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产品名称: 3,3-Dimethyl-1-butanol;化合物 3,3-Dimethyl-1-butanolNeohexanol|||DMB|||DMB ; Neohexanol;Neohexanol|||D
产品简介:3,3-dimethyl-1-butanol (dmb) is an orally active compound that inhibits trimethylamine (tma) and trimethylamine n-oxide (tmao), along with the signaling pathway..产品型号:T72383 原产地:中国大陆价格: ¥0.0
产品名称: CB1 inverse agonist 2;化合物 CB1 inverse agonist 2CB1 inverse agonist 2
产品简介:cb1 inverse agonist 2, an orally active compound, serves as an inverse agonist for the cannabinoid receptor cb1. it effectively counteracts the hypothermia and ..产品型号:T72395 原产地:中国大陆价格: ¥0.0
产品名称: LIMK1 inhibitor BMS-4;化合物 LIMK1 inhibitor BMS-4LIMK1 inhibitor BMS-4
产品简介:limk1 inhibitor bms-4 is a compound targeting lim kinase (limk) 1/2, specifically inhibiting the phosphorylation of its substrate, cofilin, but it remains noncy..产品型号:T72399 原产地:中国大陆价格: ¥0.0
产品名称: Ferroptosis inducer-1;化合物 Ferroptosis inducer-1Ferroptosis inducer-1
产品简介:ferroptosis inducer-1 is a ferroptosis inducer with antitumor potential [1] ...产品型号:T72403 原产地:中国大陆价格: ¥0.0
产品名称: Tofacitinib Prodrug-1;化合物 Tofacitinib Prodrug-1Tofacitinib Prodrug-1
产品简介:tofacitinib prodrug-1 is an effective and oral active prodrug to mitigate the systemic adverse effects of tofacitinib. tofacitinib prodrug-1 can effectively att..产品型号:T72406 原产地:中国大陆价格: ¥0.0
产品名称: c-Met/MEK1/Flt-3-IN-1;化合物 c-Met/MEK1/Flt-3-IN-1c-Met/MEK1/Flt-3-IN-1
产品简介:antiproliferative against-3 (comp 33) demonstrates significant activity against hela (ic 50 = 0.21 ?m), a549 (ic 50 = 0.39 ?m), and mcf-7 (ic 50 = 0.33 ?m) cell..产品型号:T72407 原产地:中国大陆价格: ¥0.0
产品名称: Sortilin antagonist 1;化合物 Sortilin antagonist 1Sortilin antagonist 1
产品简介:sortilin antagonist 1, a potent sortilin antagonist, exhibits an inhibition constant (ic50) of 20 nm against neurotensin (nts) binding to sortilin. neurotensin ..产品型号:T72410 原产地:中国大陆价格: ¥0.0
产品名称: AChE/Nrf2 modulator 1;化合物 AChE/Nrf2 modulator 1AChE/Nrf2 modulator 1
产品简介:ache/nrf2 modulator 1, an orally active compound, serves as a modulator of acetylcholinesterase (ache) and nuclear factor erythroid 2-related factor 2 (nrf2). i..产品型号:T72417 原产地:中国大陆价格: ¥0.0
产品名称: MTK458;化合物 MTK458Mitophagy activator 1|||EP-0035985;Mitophagy activator 1|||EP-0035985
产品简介:mtk458 (ep-0035985) is an orally active and brain-permeable pink1 activator that promotes pathological clearance of alpha-synuclein and reduces pub in a pff ino..产品型号:T72420 原产地:中国大陆价格: ¥0.0
产品名称: LRRK2/NUAK1/TYK2-IN-1;化合物 LRRK2/NUAK1/TYK2-IN-1LRRK2/NUAK1/TYK2-IN-1
产品简介:lrrk2/nuak1/tyk2-in-1 (compound 226) exhibits inhibitory activity against lrrk2 (wt), lrrk2 (g2019), tyk2, and nuak1, demonstrating ic50 values below 10 nm. thi..产品型号:T72421 原产地:中国大陆价格: ¥0.0
