-HIS-PRO;Ang-(1

    产品名称: Angiotensin (1-7);化合物Angiotensin 1-7Ang-(1-7)|||Angiotensin 1-7|||ASP-ARG-VAL-TYR-ILE-HIS-PRO;Ang-(1

    产品简介:angiotensin (1-7) (asp-arg-val-tyr-ile-his-pro) is a synthetic heptapeptide identical to endogenous angiotensin-(1-7) , inhibits purified canine ace activity (i..

    产品型号:T7339 原产地:中国大陆价格: ¥0.0

  • Cadein1;化合物 Cadein1Cadein1

    产品名称: Cadein1;化合物 Cadein1Cadein1

    产品简介:cadein1, an isoquinolinium derivative, induces g2/m phase delay and caspase-dependent apoptosis in cancer cells lacking functional p53...

    产品型号:T73413 原产地:中国大陆价格: ¥0.0

  • Con B-1;化合物 Con B-1Con B-1

    产品名称: Con B-1;化合物 Con B-1Con B-1

    产品简介:conb-1 is a potent and selective alk inhibitor with low toxicity to normal cells [1] ...

    产品型号:T73417 原产地:中国大陆价格: ¥0.0

  • AK-IN-1;化合物 AK-IN-1AK-IN-1

    产品名称: AK-IN-1;化合物 AK-IN-1AK-IN-1

    产品简介:ak-in-1, a competitive inhibitor for adenosine (ado) but not for atp, demonstrates significant inhibition of ak activity, achieving 86%, 87%, and 89% at concent..

    产品型号:T73436 原产地:中国大陆价格: ¥0.0

  • iBRD4-BD1;化合物 iBRD4-BD1iBRD4-BD1

    产品名称: iBRD4-BD1;化合物 iBRD4-BD1iBRD4-BD1

    产品简介:ibrd4-bd1 is a selective inhibitor of the brd4 bromodomain, exhibiting inhibition activity with an ic50 value of 12 nm. it is utilized in the research of inflam..

    产品型号:T73296 原产地:中国大陆价格: ¥0.0

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