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产品名称: SB 242084;化合物SB 242084 dihydrochloride hydrateSB 242084 dihydrochloride hydrate;6 - 氯-2,3 - 二氢- 5 -甲
产品简介:sb 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5ht2c receptor...产品型号:T7277 原产地:中国大陆价格: ¥0.0
产品名称: p53 Activator 7;MDM-2/p53 激活剂7p53 Activator 7
产品简介:p53 activator 7 is a highly potent and cell-permeable activator of the p53 mutation y220c (mdm-2/p53), which induces apoptosis...产品型号:T72771 原产地:中国大陆价格: ¥0.0
产品名称: GPR81 agonist 2;化合物 GPR81 agonist 2GPR81 agonist 2
产品简介:gpr81 agonist 2 is a potent agonist targeting the gpr81 receptor, demonstrating ec50 values of 0.023 ?m for hgpr81 and 0.123 ?m for hgpr109a, respectively...产品型号:T72772 原产地:中国大陆价格: ¥0.0
产品名称: NR2F1 agonist 1;化合物 NR2F1 agonist 1NR2F1 agonist 1
产品简介:nr2f1 agonist 1, a specific nuclear receptor nr2f1 activator, initiates dormancy programs in cancer cells by upregulating nr2f1 and its target genes controlling..产品型号:T72776 原产地:中国大陆价格: ¥0.0
产品名称: Keap1-Nrf2-IN-11;化合物 Keap1-Nrf2-IN-11Keap1-Nrf2-IN-11
产品简介:keap1-nrf2-in-11 (compound 6k), a potent keap1-nrf2 inhibitor, exhibits a dissociation constant (kd) of 0.21 nm. it hampers the production of reactive oxygen sp..产品型号:T72687 原产地:中国大陆价格: ¥0.0
产品名称: PKM2 activator 4;化合物 PKM2 activator 4PKM2 activator 4
产品简介:pkm2 activator 4, a chemical compound, functions as an activator of pkm2 with an activation concentration (ac 50) ranging from 1 to 10 μm. it is primarily utili..产品型号:T72692 原产地:中国大陆价格: ¥0.0
产品名称: PKM2 activator 5;PKM2 激活剂5PKM2 activator 5
产品简介:pkm2 activator 5 is a novel and potent pkm2 activator (ac50: 0.316 ?m) with potential anticancer activity for the study of cancer metabolism-related diseases...产品型号:T72693 原产地:中国大陆价格: ¥0.0
产品名称: UCK2 Inhibitor-1;化合物 UCK2 Inhibitor-1UCK2 Inhibitor-1
产品简介:uck2 inhibitor-1 is a non-competitive uck2 inhibitor with an ic 50 of 4.7 ?m [1] ...产品型号:T72695 原产地:中国大陆价格: ¥0.0
产品名称: UCK2 Inhibitor-3;化合物 UCK2 Inhibitor-3UCK2 Inhibitor-3
产品简介:uck2 inhibitor-3 is a non-competitive inhibitor targeting uridine-cytidine kinase 2 (uck2), a key enzyme in the pyrimidine salvage pathway, with an ic50 value o..产品型号:T72696 原产地:中国大陆价格: ¥0.0
产品名称: Nrf2 activator-6;化合物 Nrf2 activator-6Nrf2 activator-6
产品简介:nrf2 activator-6, a tetrahydroisoquinoline compound, functions as an nrf2 activator, demonstrating potency with an ic50 value of 5 nm in inhibiting the kelch do..产品型号:T72697 原产地:中国大陆价格: ¥0.0
产品名称: Cavα2δ1&NET-IN-1;化合物 Cavα2δ1&NET-IN-1Cavα2δ1&NET-IN-1