产品名称: Endomorphin 1 acetate;化合物 Endomorphin 1 acetateEndomorphin 1 acetate
产品简介:endomorphin-1 acetate is a highly selective and high-affinity μ-opioid receptor agonist (k i: 1.11 nm) that also demonstrates moderate affinity for kappa 3 bind..产品型号:T72423 原产地:中国大陆价格: ¥0.0
产品名称: H1k;化合物H1kH1k
产品简介:h1k is an eudistomin y fluorescent derivative and lysosome-targeted antiproliferative agent that dose-dependently increases autophagy signalling and down-regula..产品型号:T72057 原产地:中国大陆价格: ¥0.0
产品名称: S1R agonist 2;化合物S1R agonist 2S1R agonist 2
产品简介:s1r agonist 2 is a selective s1r agonist with a ki of 88 nm for s2r and 1.1 nm for s1r and is protective against ros and nmda-induced neurotoxicity...产品型号:T72059 原产地:中国大陆价格: ¥0.0
产品名称: Myosin V-IN-1;化合物Myosin V-IN-1Myosin V-IN-1
产品简介:myosin v-in-1 is a potent and selective inhibitor of myosin v with a ki value of 6 μm.myosin v-in-1 inhibits actin v and slows down actin-activated myosin v atp..产品型号:T72060 原产地:中国大陆价格: ¥0.0
产品名称: PDCD4-IN-1;化合物PDCD4-IN-1PDCD4-IN-1
产品简介:pdcd4-in-1, a pdcd4 inhibitor (kd : 350 nm), promotes bdnf expression in hippocampal neuronal cells ht-22...产品型号:T72063 原产地:中国大陆价格: ¥0.0
产品名称: TASK-1-IN-1;化合物TASK-1-IN-1TASK-1-IN-1
产品简介:task-1-in-1 is a potent and selective inhibitor of task-1 (potassium channel) (ic50: 148 nm).task-1-in-1 has a reduced inhibitory effect on the task-3 channel w..产品型号:T72064 原产地:中国大陆价格: ¥0.0
产品名称: CpCDPK1/TgCDPK1-IN-2;化合物CpCDPK1/TgCDPK1-IN-2CpCDPK1/TgCDPK1-IN-2
产品简介:cpcdpk1/tgcdpk1-in-2 is a dual inhibitor of cpcdpk1 and tgcdpk1 with ic50 values of 12 and 5 nm for cpcdpk1 and tgcdpk1, respectively.cpcdpk1/tgcdpk1-in-2 can b..产品型号:T72081 原产地:中国大陆价格: ¥0.0
产品名称: ADRA1D receptor antagonist 1 free base;化合物 ADRA1D receptor antagonist 1 free baseADRA1D receptor ant
产品简介:adra1d receptor antagonist 1 (free base) antagonist ( k i =1.6 nm). adra1d receptor antagonist 1 (free base) dose-dependently inhibits bladder contraction with..产品型号:T72091 原产地:中国大陆价格: ¥0.0
产品名称: Eleven-Nineteen-Leukemia Protein IN-1;化合物 Eleven-Nineteen-Leukemia Protein IN-1Eleven-Nineteen-Leuke
产品简介:eleven-nineteen-leukemia protein in-1 is a potent inhibitor of the enl yeats domain, exhibiting an ic50 of 14.5 nm. it binds to the enl protein, consequently in..产品型号:T72096 原产地:中国大陆价格: ¥0.0
产品名称: DYRKs-IN-1 hydrochloride;化合物 DYRKs-IN-1 hydrochlorideDYRKs-IN-1 hydrochloride
产品简介:dyrks-in-1 hydrochloride is a potent inhibitor of dual-specificity tyrosine-phosphorylation-regulated kinases (dyrks), exhibiting ic50 values of 5 nm and 8 nm f..产品型号:T72242 原产地:中国大陆价格: ¥0.0