产品简介:cavα2δ1&net-in-1 . cavα2δ1&net-in-1 inhibits ca v α2δ-1 with a k i of 112 nm. cavα2δ1&net-in-1 inhibits net with a k i of 383 nm and ic 50 of 67 nm. cavα2δ1&net..产品型号:T72699 原产地:中国大陆价格: ¥0.0
产品名称: Cavα2δ1&NET-IN-2;化合物 Cavα2δ1&NET-IN-2Cavα2δ1&NET-IN-2
产品简介:cavα2δ1&net-in-2 . cavα2δ1&net-in-2 inhibits ca v α2δ-1 with a k i of 454 nm. cavα2δ1&net-in-2 inhibits net with a k i of 59 nm and ic 50 of 7 nm. cavα2δ1&net-i..产品型号:T72700 原产地:中国大陆价格: ¥0.0
产品名称: Cavα2δ1&NET-IN-3;化合物 Cavα2δ1&NET-IN-3Cavα2δ1&NET-IN-3
产品简介:cavα2δ1&net-in-3 (example 216) is an inhibitor targeting both the α2δ subunit of voltage-gated calcium channels (vgcc) and the noradrenaline transporter (net). ..产品型号:T72701 原产地:中国大陆价格: ¥0.0
产品名称: Keap1-Nrf2-IN-13;化合物 Keap1-Nrf2-IN-13Keap1-Nrf2-IN-13
产品简介:keap1-nrf2-in-13 is a potent inhibitor of the keap1-nrf2 protein-protein interaction (ppi), exhibiting an ic50 value of 0.15 μm, indicative of its high efficacy..产品型号:T72706 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/VEGFR2-IN-1;化合物 PI3K/VEGFR2-IN-1PI3K/VEGFR2-IN-1
产品简介:pi3k/vegfr2-in-1 is a potent dual inhibitor targeting both pi3k and vegfr2 with ic50 values of 2.21 μm for pi3k and 68 μm for vegfr2, respectively. this compoun..产品型号:T72713 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2-IN-36;化合物 SARS-CoV-2-IN-36SARS-CoV-2-IN-36
产品简介:sars-cov-2-in-36 is a potent inhibitor of sars-cov-2 mpro (sars-cov), demonstrating an ic50 of 2.37 μm and a kd of 1.19 μm in enzymatic assays. this compound ex..产品型号:T72718 原产地:中国大陆价格: ¥0.0
产品名称: Tubulin/MMP-IN-2;化合物 Tubulin/MMP-IN-2Tubulin/MMP-IN-2
产品简介:tubulin/mmp-in-2, a dual inhibitor of tubulin and matrix metalloproteinases (mmps), effectively inhibits tubulin polymerization and induces cell apoptosis. it d..产品型号:T72719 原产地:中国大陆价格: ¥0.0
产品名称: 2,3,5-TRIFLUORO-4-(TRIFLUOROMETHYL)PYRIDINE;化合物 T72722,3,5-TRIFLUORO-4-(TRIFLUOROMETHYL)PYRIDINE
产品简介:2,3,5-trifluoro-4-(trifluoromethyl)pyridine is a useful organic compound for research related to life sciences. the catalog number is t7272 and the cas number i..产品型号:T7272 原产地:中国大陆价格: ¥0.0
产品名称: P-gp inhibitor 2;化合物 P-gp inhibitor 2P-gp inhibitor 2
产品简介:p-gp inhibitor 2 is a powerful p-glycoprotein (p-gp) inhibitor, effective in reversing doxorubicin resistance with an ic50 of 0.22 ?m in human colorectal carcin..产品型号:T72739 原产地:中国大陆价格: ¥0.0
产品名称: (R)-eIF4A3-IN-2;化合物 (R)-eIF4A3-IN-2(R)-eIF4A3-IN-2
产品简介:(r)-eif4a3-in-2, a less active enantiomer of eif4a3-in-2, is a highly selective and noncompetitive inhibitor of the eukaryotic initiation factor 4a-3 (eif4a3) w..产品型号:T72746 原产地:中国大陆价格: ¥0.0